GB1299246A - Imidazole derivatives - Google Patents

Imidazole derivatives

Info

Publication number
GB1299246A
GB1299246A GB1254671A GB1254671A GB1299246A GB 1299246 A GB1299246 A GB 1299246A GB 1254671 A GB1254671 A GB 1254671A GB 1254671 A GB1254671 A GB 1254671A GB 1299246 A GB1299246 A GB 1299246A
Authority
GB
United Kingdom
Prior art keywords
group
hal
hydrogen
atom
dibenzo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB1254671A
Inventor
Cornelis Van Der Stelt
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Nv Koninklijke Pharmaceutische Fabriken V/h Brocades-Stheeman & Pharmacia
Koninklijke Pharmaceutische Fabrieken NV
Original Assignee
Nv Koninklijke Pharmaceutische Fabriken V/h Brocades-Stheeman & Pharmacia
Koninklijke Pharmaceutische Fabrieken NV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nv Koninklijke Pharmaceutische Fabriken V/h Brocades-Stheeman & Pharmacia, Koninklijke Pharmaceutische Fabrieken NV filed Critical Nv Koninklijke Pharmaceutische Fabriken V/h Brocades-Stheeman & Pharmacia
Priority to US00151913A priority Critical patent/US3764609A/en
Priority to NL7108386A priority patent/NL7108386A/xx
Priority to IT6912371A priority patent/IT1044221B/en
Priority to DE19712130674 priority patent/DE2130674A1/en
Priority to FR7122498A priority patent/FR2100808A1/en
Priority to CA116,166A priority patent/CA972751A/en
Priority to AT533471A priority patent/AT303722B/en
Priority to ES392479A priority patent/ES392479A1/en
Priority to BE768807A priority patent/BE768807A/xx
Priority to LU63392D priority patent/LU63392A1/xx
Priority to CH903871A priority patent/CH560195A5/xx
Publication of GB1299246A publication Critical patent/GB1299246A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

1299246 Imidazoles KONINKLIJKE PHARMACEUTISCHE FABRIEKEN NV 22 June 1971 [22 June 1970 30 April 1971] 30246/70 and 12546/71 Heading C2C Novel imidazoles of the general formula wherein R 1 and R 2 are each a hydrogen or halogen atom or a C 1-6 alkyl group, R 3 , R 4 and R 5 are each a hydrogen atom or a C 1-12 alkyl group, X is a direct bond or a -(CH 2 ) 2 -, -(CH 2 ) 3 -, -CH=CH- or -CH=C(Hal)- group, in which Hal is a chlorine or bromine atom, and acid addition and quaternary ammonium salts thereof are prepared (a) by reacting compounds of formulae wherein Z is a hydrogen, alkali metal or silver atom and Y is the acid residue of a reactive ester or (b) when X is a -CH = CH-group, by reducing the corresponding compound wherein X is a -CH = C(Hal)- group; followed optionally by salifying the product. 5,10-Dichloro-5H-dibenzo-[a,d] cycloheptene is prepared by reaction of 5H-dibenzo [a,d]cyclohepten-5-one with phosphorus pentachloride. Fungicidal compositions for pharmaceutical and agricultural use comprise, as active ingredient, an imidazole of the first general formula above or an acid addition or quaternary ammonium salt thereof, in association with a suitable carrier or diluent.
GB1254671A 1970-06-22 1970-06-22 Imidazole derivatives Expired GB1299246A (en)

Priority Applications (11)

Application Number Priority Date Filing Date Title
US00151913A US3764609A (en) 1970-06-22 1971-06-10 1 (dibenzo {8 4,d{9 {0 cyclohepten-5-yl), 1-(dibenzo {8 a,d{9 {0 cycloheptan-5-yl) and 1-(dibenzo {8 a,d{9 {0 cyclooctanyl)imidazoles
NL7108386A NL7108386A (en) 1970-06-22 1971-06-18
IT6912371A IT1044221B (en) 1970-06-22 1971-06-21 IMIDAZOLE DERIVATIVES PROCEDURE FOR THEIR PHARMACEUTICAL PREPARATION AND COMPOSITION CONTAINING THEM
DE19712130674 DE2130674A1 (en) 1970-06-22 1971-06-21 Imidazole derivatives, their salts with acids and quaternary ammonium salts, processes for their preparation and their use as fungicides
FR7122498A FR2100808A1 (en) 1970-06-22 1971-06-21 Dibenzo cyclo alkylene and - cycloalkyl - imidazoles - - as fungicides for human animal and plant use
CA116,166A CA972751A (en) 1970-06-22 1971-06-21 Imidazole derivatives
AT533471A AT303722B (en) 1970-06-22 1971-06-21 Process for the production of new imidazole derivatives and their salts
ES392479A ES392479A1 (en) 1970-06-22 1971-06-21 Procedure for the preparation of imidazole derivatives. (Machine-translation by Google Translate, not legally binding)
BE768807A BE768807A (en) 1970-06-22 1971-06-21
LU63392D LU63392A1 (en) 1970-06-22 1971-06-21
CH903871A CH560195A5 (en) 1970-06-22 1971-06-21

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB3024670 1970-06-22

Publications (1)

Publication Number Publication Date
GB1299246A true GB1299246A (en) 1972-12-13

Family

ID=10304607

Family Applications (1)

Application Number Title Priority Date Filing Date
GB1254671A Expired GB1299246A (en) 1970-06-22 1970-06-22 Imidazole derivatives

Country Status (1)

Country Link
GB (1) GB1299246A (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4169205A (en) * 1978-10-25 1979-09-25 E. R. Squibb & Sons, Inc. Imidazole derivatives of 6,11-dihydrodibenz[b,e]oxepines and 6,11-dihydrodibenz[b,e]thiepines

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4169205A (en) * 1978-10-25 1979-09-25 E. R. Squibb & Sons, Inc. Imidazole derivatives of 6,11-dihydrodibenz[b,e]oxepines and 6,11-dihydrodibenz[b,e]thiepines

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Legal Events

Date Code Title Description
PS Patent sealed
PLNP Patent lapsed through nonpayment of renewal fees