FR2953513B1 - Nouveaux derives azabicyclo[3.2.0]hept-6-yl, leur procede de preparation et les compositions pharmaceutiques qui les contiennent - Google Patents

Nouveaux derives azabicyclo[3.2.0]hept-6-yl, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Info

Publication number
FR2953513B1
FR2953513B1 FR0905954A FR0905954A FR2953513B1 FR 2953513 B1 FR2953513 B1 FR 2953513B1 FR 0905954 A FR0905954 A FR 0905954A FR 0905954 A FR0905954 A FR 0905954A FR 2953513 B1 FR2953513 B1 FR 2953513B1
Authority
FR
France
Prior art keywords
hept
derivatives
preparing
pharmaceutical compositions
compositions containing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR0905954A
Other languages
English (en)
Other versions
FR2953513A1 (fr
Inventor
Patrick Casara
Anne Marie Chollet
Alain Dhainaut
Jean Michel Henlin
Pierre Lestage
Fany Panayi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Laboratoires Servier SAS
Original Assignee
Laboratoires Servier SAS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Laboratoires Servier SAS filed Critical Laboratoires Servier SAS
Priority to FR0905954A priority Critical patent/FR2953513B1/fr
Priority to UY0001033074A priority patent/UY33074A/es
Priority to TW099142188A priority patent/TW201144279A/zh
Priority to ARP100104485A priority patent/AR079266A1/es
Priority to PCT/FR2010/000822 priority patent/WO2011070252A1/fr
Publication of FR2953513A1 publication Critical patent/FR2953513A1/fr
Application granted granted Critical
Publication of FR2953513B1 publication Critical patent/FR2953513B1/fr
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/12Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Anesthesiology (AREA)
  • Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR0905954A 2009-12-09 2009-12-09 Nouveaux derives azabicyclo[3.2.0]hept-6-yl, leur procede de preparation et les compositions pharmaceutiques qui les contiennent Expired - Fee Related FR2953513B1 (fr)

Priority Applications (5)

Application Number Priority Date Filing Date Title
FR0905954A FR2953513B1 (fr) 2009-12-09 2009-12-09 Nouveaux derives azabicyclo[3.2.0]hept-6-yl, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
UY0001033074A UY33074A (es) 2009-12-09 2010-12-01 Nuevos derivados de azabiciclo[3.2.0]hept-6-ilo, su procedimiento de preparación y las composiciones farmacéuticas que los contienen
TW099142188A TW201144279A (en) 2009-12-09 2010-12-03 New azabicyclo[3.2.0]hept-6-yl compounds, a process for their preparation and pharmaceutical compositions containing them
ARP100104485A AR079266A1 (es) 2009-12-09 2010-12-06 Derivados de azabiciclo[3.2.0]hept-6ilo, procedimiento de preparacion de los mismos, intermediarios de sintesis, composiciones farmaceuticas que los contienen y uso de los mismos para el tratamiento de enfermedades neurodegenerativas,tales como alzheimer.
PCT/FR2010/000822 WO2011070252A1 (fr) 2009-12-09 2010-12-08 Derives d'azabicyclo[3.2.0]hept-6-yle comme antagonistes des recepteurs histaminergiques de type h3

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0905954A FR2953513B1 (fr) 2009-12-09 2009-12-09 Nouveaux derives azabicyclo[3.2.0]hept-6-yl, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Publications (2)

Publication Number Publication Date
FR2953513A1 FR2953513A1 (fr) 2011-06-10
FR2953513B1 true FR2953513B1 (fr) 2011-12-23

Family

ID=42123039

Family Applications (1)

Application Number Title Priority Date Filing Date
FR0905954A Expired - Fee Related FR2953513B1 (fr) 2009-12-09 2009-12-09 Nouveaux derives azabicyclo[3.2.0]hept-6-yl, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Country Status (5)

Country Link
AR (1) AR079266A1 (fr)
FR (1) FR2953513B1 (fr)
TW (1) TW201144279A (fr)
UY (1) UY33074A (fr)
WO (1) WO2011070252A1 (fr)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2866647B1 (fr) * 2004-02-20 2006-10-27 Servier Lab Nouveaux derives azabicycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
FR2953513A1 (fr) 2011-06-10
TW201144279A (en) 2011-12-16
WO2011070252A1 (fr) 2011-06-16
AR079266A1 (es) 2012-01-04
UY33074A (es) 2011-04-29

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Legal Events

Date Code Title Description
ST Notification of lapse

Effective date: 20130830