GT199600072A - ZWITTERIONIC FORMS OF TROVAFLOXACIN. - Google Patents

ZWITTERIONIC FORMS OF TROVAFLOXACIN.

Info

Publication number
GT199600072A
GT199600072A GT199600072A GT199600072A GT199600072A GT 199600072 A GT199600072 A GT 199600072A GT 199600072 A GT199600072 A GT 199600072A GT 199600072 A GT199600072 A GT 199600072A GT 199600072 A GT199600072 A GT 199600072A
Authority
GT
Guatemala
Prior art keywords
trovafloxacin
refers
zwitterionic forms
procedures
naftiridone
Prior art date
Application number
GT199600072A
Other languages
Spanish (es)
Inventor
Douglas John Meldrum Allen
David Bruning Joseph
Timothy Norris
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT199600072A publication Critical patent/GT199600072A/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Abstract

ESTA INVENCION SE REFIERE A LA NAFTIRIDONA ANTIBIOTICA TROVAFLOXACINA. MAS CONCRETAMENTE SE REFIERE A LOS POLIMORFOS Y EL PENTAHIDRATO DE LA FORMA ZWITTERIONICA DEL MISMO QUE TIENE LA FORMULA I, Y LOS PROCEDIMIENTOS PARA SU PREPARACION. LA INVENCION SE REFIERE ADEMAS A LOS PROCEDIMIENTOS DE UTILIZACION, Y LAS COMPOSICIONES FARMACEUTICAS QUE LOS INCLUYEN, LOS COMPUESTOS DE LA INVENCION PARA EL TRATAMIENTO DE INFECCIONES BACTERIANAS EN MAMIFEROS.THIS INVENTION REFERS TO THE ANTIBIOTIC NAFTIRIDONE TROVAFLOXACIN. MORE CONCRETEALLY, IT REFERS TO THE POLYMORPHES AND PENTAHYDRATE OF THE ZWITTERIONIC FORM OF THE SAME AS FORMULA I, AND THE PROCEDURES FOR ITS PREPARATION. THE INVENTION FURTHER REFERS TO THE PROCEDURES FOR USE, AND THE PHARMACEUTICAL COMPOSITIONS INCLUDING THEM, THE COMPOUNDS OF THE INVENTION FOR THE TREATMENT OF BACTERIAL INFECTIONS IN MAMMALS.

GT199600072A 1995-08-29 1996-08-23 ZWITTERIONIC FORMS OF TROVAFLOXACIN. GT199600072A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US297595P 1995-08-29 1995-08-29

Publications (1)

Publication Number Publication Date
GT199600072A true GT199600072A (en) 1998-02-14

Family

ID=21703460

Family Applications (1)

Application Number Title Priority Date Filing Date
GT199600072A GT199600072A (en) 1995-08-29 1996-08-23 ZWITTERIONIC FORMS OF TROVAFLOXACIN.

Country Status (30)

Country Link
EP (1) EP0850060A1 (en)
JP (1) JP3188476B2 (en)
KR (1) KR100343909B1 (en)
CN (1) CN1190889A (en)
AP (1) AP636A (en)
AR (1) AR003985A1 (en)
AU (1) AU704115B2 (en)
BR (1) BR9609998A (en)
CA (1) CA2229786C (en)
CO (1) CO4480739A1 (en)
CZ (1) CZ56698A3 (en)
DZ (1) DZ2087A1 (en)
GT (1) GT199600072A (en)
HR (1) HRP960395B1 (en)
HU (1) HUP9900170A3 (en)
IL (1) IL122651A (en)
MA (1) MA23966A1 (en)
MY (1) MY113874A (en)
NO (1) NO309814B1 (en)
NZ (1) NZ312199A (en)
OA (1) OA10669A (en)
PE (1) PE12598A1 (en)
PL (1) PL325170A1 (en)
RU (1) RU2144921C1 (en)
SK (1) SK23898A3 (en)
TN (1) TNSN96109A1 (en)
TR (1) TR199800339T1 (en)
WO (1) WO1997007800A1 (en)
YU (1) YU48396A (en)
ZA (1) ZA967282B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HN1998000106A (en) 1997-08-01 1999-01-08 Pfizer Prod Inc PARENTERAL COMPOSITIONS OF ALATROFLAXACINO
US7019142B2 (en) 1998-01-16 2006-03-28 Pfizer Inc. Process for preparing naphthyridones and intermediates
PA8466701A1 (en) * 1998-01-21 2000-09-29 Pfizer Prod Inc TROVAFLOXACINO MESYLATE TABLET
US6114531A (en) * 1998-07-28 2000-09-05 Pfizer Inc. Process for preparing quinolone and naphthyridone carboxylic acids
HN1999000141A (en) * 1998-09-03 2000-06-19 Pfizer Prod Inc PROCEDURE FOR PREPARING SALTS OF TROVAFLOXACIN FOR ADDITION OF ACIDS.
US6239141B1 (en) 1999-06-04 2001-05-29 Pfizer Inc. Trovafloxacin oral suspensions

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5164402A (en) * 1989-08-16 1992-11-17 Pfizer Inc Azabicyclo quinolone and naphthyridinone carboxylic acids

Also Published As

Publication number Publication date
KR100343909B1 (en) 2003-04-10
IL122651A (en) 2000-02-17
YU48396A (en) 1998-12-23
PE12598A1 (en) 1998-03-20
RU2144921C1 (en) 2000-01-27
WO1997007800A1 (en) 1997-03-06
CA2229786C (en) 2002-02-19
AU6367696A (en) 1997-03-19
TNSN96109A1 (en) 2005-03-15
OA10669A (en) 2000-11-06
AU704115B2 (en) 1999-04-15
HUP9900170A3 (en) 1999-11-29
NO309814B1 (en) 2001-04-02
CN1190889A (en) 1998-08-19
NO980862L (en) 1998-02-27
TR199800339T1 (en) 1998-06-22
JP3188476B2 (en) 2001-07-16
MY113874A (en) 2002-06-29
NO980862D0 (en) 1998-02-27
AR003985A1 (en) 1998-09-30
CZ56698A3 (en) 1999-02-17
NZ312199A (en) 1999-06-29
PL325170A1 (en) 1998-07-06
CA2229786A1 (en) 1997-03-06
HUP9900170A2 (en) 1999-05-28
HRP960395B1 (en) 2001-12-31
DZ2087A1 (en) 2002-07-22
IL122651A0 (en) 1998-08-16
JPH10511692A (en) 1998-11-10
KR19990044232A (en) 1999-06-25
MX9801664A (en) 1998-08-30
HRP960395A2 (en) 1998-06-30
AP636A (en) 1998-04-09
AP9600853A0 (en) 1996-10-31
ZA967282B (en) 1998-03-02
BR9609998A (en) 1999-07-06
CO4480739A1 (en) 1997-07-09
EP0850060A1 (en) 1998-07-01
SK23898A3 (en) 1999-05-07
MA23966A1 (en) 1997-04-01

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