GB0320313D0 - Process - Google Patents

Process

Info

Publication number
GB0320313D0
GB0320313D0 GBGB0320313.0A GB0320313A GB0320313D0 GB 0320313 D0 GB0320313 D0 GB 0320313D0 GB 0320313 A GB0320313 A GB 0320313A GB 0320313 D0 GB0320313 D0 GB 0320313D0
Authority
GB
United Kingdom
Prior art keywords
diaryliodium
salt
formula
ring
fluoridation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
GBGB0320313.0A
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Newcastle University Ventures Ltd
IC Innovations Ltd
Original Assignee
Newcastle University Ventures Ltd
IC Innovations Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Newcastle University Ventures Ltd, IC Innovations Ltd filed Critical Newcastle University Ventures Ltd
Priority to GBGB0320313.0A priority Critical patent/GB0320313D0/en
Publication of GB0320313D0 publication Critical patent/GB0320313D0/en
Priority to PCT/GB2004/003621 priority patent/WO2005021472A2/en
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C41/00—Preparation of ethers; Preparation of compounds having groups, groups or groups
    • C07C41/01—Preparation of ethers
    • C07C41/18—Preparation of ethers by reactions not forming ether-oxygen bonds
    • C07C41/22—Preparation of ethers by reactions not forming ether-oxygen bonds by introduction of halogens; by substitution of halogen atoms by other halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B39/00—Halogenation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/361—Preparation of halogenated hydrocarbons by reactions involving a decrease in the number of carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C25/00—Compounds containing at least one halogen atom bound to a six-membered aromatic ring
    • C07C25/18—Polycyclic aromatic halogenated hydrocarbons
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/05—Isotopically modified compounds, e.g. labelled

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Catalysts (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

The present invention provides a process for the fluoridation of the electron rich aryl group (A) in a diaryliodium salt of formula (I). The process comprises contacting a compound of formula (I) with a source of fluoride, wherein in the diaryliodium salt (1), the ring (B) is more electronegative than the ring (A).
GBGB0320313.0A 2003-08-29 2003-08-29 Process Ceased GB0320313D0 (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
GBGB0320313.0A GB0320313D0 (en) 2003-08-29 2003-08-29 Process
PCT/GB2004/003621 WO2005021472A2 (en) 2003-08-29 2004-08-24 Fluoridation of electron rich aromatic systems

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0320313.0A GB0320313D0 (en) 2003-08-29 2003-08-29 Process

Publications (1)

Publication Number Publication Date
GB0320313D0 true GB0320313D0 (en) 2003-10-01

Family

ID=28686597

Family Applications (1)

Application Number Title Priority Date Filing Date
GBGB0320313.0A Ceased GB0320313D0 (en) 2003-08-29 2003-08-29 Process

Country Status (2)

Country Link
GB (1) GB0320313D0 (en)
WO (1) WO2005021472A2 (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0808986D0 (en) 2008-05-16 2008-06-25 Univ Newcastle Formation of 18F and 19F fluoroarenes bearing reactive functionalities
EP2349977A4 (en) 2008-10-21 2012-03-28 Nutech Ventures Fluorination of aromatic ring systems
US9302990B2 (en) 2008-10-21 2016-04-05 Nutech Ventures Fluorination of aromatic ring systems
US8546578B2 (en) 2010-02-04 2013-10-01 Nutech Ventures Iodonium Cyclophanes for SECURE arene functionalization
WO2017089492A1 (en) * 2015-11-24 2017-06-01 Institut National De La Sante Et De La Recherche Medicale (Inserm) Method for synthesizing iodo- or astatoarenes using diaryliodonium salts

Also Published As

Publication number Publication date
WO2005021472A3 (en) 2005-04-21
WO2005021472A2 (en) 2005-03-10

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Legal Events

Date Code Title Description
AT Applications terminated before publication under section 16(1)