GB1378381A - Imidazoles - Google Patents

Imidazoles

Info

Publication number
GB1378381A
GB1378381A GB3871671A GB3871671A GB1378381A GB 1378381 A GB1378381 A GB 1378381A GB 3871671 A GB3871671 A GB 3871671A GB 3871671 A GB3871671 A GB 3871671A GB 1378381 A GB1378381 A GB 1378381A
Authority
GB
United Kingdom
Prior art keywords
group
benzyloxyl
amino
hydrogen atom
imidazoles
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB3871671A
Inventor
J Heyes
N Ward
C J Rose
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Beecham Group PLC
Original Assignee
Beecham Group PLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beecham Group PLC filed Critical Beecham Group PLC
Priority to GB3871671A priority Critical patent/GB1378381A/en
Priority to IL38357A priority patent/IL38357A/en
Priority to SE7116177A priority patent/SE376418B/xx
Priority to JP47004138A priority patent/JPS4829771A/ja
Priority to ZA720038A priority patent/ZA7238B/en
Priority to FR7200104A priority patent/FR2149329B1/fr
Priority to NL7200080A priority patent/NL7200080A/xx
Priority to ES398587A priority patent/ES398587A1/en
Priority to BE777738A priority patent/BE777738A/en
Priority to CH13772A priority patent/CH584203A5/xx
Priority to DE19722200499 priority patent/DE2200499A1/en
Priority to US337062A priority patent/US3876655A/en
Publication of GB1378381A publication Critical patent/GB1378381A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Abstract

1378381 Imidazoles BEECHAM GROUP Ltd 13 July 1972 [18 Aug 1971] 38716/71 Heading C2C The invention comprises novel compounds (I) wherein R and R 1 are each a hydrogen or halogen atom or a methoxycarbonyl, ethoxycarbonyl, carboxamido, nitro, trifluoromethyl, C 1-4 alkyl, hydroxyl, methoxyl, ethoxyl, benzyloxyl, acetoxyl, amino, methylamino, ethylamino, dimethylamino or acetamido group; R 2 is an amino or C 1-4 alkoxyl or benzyloxyl group; R 3 is a hydrogen atom or a C 1-7 hydrocarbon group; and R 4 is a hydrogen atom or a methyl group; or a tautomer, acid addition salt or hydrate thereof. They are made by standard methods. Pharmaceutical preparations showing antiinflammatory action contain (I) as active ingredient; administration may be orally, parenterally or by suppository.
GB3871671A 1971-08-18 1971-08-18 Imidazoles Expired GB1378381A (en)

Priority Applications (12)

Application Number Priority Date Filing Date Title
GB3871671A GB1378381A (en) 1971-08-18 1971-08-18 Imidazoles
IL38357A IL38357A (en) 1971-08-18 1971-12-14 2-phenyl-4-acylamido-imidazole derivatives,their preparation and pharmaceutical compositions containing them
SE7116177A SE376418B (en) 1971-08-18 1971-12-16
JP47004138A JPS4829771A (en) 1971-08-18 1971-12-31
ZA720038A ZA7238B (en) 1971-08-18 1972-01-04 Anti-inflammatory acyl imidazoles
FR7200104A FR2149329B1 (en) 1971-08-18 1972-01-04
NL7200080A NL7200080A (en) 1971-08-18 1972-01-04
ES398587A ES398587A1 (en) 1971-08-18 1972-01-04 Imidazoles
BE777738A BE777738A (en) 1971-08-18 1972-01-05 HETEROCYCLIC COMPOUNDS
CH13772A CH584203A5 (en) 1971-08-18 1972-01-05
DE19722200499 DE2200499A1 (en) 1971-08-18 1972-01-05 2-PHENYL-5-AMINO-IMIDAZOLE, THEIR PHARMACOLOGICALLY COMPATIBLE SALTS, PROCESS FOR THEIR PRODUCTION AND ANTIPHLOGISTIC MEDICINAL PREPARATIONS CONTAINING THESE COMPOUNDS
US337062A US3876655A (en) 1971-08-18 1973-03-01 Anti-inflammatory acyl imidazoles

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB3871671A GB1378381A (en) 1971-08-18 1971-08-18 Imidazoles

Publications (1)

Publication Number Publication Date
GB1378381A true GB1378381A (en) 1974-12-27

Family

ID=10405251

Family Applications (1)

Application Number Title Priority Date Filing Date
GB3871671A Expired GB1378381A (en) 1971-08-18 1971-08-18 Imidazoles

Country Status (11)

Country Link
JP (1) JPS4829771A (en)
BE (1) BE777738A (en)
CH (1) CH584203A5 (en)
DE (1) DE2200499A1 (en)
ES (1) ES398587A1 (en)
FR (1) FR2149329B1 (en)
GB (1) GB1378381A (en)
IL (1) IL38357A (en)
NL (1) NL7200080A (en)
SE (1) SE376418B (en)
ZA (1) ZA7238B (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4197596A1 (en) * 2021-12-15 2023-06-21 Eberhard Karls Universität Tübingen Medizinische Fakultät Imidazole derivatives for the treatment and prophylaxis of infectious diseases

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4197596A1 (en) * 2021-12-15 2023-06-21 Eberhard Karls Universität Tübingen Medizinische Fakultät Imidazole derivatives for the treatment and prophylaxis of infectious diseases
WO2023110759A1 (en) * 2021-12-15 2023-06-22 Eberhard Karls Universitaet Tuebingen Medizinische Fakultaet New compound for the treatment and prophylaxis of infectious diseases

Also Published As

Publication number Publication date
FR2149329B1 (en) 1975-12-26
ZA7238B (en) 1972-09-27
CH584203A5 (en) 1977-01-31
SE376418B (en) 1975-05-26
JPS4829771A (en) 1973-04-19
BE777738A (en) 1972-07-05
IL38357A (en) 1976-08-31
FR2149329A1 (en) 1973-03-30
IL38357A0 (en) 1972-02-29
DE2200499A1 (en) 1973-03-08
NL7200080A (en) 1973-02-20
ES398587A1 (en) 1974-09-16

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Legal Events

Date Code Title Description
PS Patent sealed [section 19, patents act 1949]
PCNP Patent ceased through non-payment of renewal fee