GT200500381A - DERIVATIVE OF QUINOLINA, ITS USE, PREPARATION AND MEDICINAL PRODUCT CONTAINING IT - Google Patents
DERIVATIVE OF QUINOLINA, ITS USE, PREPARATION AND MEDICINAL PRODUCT CONTAINING ITInfo
- Publication number
- GT200500381A GT200500381A GT200500381A GT200500381A GT200500381A GT 200500381 A GT200500381 A GT 200500381A GT 200500381 A GT200500381 A GT 200500381A GT 200500381 A GT200500381 A GT 200500381A GT 200500381 A GT200500381 A GT 200500381A
- Authority
- GT
- Guatemala
- Prior art keywords
- preparation
- derivative
- quinolina
- product containing
- medicinal product
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/64—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Abstract
LA PRESENTE INVENCION SE REFIERE A UN DERIVADO DE QUINOLINA DE LA FORMULA GENERAL A EN LA QUE R1, R2, R3, X, Y, Z Y A SE INDICAN EN LA DESCRIPCION Y EN LAS REIVINDICACIONES, AL USO Y PREPARACIÓN DE LOS COMPUESTOS LA FORMULA GENERAL A PARA EL TRATAMIENTO DE DIVERSAS ENFERMEDADES.THIS INVENTION REFERS TO A QUINOLINE DERIVATIVE OF THE GENERAL FORM A IN WHICH R1, R2, R3, X, Y, ZYA ARE INDICATED IN THE DESCRIPTION AND IN THE CLAIMS, THE USE AND PREPARATION OF THE COMPOUNDS THE GENERAL FORMULA A FOR THE TREATMENT OF DIFFERENT DISEASES.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE102004063223A DE102004063223A1 (en) | 2004-12-22 | 2004-12-22 | New quinoline derivatives are ephrin receptor kinase inhibitors useful for the treatment of e.g. blood vessels diseases, hyperproliferations, chronic or acute neurodegenerative diseases, psoriasis, eczema and scleroderma |
Publications (1)
Publication Number | Publication Date |
---|---|
GT200500381A true GT200500381A (en) | 2006-08-03 |
Family
ID=36599298
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GT200500381A GT200500381A (en) | 2004-12-22 | 2005-12-21 | DERIVATIVE OF QUINOLINA, ITS USE, PREPARATION AND MEDICINAL PRODUCT CONTAINING IT |
Country Status (7)
Country | Link |
---|---|
CN (1) | CN101087788A (en) |
AR (1) | AR052544A1 (en) |
DE (1) | DE102004063223A1 (en) |
GT (1) | GT200500381A (en) |
PA (1) | PA8657701A1 (en) |
SV (1) | SV2007002357A (en) |
UY (1) | UY29308A1 (en) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN103382206B (en) * | 2012-05-04 | 2016-09-28 | 上海恒瑞医药有限公司 | Quinoline or quinazoline derivative, its preparation method and in application pharmaceutically |
CN106565823B (en) * | 2016-11-10 | 2020-09-11 | 珠海诺贝尔国际生物医药研究院有限公司 | Eph receptor small molecule inhibitor and preparation method thereof |
CN110577546B (en) * | 2018-06-08 | 2021-09-07 | 江苏威凯尔医药科技有限公司 | VEGFR inhibitor and preparation method and application thereof |
WO2019233458A1 (en) * | 2018-06-08 | 2019-12-12 | 江苏威凯尔医药科技有限公司 | Vegfr inhibitor, preparation method therefor and use thereof |
CN113150009B (en) * | 2020-01-07 | 2023-05-23 | 爱科诺生物医药(香港)有限公司 | Heterocyclic compound with activity of inhibiting programmed cell necrosis pathway and application thereof |
CN113061142A (en) * | 2020-01-02 | 2021-07-02 | 爱科诺生物医药股份有限公司 | Heterocyclic compounds with programmed cell necrosis pathway inhibition activity and application thereof |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3919238A (en) * | 1973-06-06 | 1975-11-11 | Morton Norwich Products Inc | 9-(Substituted amino)imidazo(4,5-f) quinolines |
CA1263378A (en) * | 1985-01-08 | 1989-11-28 | Robert James Alaimo | Imidazo¬4,5-f|quinolines useful as immunomodulating agents |
WO1993003030A1 (en) * | 1991-08-02 | 1993-02-18 | Pfizer Inc. | Quinoline derivatives as immunostimulants |
-
2004
- 2004-12-22 DE DE102004063223A patent/DE102004063223A1/en not_active Ceased
-
2005
- 2005-12-19 CN CNA2005800444603A patent/CN101087788A/en active Pending
- 2005-12-21 GT GT200500381A patent/GT200500381A/en unknown
- 2005-12-22 SV SV2005002357A patent/SV2007002357A/en not_active Application Discontinuation
- 2005-12-22 PA PA20058657701A patent/PA8657701A1/en unknown
- 2005-12-22 AR ARP050105485A patent/AR052544A1/en not_active Application Discontinuation
- 2005-12-22 UY UY29308A patent/UY29308A1/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
AR052544A1 (en) | 2007-03-21 |
SV2007002357A (en) | 2007-02-16 |
PA8657701A1 (en) | 2006-09-08 |
UY29308A1 (en) | 2006-06-30 |
DE102004063223A1 (en) | 2006-07-13 |
CN101087788A (en) | 2007-12-12 |
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