GB1390485A - Pyrazoles - Google Patents
PyrazolesInfo
- Publication number
- GB1390485A GB1390485A GB2047573A GB2047573A GB1390485A GB 1390485 A GB1390485 A GB 1390485A GB 2047573 A GB2047573 A GB 2047573A GB 2047573 A GB2047573 A GB 2047573A GB 1390485 A GB1390485 A GB 1390485A
- Authority
- GB
- United Kingdom
- Prior art keywords
- alkyl
- pyrazoles
- alkoxy
- indolyl
- merck
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 150000003217 pyrazoles Chemical class 0.000 title abstract 3
- 125000000217 alkyl group Chemical group 0.000 abstract 4
- 125000003545 alkoxy group Chemical group 0.000 abstract 2
- 125000006273 (C1-C3) alkyl group Chemical group 0.000 abstract 1
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 1
- 239000000674 adrenergic antagonist Substances 0.000 abstract 1
- 125000000304 alkynyl group Chemical group 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 125000002768 hydroxyalkyl group Chemical group 0.000 abstract 1
- 125000001041 indolyl group Chemical group 0.000 abstract 1
- 239000000825 pharmaceutical preparation Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
- C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/28—Two oxygen or sulfur atoms
- C07D231/30—Two oxygen or sulfur atoms attached in positions 3 and 5
- C07D231/32—Oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CA141470A CA1001161A (en) | 1972-05-05 | 1972-05-05 | 5-(3-substituted amino-2-hydroxypropoxy)1,3-disubstituted pyrazoles and method of preparation |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1390485A true GB1390485A (en) | 1975-04-16 |
Family
ID=4093188
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB2047573A Expired GB1390485A (en) | 1972-05-05 | 1973-04-30 | Pyrazoles |
Country Status (14)
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2619164C2 (de) * | 1976-04-30 | 1985-07-11 | Boehringer Mannheim Gmbh, 6800 Mannheim | Indazolyl-(4)-oxy-propanolamine, Verfahren zu ihrer Herstellung und deren Verwendung |
| FI57617C (fi) * | 1979-01-18 | 1980-09-10 | Viljanmaa Antti | Spaennanordning foer skinn |
| DE2926517A1 (de) * | 1979-06-30 | 1981-01-15 | Beiersdorf Ag | Substituierte 3-aryl-pyrazole und 5-aryl-isoxazole und verfahren zu ihrer herstellung |
| US5547967A (en) * | 1993-12-08 | 1996-08-20 | Kali-Chemie Pharma Gmbh | (Phenylalkylaminoalkyloxy)-heteroaryl-compounds, processes and intermediates for their production and pharmaceutical compositions containing them |
| DE4341749A1 (de) * | 1993-12-08 | 1995-06-14 | Kali Chemie Pharma Gmbh | 3-(Phenylalkylaminoalkyloxy)-5-phenylpyrazol- Verbindungen sowie Verfahren und Zwischenprodukte zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel |
| CO5011072A1 (es) * | 1997-12-05 | 2001-02-28 | Lilly Co Eli | Etanolaminas pirazinil substituidas como agfonistas de los receptores |
| EP1036064A4 (en) * | 1997-12-05 | 2002-11-27 | Lilly Co Eli | SELECTIVE BETA 3-ADRENERGIC ANTAGONISTS |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1201061A (en) * | 1966-08-26 | 1970-08-05 | Endo Lab | Oxo pyrroles and process for preparing same |
| US3629433A (en) * | 1968-09-16 | 1971-12-21 | Ciba Geigy Corp | Antidepressant compositions of cycloalkano(c)pyrazole ethers |
| US3637738A (en) * | 1969-02-12 | 1972-01-25 | Ciba Geigy Corp | Cycloalkano(c)pyrazole ethers |
| US3726896A (en) * | 1970-05-06 | 1973-04-10 | Szabo Hnos Kessler & Cia | 1-benzyl-3(2,3-dihydroxypropoxy)indazole |
-
1972
- 1972-05-05 CA CA141470A patent/CA1001161A/en not_active Expired
-
1973
- 1973-04-16 SE SE7305383A patent/SE400076B/xx unknown
- 1973-04-18 NL NL7305477A patent/NL7305477A/xx not_active Application Discontinuation
- 1973-04-27 AU AU54937/73A patent/AU474793B2/en not_active Expired
- 1973-04-30 GB GB2047573A patent/GB1390485A/en not_active Expired
- 1973-05-01 JP JP48047644A patent/JPS4947367A/ja active Pending
- 1973-05-03 ES ES414320A patent/ES414320A1/es not_active Expired
- 1973-05-03 FR FR7315861A patent/FR2183751B1/fr not_active Expired
- 1973-05-03 DE DE2322313A patent/DE2322313A1/de not_active Ceased
- 1973-05-04 BE BE130745A patent/BE799098A/xx unknown
- 1973-05-04 ZA ZA733049A patent/ZA733049B/xx unknown
- 1973-05-04 CH CH636973A patent/CH582677A5/xx not_active IP Right Cessation
- 1973-05-04 HU HUME1624A patent/HU165583B/hu unknown
-
1974
- 1974-11-06 US US521416A patent/US3920691A/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| SE400076B (sv) | 1978-03-13 |
| ZA733049B (en) | 1974-12-24 |
| FR2183751B1 (US06653308-20031125-C00199.png) | 1976-10-22 |
| CH582677A5 (US06653308-20031125-C00199.png) | 1976-12-15 |
| NL7305477A (US06653308-20031125-C00199.png) | 1973-11-07 |
| AU5493773A (en) | 1974-10-31 |
| FR2183751A1 (US06653308-20031125-C00199.png) | 1973-12-21 |
| DE2322313A1 (de) | 1973-11-22 |
| CA1001161A (en) | 1976-12-07 |
| BE799098A (fr) | 1973-11-05 |
| US3920691A (en) | 1975-11-18 |
| JPS4947367A (US06653308-20031125-C00199.png) | 1974-05-08 |
| HU165583B (US06653308-20031125-C00199.png) | 1974-09-28 |
| AU474793B2 (en) | 1976-08-05 |
| ES414320A1 (es) | 1976-02-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed [section 19, patents act 1949] | ||
| PCNP | Patent ceased through non-payment of renewal fee |