GT200300283A - HETEROAROMATIC GLUCOQUINASE ACTIVATORS OF SIX 5-SUBSTITUTED MEMBERS - Google Patents

HETEROAROMATIC GLUCOQUINASE ACTIVATORS OF SIX 5-SUBSTITUTED MEMBERS

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Publication number
GT200300283A
GT200300283A GT200300283A GT200300283A GT200300283A GT 200300283 A GT200300283 A GT 200300283A GT 200300283 A GT200300283 A GT 200300283A GT 200300283 A GT200300283 A GT 200300283A GT 200300283 A GT200300283 A GT 200300283A
Authority
GT
Guatemala
Prior art keywords
activators
glucoquinase
heteroaromatic
substituted members
compounds
Prior art date
Application number
GT200300283A
Other languages
Spanish (es)
Inventor
Shaoqing Chen
Wendy Lea Corbett
Kevin Richard Guertin
Nancy-Ellen Haynes
Robert Francis Kester
Francis A Mennona
Steven Gregory Mischke
Yimin Qian
Ramakanth Sarabu
Nathan Robert Scott
Kahitij Chhabilbhai Thakkar
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT200300283A publication Critical patent/GT200300283A/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

LA PRESENTE INVENCION SE REFIERE A COMPUESTOS DE LA FORMULA GENERAL I EN LA QUE R1,R2,R3,R4,Y, SON GRUPOS FUNCIONALES DESCRITOS EN EL EXPEDIENTE. ESTOS COMPUESTOS SON ACTIVADORES DE GLUCOQUINASA POR LO QUE SON DE UTILIDAD EN CUADROS DE DIABETES, PRINCIPALMENTE.THE PRESENT INVENTION REFERS TO COMPOUNDS OF GENERAL FORMULA I IN WHICH R1, R2, R3, R4, AND, ARE FUNCTIONAL GROUPS DESCRIBED IN THE RECORD. THESE COMPOUNDS ARE GLUCOKINASE ACTIVATORS, SO THEY ARE USEFUL IN PICTURES OF DIABETES, MAINLY.

GT200300283A 2002-12-12 2003-12-11 HETEROAROMATIC GLUCOQUINASE ACTIVATORS OF SIX 5-SUBSTITUTED MEMBERS GT200300283A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US43280602P 2002-12-12 2002-12-12

Publications (1)

Publication Number Publication Date
GT200300283A true GT200300283A (en) 2004-07-14

Family

ID=35925145

Family Applications (1)

Application Number Title Priority Date Filing Date
GT200300283A GT200300283A (en) 2002-12-12 2003-12-11 HETEROAROMATIC GLUCOQUINASE ACTIVATORS OF SIX 5-SUBSTITUTED MEMBERS

Country Status (3)

Country Link
CN (1) CN100469770C (en)
GT (1) GT200300283A (en)
ZA (1) ZA200504474B (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8258134B2 (en) * 2008-04-16 2012-09-04 Hoffmann-La Roche Inc. Pyridazinone glucokinase activators
EP2870138B1 (en) * 2012-07-06 2018-08-22 Genentech, Inc. N-substituted benzamides and methods of use thereof
EP3101005A1 (en) * 2015-06-05 2016-12-07 Lead Pharma Cel Models IP B.V. Ror gamma (rory) modulators
EP3101007A1 (en) * 2015-06-05 2016-12-07 Lead Pharma Cel Models IP B.V. Ror gamma (rory) modulators
CN106187838B (en) * 2016-07-13 2018-05-01 广东东阳光药业有限公司 Aryl alkynes compound and its preparation method and application

Also Published As

Publication number Publication date
CN100469770C (en) 2009-03-18
ZA200504474B (en) 2006-02-22
CN1726197A (en) 2006-01-25

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