GB1284681A - Improvements in or relating to 4,5,6,7-tetrahydroindazoles - Google Patents
Improvements in or relating to 4,5,6,7-tetrahydroindazolesInfo
- Publication number
- GB1284681A GB1284681A GB43847/70A GB4384770A GB1284681A GB 1284681 A GB1284681 A GB 1284681A GB 43847/70 A GB43847/70 A GB 43847/70A GB 4384770 A GB4384770 A GB 4384770A GB 1284681 A GB1284681 A GB 1284681A
- Authority
- GB
- United Kingdom
- Prior art keywords
- group
- carbon atoms
- radical
- alkyl group
- straight
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- GDSQTWDUCDSZEY-UHFFFAOYSA-N 4,5,6,7-tetrahydro-1h-indazole Chemical class C1CCCC2=C1C=NN2 GDSQTWDUCDSZEY-UHFFFAOYSA-N 0.000 title abstract 3
- 125000004432 carbon atom Chemical group C* 0.000 abstract 13
- 125000000217 alkyl group Chemical group 0.000 abstract 9
- -1 4-acetaminocyclohexyl radical Chemical class 0.000 abstract 7
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 4
- 150000003254 radicals Chemical class 0.000 abstract 4
- KDLHZDBZIXYQEI-UHFFFAOYSA-N Palladium Chemical compound [Pd] KDLHZDBZIXYQEI-UHFFFAOYSA-N 0.000 abstract 2
- 239000002253 acid Substances 0.000 abstract 2
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 2
- 125000004181 carboxyalkyl group Chemical group 0.000 abstract 2
- BASFCYQUMIYNBI-UHFFFAOYSA-N platinum Chemical compound [Pt] BASFCYQUMIYNBI-UHFFFAOYSA-N 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- BAXOFTOLAUCFNW-UHFFFAOYSA-N 1H-indazole Chemical compound C1=CC=C2C=NNC2=C1 BAXOFTOLAUCFNW-UHFFFAOYSA-N 0.000 abstract 1
- NYOWYNSNCXRVNQ-UHFFFAOYSA-N 2,3,3a,4-tetrahydro-1h-indazole Chemical class C1=CCC2CNNC2=C1 NYOWYNSNCXRVNQ-UHFFFAOYSA-N 0.000 abstract 1
- 125000000824 D-ribofuranosyl group Chemical group [H]OC([H])([H])[C@@]1([H])OC([H])(*)[C@]([H])(O[H])[C@]1([H])O[H] 0.000 abstract 1
- YUDRVAHLXDBKSR-UHFFFAOYSA-N [CH]1CCCCC1 Chemical compound [CH]1CCCCC1 YUDRVAHLXDBKSR-UHFFFAOYSA-N 0.000 abstract 1
- 125000002252 acyl group Chemical group 0.000 abstract 1
- 150000007933 aliphatic carboxylic acids Chemical class 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000002877 alkyl aryl group Chemical group 0.000 abstract 1
- 125000005119 alkyl cycloalkyl group Chemical group 0.000 abstract 1
- 125000005037 alkyl phenyl group Chemical group 0.000 abstract 1
- 125000002947 alkylene group Chemical group 0.000 abstract 1
- 125000000089 arabinosyl group Chemical group C1([C@@H](O)[C@H](O)[C@H](O)CO1)* 0.000 abstract 1
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 239000002585 base Substances 0.000 abstract 1
- 239000003054 catalyst Substances 0.000 abstract 1
- 125000001316 cycloalkyl alkyl group Chemical group 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 125000001511 cyclopentyl group Chemical group [H]C1([H])C([H])([H])C([H])([H])C([H])(*)C1([H])[H] 0.000 abstract 1
- 125000004663 dialkyl amino group Chemical group 0.000 abstract 1
- 239000012458 free base Substances 0.000 abstract 1
- 125000002791 glucosyl group Chemical group C1([C@H](O)[C@@H](O)[C@H](O)[C@H](O1)CO)* 0.000 abstract 1
- 150000002402 hexoses Chemical class 0.000 abstract 1
- 125000002768 hydroxyalkyl group Chemical group 0.000 abstract 1
- 125000004029 hydroxymethyl group Chemical group [H]OC([H])([H])* 0.000 abstract 1
- 125000001160 methoxycarbonyl group Chemical group [H]C([H])([H])OC(*)=O 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 125000004573 morpholin-4-yl group Chemical group N1(CCOCC1)* 0.000 abstract 1
- 229910052763 palladium Inorganic materials 0.000 abstract 1
- 150000002972 pentoses Chemical class 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 229910052697 platinum Inorganic materials 0.000 abstract 1
- 239000002243 precursor Substances 0.000 abstract 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
- 229910052703 rhodium Inorganic materials 0.000 abstract 1
- 239000010948 rhodium Substances 0.000 abstract 1
- MHOVAHRLVXNVSD-UHFFFAOYSA-N rhodium atom Chemical compound [Rh] MHOVAHRLVXNVSD-UHFFFAOYSA-N 0.000 abstract 1
- 239000000126 substance Substances 0.000 abstract 1
- 125000003718 tetrahydrofuranyl group Chemical group 0.000 abstract 1
- 150000003538 tetroses Chemical class 0.000 abstract 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 1
- 125000000969 xylosyl group Chemical group C1([C@H](O)[C@@H](O)[C@H](O)CO1)* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
- C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Catalysts (AREA)
- Compositions Of Macromolecular Compounds (AREA)
- Preventing Corrosion Or Incrustation Of Metals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19691948793 DE1948793A1 (de) | 1969-09-26 | 1969-09-26 | Verfahren zur Herstellung von 4,5,6,7-Tetrahydroindazolen |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1284681A true GB1284681A (en) | 1972-08-09 |
Family
ID=5746641
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB43847/70A Expired GB1284681A (en) | 1969-09-26 | 1970-09-14 | Improvements in or relating to 4,5,6,7-tetrahydroindazoles |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US3736332A (https=) |
| JP (1) | JPS4924069B1 (https=) |
| DE (1) | DE1948793A1 (https=) |
| FR (1) | FR2062635A5 (https=) |
| GB (1) | GB1284681A (https=) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1052111B (it) * | 1972-02-29 | 1981-06-20 | Acraf | Acidi i benzil i h indazol 3 carbossilici sostituiti e loro derivati |
| US3994890A (en) * | 1974-01-31 | 1976-11-30 | Chugai Seiyaku Kabushiki Kaisha | 1-Aminoalkyl, 3-phenyl indazoles |
| FR2265739B1 (https=) * | 1974-03-29 | 1976-12-17 | Ugine Kuhlmann | |
| GB1447923A (en) * | 1974-05-02 | 1976-09-02 | Science Union & Cie | Indazole derivatives processes for their preparation and pharma ceutical compositions containing them |
| US4014878A (en) * | 1974-05-23 | 1977-03-29 | Morton-Norwich Products, Inc. | 2-(3-Morpholinopropyl)-5,6-dimethoxy indazole |
| US4014886A (en) * | 1974-05-23 | 1977-03-29 | Morton-Norwich Products, Inc. | 2-Substituted-5,6-dimethoxyindazoles |
| FR2315924A1 (fr) * | 1975-07-03 | 1977-01-28 | Enzypha | Nouveaux polymethylene-4,5 pyrazoles, leur procede de preparation et leur application en therapeutique |
| US4322540A (en) * | 1979-03-15 | 1982-03-30 | Eli Lilly And Company | Substituted 4,5,6,7-tetrahydro-1H (or 2H)-indazoles |
| DE3132916A1 (de) * | 1981-08-20 | 1983-03-03 | Kali-Chemie Pharma Gmbh, 3000 Hannover | 1-phenylindazol-3-on-verbindungen sowie verfahren und zwischenprodukte zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
| GR80558B (en) * | 1983-10-08 | 1985-02-06 | Nippon Kayaku Kk | Derivative of pyrazole and use thereof as a herbicide |
| EP0226624A1 (en) * | 1985-06-14 | 1987-07-01 | The Upjohn Company | Cyclopentapyrazole and tetrahydroindazole compounds |
| GB8729801D0 (en) * | 1987-12-22 | 1988-02-03 | Beecham Group Plc | Novel process |
| US7888381B2 (en) * | 2005-06-14 | 2011-02-15 | Bristol-Myers Squibb Company | Modulators of glucocorticoid receptor, AP-1, and/or NF-κB activity, and use thereof |
| JP7312024B2 (ja) * | 2019-06-06 | 2023-07-20 | 大塚化学株式会社 | ゴム組成物、及びタイヤ |
| KR102859100B1 (ko) * | 2018-08-30 | 2025-09-12 | 오츠카 가가쿠 가부시키가이샤 | 고무 조성물, 고무 재료, 및 그들의 용도, 그리고 첨가제 |
-
1969
- 1969-09-26 DE DE19691948793 patent/DE1948793A1/de active Pending
-
1970
- 1970-09-14 GB GB43847/70A patent/GB1284681A/en not_active Expired
- 1970-09-18 US US00073643A patent/US3736332A/en not_active Expired - Lifetime
- 1970-09-24 JP JP45083058A patent/JPS4924069B1/ja active Pending
- 1970-09-25 FR FR7034760A patent/FR2062635A5/fr not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| FR2062635A5 (https=) | 1971-06-25 |
| DE1948793A1 (de) | 1971-04-01 |
| JPS4924069B1 (https=) | 1974-06-20 |
| US3736332A (en) | 1973-05-29 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed [section 19, patents act 1949] | ||
| PLNP | Patent lapsed through nonpayment of renewal fees |