FR2951173B1 - Nouveaux derives de 2,3-dihydro-1h-imidazo{1,2-a}pyrimidin-5-one, leur preparation et leur utilisation pharmaceutique comme inhibiteurs de phosphorylation d'akt(pkb) - Google Patents
Nouveaux derives de 2,3-dihydro-1h-imidazo{1,2-a}pyrimidin-5-one, leur preparation et leur utilisation pharmaceutique comme inhibiteurs de phosphorylation d'akt(pkb)Info
- Publication number
- FR2951173B1 FR2951173B1 FR0957067A FR0957067A FR2951173B1 FR 2951173 B1 FR2951173 B1 FR 2951173B1 FR 0957067 A FR0957067 A FR 0957067A FR 0957067 A FR0957067 A FR 0957067A FR 2951173 B1 FR2951173 B1 FR 2951173B1
- Authority
- FR
- France
- Prior art keywords
- pkb
- imidazo
- pyrimidin
- dihydro
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (27)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0957067A FR2951173B1 (fr) | 2009-10-09 | 2009-10-09 | Nouveaux derives de 2,3-dihydro-1h-imidazo{1,2-a}pyrimidin-5-one, leur preparation et leur utilisation pharmaceutique comme inhibiteurs de phosphorylation d'akt(pkb) |
HUE10742012A HUE034503T2 (en) | 2009-07-02 | 2010-07-01 | 2,3-Dihydro-1-imidazo [1,2-a] pyrimidin-5-one derivatives, their preparation process and their use in medicine |
RU2012103460/04A RU2554868C2 (ru) | 2009-07-02 | 2010-07-01 | НОВЫЕ ПРОИЗВОДНЫЕ 2,3-ДИГИДРО-1Н-ИМИДАЗО[1,2-а]ПИРИМИДИН-5-ОНА, СПОСОБ ИХ ПОЛУЧЕНИЯ И ПРИМЕНЕНИЕ В ФАРМАЦИИ |
CN201080039104.3A CN102482285B (zh) | 2009-07-02 | 2010-07-01 | 2,3-二氢-1H-咪唑并{1,2-a}嘧啶-5-酮衍生物,其制备和其药物用途 |
ES10742012.7T ES2627428T3 (es) | 2009-07-02 | 2010-07-01 | Nuevos derivados de 2,3-dihidro-1H-imidazo{1,2-a}pirimidin-5-ona, su preparación y su utilización farmacéutica |
BRPI1015949A BRPI1015949A2 (pt) | 2009-07-02 | 2010-07-01 | derivados de 2,3-di-hidro-1h-imidazo [1,2-a] pirimidin-5-ona, o respectivo preparo e a respectiva utilização farmacêutica |
PL10742012T PL2448939T3 (pl) | 2009-07-02 | 2010-07-01 | Pochodne 2,3-dihydro-1h-imidazo {1,2-a} pirymidyn-5-onu, ich wytwarzanie i ich zastosowanie farmaceutyczne |
PCT/FR2010/051373 WO2011001112A1 (fr) | 2009-07-02 | 2010-07-01 | NOUVEAUX DERIVES DE 2,3-DIHYDRO-1H-IMIDAZO{1,2-a}PYRIMIDIN-5-ONE, LEUR PREPARATION ET LEUR UTILISATION PHARMACEUTIQUE |
LTEP10742012.7T LT2448939T (lt) | 2009-07-02 | 2010-07-01 | 2,3-dihidro-1h-imidazo {1,2-a} pirimidin-5-ono dariniai, jų gamyba ir farmacinis panaudojimas |
PT107420127T PT2448939T (pt) | 2009-07-02 | 2010-07-01 | Derivados de 2,3-dihidro-1h-imidazo{1,2-a}pirimidin-5-ona, sua preparação e sua utilização farmacêutica |
US13/381,571 US8828997B2 (en) | 2009-07-02 | 2010-07-01 | 2,3-dihydro-1H-imidazo(1,2-a)pyrimidin-5-one derivatives, preparation thereof, and pharmaceutical use thereof |
EP10742012.7A EP2448939B1 (fr) | 2009-07-02 | 2010-07-01 | Derives de 2,3-dihydro-1h-imidazo {1,2-a} pyrimidin-5-one, leur preparation et leur utilisation pharmaceutique |
SI201031451A SI2448939T1 (sl) | 2009-07-02 | 2010-07-01 | Derivati 2,3-dihidro-1H-imidazo(1,2-a)pirimidin-5-ona, njihova priprava in farmacevtska uporaba |
MX2012000097A MX2012000097A (es) | 2009-07-02 | 2010-07-01 | Nuevos derivados de 2,3-dihidro-1h-imidazo {1,2-a} pirimidin-5-ona, su preparacion y su uso en farmaceutica. |
DK10742012.7T DK2448939T3 (en) | 2009-07-02 | 2010-07-01 | DERIVATIVES OF 2,3-DIHYDRO-1H-IMIDAZO {1,2-A} PYRIMIDIN-5-ON, PREPARATION AND PHARMACEUTICAL USE thereof |
ARP100102346A AR077446A1 (es) | 2009-07-02 | 2010-07-01 | Derivados de 2,3-dihidro-1h-imidazo(1,2-a) pirimidin-5-ona. su preparacion y su utilizacion farmaceutica |
CA2767051A CA2767051C (fr) | 2009-07-02 | 2010-07-01 | Nouveaux derives de 2,3-dihydro-1h-imidazo{1,2-a}pyrimidin-5-one, leur preparation et leur utilisation pharmaceutique |
SG2011097227A SG177421A1 (en) | 2009-07-02 | 2010-07-01 | Novel 2,3-dihydro-1h-imidazo(1,2-a)pyrimidin-5-one derivatives, preparation thereof, and pharmaceutical use thereof |
JP2012518118A JP5663571B2 (ja) | 2009-07-02 | 2010-07-01 | 新規2,3−ジヒドロ−1H−イミダゾ{1,2−a}ピリミジン−5−オン誘導体、これらの調製およびこれらの薬学的使用 |
AU2010267814A AU2010267814B2 (en) | 2009-07-02 | 2010-07-01 | Novel 2,3-dihydro-1H-imidazo(1,2-a)pyrimidin-5-one derivatives, preparation thereof, and pharmaceutical use thereof |
SG10201403138WA SG10201403138WA (en) | 2009-07-02 | 2010-07-01 | Novel 2,3-dihydro-1h-imidazo(1,2-a)pyrimidin-5-one derivatives, preparation thereof and pharmaceutical use thereof |
KR1020127002797A KR101745028B1 (ko) | 2009-07-02 | 2010-07-01 | 신규 2,3-디히드로-1h-이미다조(1,2-a)피리미딘-5-온 유도체, 그의 제조법 및 그의 제약 용도 |
TW099121898A TWI458730B (zh) | 2009-07-02 | 2010-07-02 | 新穎2,3-二氫-1H-咪唑并{1,2-a}嘧啶-5-酮衍生物,其製法及其醫藥用途 |
UY0001032753A UY32753A (es) | 2009-07-02 | 2010-07-02 | NUEVOS DERIVADOS DE 2,3-DIHIDRO-1H-IMIDAZO{1,2-a}PIRIMIDIN-5-ONA, SU PREPARACIÓN Y SU UTILIZACIÓN EN FARMACÉUTICA |
IL217294A IL217294A (en) | 2009-07-02 | 2011-12-29 | History 3,2 - Dihydro - 1h - Imidazo [1, 2 - a] - Pyrimidin - 5 - On, process for their preparation, pharmaceutical preparations containing them and their use in the preparation of medicines |
HRP20170827TT HRP20170827T1 (hr) | 2009-07-02 | 2017-05-30 | Derivati 2,3-dihidro-1h-imidazo {1,2-a} pirimidin-5-ona, njihova priprava i farmaceutska primjena |
CY20171100567T CY1119442T1 (el) | 2009-07-02 | 2017-05-31 | Παραγωγα 2,3-διϋδρο-1η-ιμιδαζο {1,2-α} πυριμιδιν-5-ονης, παρασκευη αυτων και φαρμακευτικη χρηση αυτων |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0957067A FR2951173B1 (fr) | 2009-10-09 | 2009-10-09 | Nouveaux derives de 2,3-dihydro-1h-imidazo{1,2-a}pyrimidin-5-one, leur preparation et leur utilisation pharmaceutique comme inhibiteurs de phosphorylation d'akt(pkb) |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2951173A1 FR2951173A1 (fr) | 2011-04-15 |
FR2951173B1 true FR2951173B1 (fr) | 2011-12-02 |
Family
ID=42077171
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR0957067A Expired - Fee Related FR2951173B1 (fr) | 2009-07-02 | 2009-10-09 | Nouveaux derives de 2,3-dihydro-1h-imidazo{1,2-a}pyrimidin-5-one, leur preparation et leur utilisation pharmaceutique comme inhibiteurs de phosphorylation d'akt(pkb) |
Country Status (1)
Country | Link |
---|---|
FR (1) | FR2951173B1 (fr) |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2008148074A2 (fr) * | 2007-05-24 | 2008-12-04 | Research Foundation Of State University Of New York | Inhibiteurs de mtor et methodes de traitement mettant en œuvre ces inhibiteurs |
-
2009
- 2009-10-09 FR FR0957067A patent/FR2951173B1/fr not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
FR2951173A1 (fr) | 2011-04-15 |
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Legal Events
Date | Code | Title | Description |
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ST | Notification of lapse |
Effective date: 20160630 |