GB2105329B - Penem-3-carboxylic acid derivatives their preparation and their use as antimicrobial agents - Google Patents

Penem-3-carboxylic acid derivatives their preparation and their use as antimicrobial agents

Info

Publication number
GB2105329B
GB2105329B GB08224330A GB8224330A GB2105329B GB 2105329 B GB2105329 B GB 2105329B GB 08224330 A GB08224330 A GB 08224330A GB 8224330 A GB8224330 A GB 8224330A GB 2105329 B GB2105329 B GB 2105329B
Authority
GB
United Kingdom
Prior art keywords
penem
preparation
carboxylic acid
acid derivatives
antimicrobial agents
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB08224330A
Other languages
English (en)
Other versions
GB2105329A (en
Inventor
Tetsuo Miyadera
Isao Kawamoto
Yukio Sugimura
Toshihiko Hashimoto
Shinichi Sugawara
Teruo Tanaka
Kimio Iino
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sankyo Co Ltd
Original Assignee
Sankyo Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankyo Co Ltd filed Critical Sankyo Co Ltd
Publication of GB2105329A publication Critical patent/GB2105329A/en
Application granted granted Critical
Publication of GB2105329B publication Critical patent/GB2105329B/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
GB08224330A 1981-08-25 1982-08-25 Penem-3-carboxylic acid derivatives their preparation and their use as antimicrobial agents Expired GB2105329B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP56133203A JPS5835190A (ja) 1981-08-25 1981-08-25 ペネム−３−カルボン酸誘導体

Publications (2)

Publication Number Publication Date
GB2105329A GB2105329A (en) 1983-03-23
GB2105329B true GB2105329B (en) 1985-05-30

Family

ID=15099135

Family Applications (1)

Application Number Title Priority Date Filing Date
GB08224330A Expired GB2105329B (en) 1981-08-25 1982-08-25 Penem-3-carboxylic acid derivatives their preparation and their use as antimicrobial agents

Country Status (6)

Country Link
JP (1) JPS5835190A (pt)
CH (1) CH654308A5 (pt)
DE (1) DE3231596A1 (pt)
FR (1) FR2512027A1 (pt)
GB (1) GB2105329B (pt)
IT (1) IT1156494B (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5921692A (ja) * 1982-07-29 1984-02-03 Sankyo Co Ltd 経口ペネム化合物及びその製法
EP0345827A1 (en) * 1982-11-29 1989-12-13 Schering Corporation Process for the production of penem compounds
US4791198A (en) * 1984-07-05 1988-12-13 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha Beta-lactam compound and preparation thereof
US4861877A (en) * 1984-07-05 1989-08-29 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha Process for preparing 4-acetoxy-3-hydroxyethylazetidin-2-one derivatives
US5416208A (en) * 1989-07-05 1995-05-16 Farmitalia Carlo Erba S R L Process for penems
GB8915392D0 (en) * 1989-07-05 1989-08-23 Erba Carlo Spa Process for penems

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LU77306A1 (pt) * 1977-05-09 1979-01-18
US4168314A (en) * 1977-11-17 1979-09-18 Merck & Co., Inc. 6-(1'-Hydroxyethyl)-2-aminoethylthio-pen-2-em-3-carboxylic acid
EP0042026B1 (de) * 1978-02-02 1986-01-08 Ciba-Geigy Ag 3,4-Disubstituierte Azetidin-2-onverbindungen und Verfahren zu ihrer Herstellung
JPS55153789A (en) * 1979-04-11 1980-11-29 Sankyo Co Ltd Penem-3-carboxylic acid derivative and its preparation
CA1212105A (en) * 1980-04-30 1986-09-30 Shoji Ikeda Ampicillin esters and production thereof
JPS572290A (en) * 1980-06-03 1982-01-07 Sankyo Co Ltd Production of penem-3-carboxylic derivative
US4411906A (en) * 1981-11-25 1983-10-25 Schering Corporation (5R,6S,8R)-6-(1-Hydroxyethyl)-2-(2-fluoroethylthio)-penem-3-carboxylates

Also Published As

Publication number Publication date
CH654308A5 (de) 1986-02-14
JPS6324515B2 (pt) 1988-05-20
FR2512027B1 (pt) 1984-12-14
IT1156494B (it) 1987-02-04
GB2105329A (en) 1983-03-23
IT8268039A0 (it) 1982-08-25
FR2512027A1 (fr) 1983-03-04
JPS5835190A (ja) 1983-03-01
DE3231596C2 (pt) 1989-03-09
DE3231596A1 (de) 1983-03-10

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Legal Events

Date Code Title Description
PCNP Patent ceased through non-payment of renewal fee

Effective date: 19970825