GB1265600A - - Google Patents
Info
- Publication number
- GB1265600A GB1265600A GB1265600DA GB1265600A GB 1265600 A GB1265600 A GB 1265600A GB 1265600D A GB1265600D A GB 1265600DA GB 1265600 A GB1265600 A GB 1265600A
- Authority
- GB
- United Kingdom
- Prior art keywords
- alkyl
- compounds
- indole
- july
- prepared
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Indole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
1,265,600. Indole-derived amino-thioethers. AGENCE NATIONALE DE VALORISATION DE LA RECHERCHE. 3 July, 1970 [7 July, 1969], No. 32396/70. Heading C2C; The invention comprises compounds of formula and their pharmacologically acceptable acid addition salts, wherein R 1 is C 1-6 -alkyl, C 1-6 - hydroxyalkyl- or (optionally substituted) phenyl- C 1-6 -alkyl; and R 2 , R 3 are each H, C 1-6 alkyl (optionally Ph-substituted) or aryl, or NR 2 R 3 constitute a 5, 6 or 7 membered heterocyclic ring. These compounds are prepared by reducing a 2-R 1 S-3-R 4 X-indole, where X is CH 2 or CO, and R 4 is CN or CONR 2 R 3 . Intermediates otherwise prepared are 2-R 1 S-3-Y-indoles, where Y is H, CH 2 NMe 2 , CH 2 CN, CH 2 CO 2 H, CH 2 CO 2 CO 2 Me or COCOCI. Therapeutic compositions, having, a sedative, neuroleptic and. tranquillizing activity; comprise compounds .of the above formula, which may beadministered orally, parenterally or rectally.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR6922947A FR2054460B1 (en) | 1969-07-07 | 1969-07-07 | |
| FR6922948A FR2054461B1 (en) | 1969-07-07 | 1969-07-07 | |
| FR7024841A FR2096837B2 (en) | 1969-07-07 | 1970-07-03 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1265600A true GB1265600A (en) | 1972-03-01 |
Family
ID=27249164
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB1265600D Expired GB1265600A (en) | 1969-07-07 | 1970-07-03 |
Country Status (6)
| Country | Link |
|---|---|
| BE (1) | BE752808A (en) |
| CH (1) | CH511228A (en) |
| DE (1) | DE2033668A1 (en) |
| FR (3) | FR2054461B1 (en) |
| GB (1) | GB1265600A (en) |
| SE (1) | SE367192B (en) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20160052923A1 (en) * | 2013-03-27 | 2016-02-25 | Bristol-Myers Squibb Company | Piperazine and homopiperazine derivatives as hiv attachment inhibitors |
-
1969
- 1969-07-07 FR FR6922948A patent/FR2054461B1/fr not_active Expired
- 1969-07-07 FR FR6922947A patent/FR2054460B1/fr not_active Expired
-
1970
- 1970-07-01 BE BE752808D patent/BE752808A/en unknown
- 1970-07-03 FR FR7024841A patent/FR2096837B2/fr not_active Expired
- 1970-07-03 GB GB1265600D patent/GB1265600A/en not_active Expired
- 1970-07-06 CH CH1020670A patent/CH511228A/en not_active IP Right Cessation
- 1970-07-06 SE SE09334/70A patent/SE367192B/xx unknown
- 1970-07-07 DE DE19702033668 patent/DE2033668A1/en active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| FR2096837A2 (en) | 1972-03-03 |
| CH511228A (en) | 1971-08-15 |
| FR2054461A1 (en) | 1971-04-23 |
| FR2096837B2 (en) | 1973-08-10 |
| DE2033668A1 (en) | 1971-01-21 |
| FR2054461B1 (en) | 1973-06-08 |
| FR2054460B1 (en) | 1973-06-08 |
| BE752808A (en) | 1971-01-04 |
| FR2054460A1 (en) | 1971-04-23 |
| SE367192B (en) | 1974-05-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed | ||
| PLNP | Patent lapsed through nonpayment of renewal fees |