GB1567341A - Somatostatin analogues with dissociated biological activities - Google Patents

Somatostatin analogues with dissociated biological activities Download PDF

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Publication number
GB1567341A
GB1567341A GB23695/77A GB2369577A GB1567341A GB 1567341 A GB1567341 A GB 1567341A GB 23695/77 A GB23695/77 A GB 23695/77A GB 2369577 A GB2369577 A GB 2369577A GB 1567341 A GB1567341 A GB 1567341A
Authority
GB
United Kingdom
Prior art keywords
peptide
cys
accordance
ser
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB23695/77A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Salk Institute for Biological Studies
Original Assignee
Salk Institute for Biological Studies
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/785,533 external-priority patent/US4133782A/en
Application filed by Salk Institute for Biological Studies filed Critical Salk Institute for Biological Studies
Publication of GB1567341A publication Critical patent/GB1567341A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/655—Somatostatins
    • C07K14/6555—Somatostatins at least 1 amino acid in D-form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Endocrinology (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Zoology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Toxicology (AREA)
  • Engineering & Computer Science (AREA)
  • Biophysics (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
GB23695/77A 1976-06-07 1977-06-03 Somatostatin analogues with dissociated biological activities Expired GB1567341A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US69328276A 1976-06-07 1976-06-07
US05/785,533 US4133782A (en) 1976-06-07 1977-04-07 Somatostatin analogs with dissociated biological activities

Publications (1)

Publication Number Publication Date
GB1567341A true GB1567341A (en) 1980-05-14

Family

ID=27105142

Family Applications (1)

Application Number Title Priority Date Filing Date
GB23695/77A Expired GB1567341A (en) 1976-06-07 1977-06-03 Somatostatin analogues with dissociated biological activities

Country Status (11)

Country Link
JP (1) JPS52156885A (sv)
AU (1) AU509631B2 (sv)
CA (1) CA1102313A (sv)
CH (1) CH640827A5 (sv)
DE (1) DE2725735A1 (sv)
DK (1) DK250977A (sv)
FR (1) FR2375190A1 (sv)
GB (1) GB1567341A (sv)
IL (1) IL52231A (sv)
NL (1) NL7706002A (sv)
SE (1) SE441452B (sv)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3904594A (en) * 1973-07-02 1975-09-09 Salk Inst For Biological Studi Somatostatin and acylated des-(ala' 1', gly' 2') derivatives thereof
US3842067A (en) * 1973-07-27 1974-10-15 American Home Prod Synthesis of(des-asn5)-srif and intermediates

Also Published As

Publication number Publication date
NL7706002A (nl) 1977-12-09
FR2375190A1 (fr) 1978-07-21
AU2577577A (en) 1978-12-07
CA1102313A (en) 1981-06-02
JPS52156885A (en) 1977-12-27
DE2725735A1 (de) 1977-12-15
IL52231A (en) 1980-05-30
FR2375190B1 (sv) 1981-10-30
SE441452B (sv) 1985-10-07
DK250977A (da) 1977-12-08
CH640827A5 (en) 1984-01-31
AU509631B2 (en) 1980-05-22
IL52231A0 (en) 1977-08-31
SE7706567L (sv) 1977-12-08
JPS6315280B2 (sv) 1988-04-04

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Legal Events

Date Code Title Description
PS Patent sealed [section 19, patents act 1949]
PCNP Patent ceased through non-payment of renewal fee