GB1269081A - P-aminoalkylbenzene sulfonamide derivatives their preparation and composition containing same - Google Patents
P-aminoalkylbenzene sulfonamide derivatives their preparation and composition containing sameInfo
- Publication number
- GB1269081A GB1269081A GB03512/69A GB1351269A GB1269081A GB 1269081 A GB1269081 A GB 1269081A GB 03512/69 A GB03512/69 A GB 03512/69A GB 1351269 A GB1351269 A GB 1351269A GB 1269081 A GB1269081 A GB 1269081A
- Authority
- GB
- United Kingdom
- Prior art keywords
- alkyl
- carbons
- carbamide
- cycloalkyl
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D203/00—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom
- C07D203/04—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D203/06—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D203/22—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
- C07D203/24—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/44—Nitrogen atoms not forming part of a nitro radical
- C07D233/46—Nitrogen atoms not forming part of a nitro radical with only hydrogen atoms attached to said nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
1,269,081. Hypoglycaemic compositions. J. R. GEIGY A.G. 14 March, 1969 [14 March, 1968], No. 13512/69. Heading A5B. [Also in Division C2] Pharmaceutical preparations showing hypoglycaemic action contain as active ingredient compounds I (including salts thereof) wherein R 1 is C 1 to 12 alkyl, C 3 to 5 alkenyl, optionally alkyl-substituted, cycloalkyl or cycloalkenyl of not more than 7 carbons or phenylalkyl of not more than 9 carbons, R 2 is H, Me or Et, R 3 is H, C 1 to 7 alkyl, C 1 to 7 chloroalkyl, alkenyl with not more than 5 carbons, optionally alkyl-substituted, cycloalkyl or cycloalkenyl or cycloalkyl-alkyl of not more than 8 carbons, phenyl phenylalkyl or phenylalkenyl of not more than 10 carbons wherein the phenyl group can be mono-, di- or tri-substituted by F, Cl, Br, CF 3 , C 1 to 4 alkyl, OH, MeO, EtO, MeS and/or EtS, R 4 is H or Me and m is 2 or 3. In addition to the usual acids, the salt forming component may be a sulphonyl - urea, e.g. N 1 - p - tolylsulphonyl - N 2 - butyl - carbamide, N 1 - p -chlorobenzenesulphonyl - N 2 - propyl - carbamide and N 1 - p - [2 - (2 - methoxy - 5 - chlorobenzamido) - ethyl] - phenylsulphonyl - N 2 - cyclohexyl - carbamide. Administration is preferably by the oral route.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH388468A CH505829A (en) | 1968-03-14 | 1968-03-14 | Process for the preparation of new derivatives of p-aminoalkylbenzenesulfonamide |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1269081A true GB1269081A (en) | 1972-03-29 |
Family
ID=4265567
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB03512/69A Expired GB1269081A (en) | 1968-03-14 | 1969-03-14 | P-aminoalkylbenzene sulfonamide derivatives their preparation and composition containing same |
Country Status (18)
| Country | Link |
|---|---|
| JP (6) | JPS5020071B1 (en) |
| AT (1) | AT287694B (en) |
| BE (1) | BE729837A (en) |
| BG (6) | BG17303A3 (en) |
| CH (1) | CH505829A (en) |
| CS (1) | CS166693B2 (en) |
| DE (1) | DE1912847B2 (en) |
| DK (1) | DK126327B (en) |
| FI (1) | FI51179C (en) |
| FR (1) | FR2003887A1 (en) |
| GB (1) | GB1269081A (en) |
| IE (1) | IE32670B1 (en) |
| IL (1) | IL31802A (en) |
| MY (1) | MY7500049A (en) |
| NL (1) | NL144931B (en) |
| NO (1) | NO124726B (en) |
| PL (1) | PL79938B1 (en) |
| SE (1) | SE354863B (en) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU579997B2 (en) * | 1983-04-05 | 1988-12-22 | Ciba-Geigy Ag | Iminosulphonamides and processes for the manufacture thereof, pharmaceutical preparations containing such compounds, and their use |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE754597A (en) * | 1969-08-08 | 1971-02-08 | Geigy Ag J R | ALKYL-BENZENE-SULFONAMIDES AND MEDICINAL PRODUCTS CONTAINING SUCH COMPOUNDS |
| BE755684A (en) * | 1969-09-04 | 1971-03-03 | Geigy Ag J R | P-AMINOALKYL-BENZENE-SULFONAMIDES AND MEDICINAL PRODUCTS CONTAINING SUCH COMPOUNDS |
| BE755686A (en) * | 1969-09-04 | 1971-03-03 | Geigy Ag J R | AMINOALKYL-BENZENE-SULFONAMIDES AND MEDICINAL PRODUCTS CONTAINING SUCH COMPOUNDS |
| BE755681A (en) * | 1969-09-04 | 1971-03-03 | Geigy Ag J R | P-AMINOALKYL-BENZENE-SULFONAMIDES AND MEDICINAL PRODUCTS CONTAINING SUCH COMPOUNDS |
| BE755682A (en) * | 1969-09-04 | 1971-03-03 | Geigy Ag J R | P-AMINOALKYL-BENZENE-SULFONAMIDES AND MEDICINAL PRODUCTS CONTAINING SUCH COMPOUNDS |
| US6335445B1 (en) * | 1997-03-24 | 2002-01-01 | Societe De Conseils De Recherches Et D'applications Scientifiques (S.C.R.A.S.) | Derivatives of 2-(iminomethyl)amino-phenyl, their preparation, their use as medicaments and the pharmaceutical compositions containing them |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1224812A (en) * | 1956-12-28 | 1960-06-27 | Geigy Ag J R | Novel 2-imino-1.3-di-n-heterocycles and their preparation process |
| GB1052113A (en) * | 1963-02-07 |
-
1968
- 1968-03-14 CH CH388468A patent/CH505829A/en not_active IP Right Cessation
-
1969
- 1969-03-05 FI FI690664A patent/FI51179C/en active
- 1969-03-07 DK DK127669AA patent/DK126327B/en not_active IP Right Cessation
- 1969-03-07 NO NO69968A patent/NO124726B/no unknown
- 1969-03-07 SE SE03171/69A patent/SE354863B/xx unknown
- 1969-03-12 NL NL696903831A patent/NL144931B/en not_active IP Right Cessation
- 1969-03-13 FR FR6907109A patent/FR2003887A1/fr not_active Withdrawn
- 1969-03-13 DE DE1912847A patent/DE1912847B2/en active Granted
- 1969-03-13 BG BG11840A patent/BG17303A3/xx unknown
- 1969-03-13 AT AT248269A patent/AT287694B/en not_active IP Right Cessation
- 1969-03-13 IE IE333/69A patent/IE32670B1/en unknown
- 1969-03-13 PL PL1969132326A patent/PL79938B1/en unknown
- 1969-03-13 IL IL31802A patent/IL31802A/en unknown
- 1969-03-13 CS CS1829A patent/CS166693B2/cs unknown
- 1969-03-13 BE BE729837D patent/BE729837A/xx not_active IP Right Cessation
- 1969-03-14 GB GB03512/69A patent/GB1269081A/en not_active Expired
- 1969-06-13 BG BG12441A patent/BG21216A3/xx unknown
- 1969-06-13 BG BG12439A patent/BG17304A3/xx unknown
- 1969-06-13 BG BG12438A patent/BG17539A3/xx unknown
- 1969-06-13 BG BG12440A patent/BG17540A3/xx unknown
- 1969-06-13 BG BG12442A patent/BG17305A3/xx unknown
-
1971
- 1971-02-20 JP JP46007935A patent/JPS5020071B1/ja active Pending
- 1971-02-20 JP JP46007932A patent/JPS5020068B1/ja active Pending
- 1971-02-20 JP JP46007934A patent/JPS5020070B1/ja active Pending
- 1971-02-20 JP JP46007931A patent/JPS5020067B1/ja active Pending
- 1971-02-20 JP JP46007933A patent/JPS5020069B1/ja active Pending
-
1975
- 1975-01-16 JP JP50006498A patent/JPS512468B1/ja active Pending
- 1975-12-30 MY MY49/75A patent/MY7500049A/en unknown
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU579997B2 (en) * | 1983-04-05 | 1988-12-22 | Ciba-Geigy Ag | Iminosulphonamides and processes for the manufacture thereof, pharmaceutical preparations containing such compounds, and their use |
Also Published As
| Publication number | Publication date |
|---|---|
| BE729837A (en) | 1969-09-15 |
| IL31802A0 (en) | 1969-05-28 |
| FR2003887A1 (en) | 1969-11-14 |
| IE32670L (en) | 1969-09-14 |
| JPS5020071B1 (en) | 1975-07-11 |
| BG17303A3 (en) | 1973-07-25 |
| IE32670B1 (en) | 1973-10-17 |
| DE1912847A1 (en) | 1969-10-16 |
| NO124726B (en) | 1972-05-29 |
| BG17540A3 (en) | 1973-11-10 |
| IL31802A (en) | 1972-09-28 |
| MY7500049A (en) | 1975-12-31 |
| CS166693B2 (en) | 1976-03-29 |
| FI51179B (en) | 1976-08-02 |
| DK126327B (en) | 1973-07-02 |
| JPS5020067B1 (en) | 1975-07-11 |
| DE1912847B2 (en) | 1978-09-14 |
| JPS5020068B1 (en) | 1975-07-11 |
| BG17304A3 (en) | 1973-07-25 |
| FI51179C (en) | 1976-11-10 |
| JPS512468B1 (en) | 1976-01-26 |
| BG21216A3 (en) | 1976-03-20 |
| JPS5020069B1 (en) | 1975-07-11 |
| BG17539A3 (en) | 1973-11-10 |
| NL6903831A (en) | 1969-09-16 |
| JPS5020070B1 (en) | 1975-07-11 |
| DE1912847C3 (en) | 1979-05-23 |
| NL144931B (en) | 1975-02-17 |
| SE354863B (en) | 1973-03-26 |
| PL79938B1 (en) | 1975-08-30 |
| BG17305A3 (en) | 1973-07-25 |
| AT287694B (en) | 1971-02-10 |
| CH505829A (en) | 1971-04-15 |
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