GB1040547A - Benzodiazepine derivatives and their manufacture - Google Patents

Benzodiazepine derivatives and their manufacture

Info

Publication number
GB1040547A
GB1040547A GB823863A GB823863A GB1040547A GB 1040547 A GB1040547 A GB 1040547A GB 823863 A GB823863 A GB 823863A GB 823863 A GB823863 A GB 823863A GB 1040547 A GB1040547 A GB 1040547A
Authority
GB
United Kingdom
Prior art keywords
stands
compound
formula
symbol
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB823863A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of GB1040547A publication Critical patent/GB1040547A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24—Oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24—Oxygen atoms
    • C07D243/26—Preparation from compounds already containing the benzodiazepine skeleton

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
GB823863A 1962-03-02 1963-03-01 Benzodiazepine derivatives and their manufacture Expired GB1040547A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17690162A 1962-03-02 1962-03-02

Publications (1)

Publication Number Publication Date
GB1040547A true GB1040547A (en) 1966-09-01

Family

ID=22646360

Family Applications (2)

Application Number Title Priority Date Filing Date
GB823863A Expired GB1040547A (en) 1962-03-02 1963-03-01 Benzodiazepine derivatives and their manufacture
GB4791164A Expired GB1040548A (en) 1962-03-02 1963-03-01 Benzodiazepine derivatives and the manufacture thereof

Family Applications After (1)

Application Number Title Priority Date Filing Date
GB4791164A Expired GB1040548A (en) 1962-03-02 1963-03-01 Benzodiazepine derivatives and the manufacture thereof

Country Status (8)

Country Link
BE (1) BE629005A (enExample)
BR (1) BR6347108D0 (enExample)
CH (3) CH438336A (enExample)
CY (1) CY418A (enExample)
DE (1) DE1445874A1 (enExample)
GB (2) GB1040547A (enExample)
MY (1) MY6800032A (enExample)
SE (1) SE302127B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5662911A (en) * 1995-02-02 1997-09-02 Boehringer Mannheim Gmbh Benzodiazepine protein conjugates

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5218114A (en) * 1991-04-10 1993-06-08 Merck & Co., Inc. Cholecystokinin antagonists

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5662911A (en) * 1995-02-02 1997-09-02 Boehringer Mannheim Gmbh Benzodiazepine protein conjugates

Also Published As

Publication number Publication date
CH455815A (de) 1968-05-15
CH454887A (de) 1968-04-30
CH438336A (de) 1967-06-30
BE629005A (fr) 1963-08-28
MY6800032A (en) 1968-12-31
BR6347108D0 (pt) 1973-07-19
SE302127B (enExample) 1968-07-08
DE1445874A1 (enExample) 1970-07-23
GB1040548A (en) 1966-09-01
CY418A (en) 1967-11-30

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