GB1421006A - Imidazolidine derivatives - Google Patents
Imidazolidine derivativesInfo
- Publication number
- GB1421006A GB1421006A GB1006173A GB1006173A GB1421006A GB 1421006 A GB1421006 A GB 1421006A GB 1006173 A GB1006173 A GB 1006173A GB 1006173 A GB1006173 A GB 1006173A GB 1421006 A GB1421006 A GB 1421006A
- Authority
- GB
- United Kingdom
- Prior art keywords
- alkyl
- acid addition
- compounds
- march
- quaternary ammonium
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
1421006 Fused imidazolidines AKZO NV 1 March 1973 [7 March 1972] 10061/73 Heading C2C Compounds of the general formula (R 1,2 =H, OH, halogen, CF 3 , C 1-6 alkyl or alkoxy, C 1-8 acyloxy; R 3 =H, C 1-6 alkyl, C 7-10 aralkyl; X = O, S, NR 4 ; R 4 = H, C 1-6 alkyl) and their acid addition salts and quaternary ammonium compounds are prepared by reacting a compound of the formula or acid addition salt thereof with Y = CZ 1 Z 2 (Y = H 2 , O, S; Z 1,2 =leaving atom or group or Z 1+2 =reactive atom or group) followed by reduction when Y=O or S, and optionally followed by conversion to an acid addition salt or quaternary ammonium compound. The product or intermediate may be resolved, or an optically active starting material used. The above compounds are antidepressants, and may be administered in the form of pharmaceutical preparations containing them in association with a carrier.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
NL7202963A NL7202963A (en) | 1972-03-07 | 1972-03-07 |
Publications (1)
Publication Number | Publication Date |
---|---|
GB1421006A true GB1421006A (en) | 1976-01-14 |
Family
ID=19815531
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GB1006173A Expired GB1421006A (en) | 1972-03-07 | 1973-03-01 | Imidazolidine derivatives |
Country Status (16)
Country | Link |
---|---|
US (1) | US3860606A (en) |
JP (1) | JPS4899198A (en) |
AR (3) | AR202388A1 (en) |
AT (1) | AT326667B (en) |
AU (1) | AU471800B2 (en) |
BE (1) | BE796341A (en) |
CA (1) | CA1010032A (en) |
CH (1) | CH589083A5 (en) |
DE (1) | DE2311019A1 (en) |
ES (1) | ES412372A1 (en) |
FR (1) | FR2181796B1 (en) |
GB (1) | GB1421006A (en) |
HU (1) | HU166348B (en) |
IE (1) | IE37322B1 (en) |
NL (1) | NL7202963A (en) |
ZA (1) | ZA731086B (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1984002704A3 (en) * | 1982-12-30 | 1984-08-02 | Beecham Group Plc | Tetracyclic compounds |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NL178593C (en) * | 1974-01-31 | 1986-04-16 | Akzo Nv | PROCESS FOR PREPARING A PHARMACEUTICAL PREPARATION BASED ON A TETRACYCLIC COMPOUND AND METHOD FOR PREPARING THE TETRACYCLIC COMPOUNDS TO BE USED THEREOF |
NL7414038A (en) * | 1974-10-28 | 1976-05-03 | Akzo Nv | NEW TETRACYCLIC PYRROLIDINO DERIVATIVES. |
NL189199C (en) * | 1975-04-05 | 1993-02-01 | Akzo Nv | PROCESS FOR THE PREPARATION OF PHARMACEUTICAL PREPARATIONS WITH ACTION ON THE CENTRAL NERVOUS SYSTEM BASED ON BENZ (ARYL) AZEPINE DERIVATIVES, THE PHARMACEUTICAL PREPARATIONS OBTAINED, AND METHOD FOR PREPARING THE PRODUCT TO BE USED. |
DE3008944A1 (en) * | 1980-03-08 | 1981-09-24 | C.H. Boehringer Sohn, 6507 Ingelheim | DIBENZIMIDAZOAZEPINE, THEIR PRODUCTION AND USE |
DE3134672A1 (en) * | 1981-09-02 | 1983-03-17 | Boehringer Ingelheim KG, 6507 Ingelheim | HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE |
US4728735A (en) * | 1984-10-15 | 1988-03-01 | Merck & Co., Inc. | 10,11-dihydro-dibenzo-[b,f][1,4]-thiazepin derivatives |
HU195491B (en) * | 1985-12-20 | 1988-05-30 | Egyt Gyogyszervegyeszeti Gyar | Process for production of optically active 2-chlor-12-/3-/dimethil-amin/-2-methil-prophil/-12h-dibenzol /d,g/ /1,3,6/-diaxazocine and medical compositions containing such compounds |
US5478934A (en) * | 1994-11-23 | 1995-12-26 | Yuan; Jun | Certain 1-substituted aminomethyl imidazole and pyrrole derivatives: novel dopamine receptor subtype specific ligands |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3435042A (en) * | 1965-03-30 | 1969-03-25 | Colgate Palmolive Co | Novel morphanthridine derivatives |
-
1972
- 1972-03-07 NL NL7202963A patent/NL7202963A/xx unknown
-
1973
- 1973-02-15 ZA ZA731086A patent/ZA731086B/en unknown
- 1973-02-19 AU AU52303/73A patent/AU471800B2/en not_active Expired
- 1973-02-26 IE IE297/73A patent/IE37322B1/en unknown
- 1973-03-01 AR AR246878A patent/AR202388A1/en active
- 1973-03-01 GB GB1006173A patent/GB1421006A/en not_active Expired
- 1973-03-02 US US337323A patent/US3860606A/en not_active Expired - Lifetime
- 1973-03-06 ES ES412372A patent/ES412372A1/en not_active Expired
- 1973-03-06 CA CA165,357A patent/CA1010032A/en not_active Expired
- 1973-03-06 BE BE128428A patent/BE796341A/en unknown
- 1973-03-06 HU HUAO353A patent/HU166348B/hu unknown
- 1973-03-06 CH CH328773A patent/CH589083A5/xx not_active IP Right Cessation
- 1973-03-06 JP JP48026503A patent/JPS4899198A/ja active Pending
- 1973-03-06 DE DE19732311019 patent/DE2311019A1/en active Pending
- 1973-03-07 FR FR7308169A patent/FR2181796B1/fr not_active Expired
- 1973-03-07 AT AT203073A patent/AT326667B/en not_active IP Right Cessation
-
1974
- 1974-11-08 AR AR256461A patent/AR202429A1/en active
- 1974-11-08 AR AR256460A patent/AR203866A1/en active
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1984002704A3 (en) * | 1982-12-30 | 1984-08-02 | Beecham Group Plc | Tetracyclic compounds |
Also Published As
Publication number | Publication date |
---|---|
ATA203073A (en) | 1975-03-15 |
AR203866A1 (en) | 1975-10-31 |
ZA731086B (en) | 1973-11-28 |
BE796341A (en) | 1973-09-06 |
US3860606A (en) | 1975-01-14 |
IE37322L (en) | 1973-09-07 |
CA1010032A (en) | 1977-05-10 |
NL7202963A (en) | 1973-09-11 |
IE37322B1 (en) | 1977-06-22 |
CH589083A5 (en) | 1977-06-30 |
HU166348B (en) | 1975-03-28 |
FR2181796A1 (en) | 1973-12-07 |
FR2181796B1 (en) | 1976-10-22 |
AR202429A1 (en) | 1975-06-06 |
AU471800B2 (en) | 1976-05-06 |
AR202388A1 (en) | 1975-06-06 |
JPS4899198A (en) | 1973-12-15 |
ES412372A1 (en) | 1976-05-01 |
AU5230373A (en) | 1974-08-22 |
AT326667B (en) | 1975-12-29 |
DE2311019A1 (en) | 1973-09-20 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PS | Patent sealed [section 19, patents act 1949] | ||
PCNP | Patent ceased through non-payment of renewal fee |