FR2874611A1 - NOVEL IMIDAZOPYRIDINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM - Google Patents

NOVEL IMIDAZOPYRIDINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Info

Publication number
FR2874611A1
FR2874611A1 FR0409202A FR0409202A FR2874611A1 FR 2874611 A1 FR2874611 A1 FR 2874611A1 FR 0409202 A FR0409202 A FR 0409202A FR 0409202 A FR0409202 A FR 0409202A FR 2874611 A1 FR2874611 A1 FR 2874611A1
Authority
FR
France
Prior art keywords
preparation
pharmaceutical compositions
compositions containing
imidazopyridine derivatives
novel imidazopyridine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR0409202A
Other languages
French (fr)
Other versions
FR2874611B1 (en
Inventor
Gerald Guillaumet
Raboin Sabine Berteina
Kazzouli Said El
Philippe Delagrange
Daniel Henri Caignard
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Laboratoires Servier SAS
Original Assignee
Laboratoires Servier SAS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Laboratoires Servier SAS filed Critical Laboratoires Servier SAS
Priority to FR0409202A priority Critical patent/FR2874611B1/en
Priority to PCT/FR2005/002162 priority patent/WO2006027474A2/en
Priority to ARP050103619A priority patent/AR050542A1/en
Publication of FR2874611A1 publication Critical patent/FR2874611A1/en
Application granted granted Critical
Publication of FR2874611B1 publication Critical patent/FR2874611B1/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Composés de formule (I) :dans laquelle :• A représente un groupement -NHCOR1 ou -CONHR1 dans lesquels R1 est tel que défini dans la description,• R2 représente un groupement alkoxy,• R3 représente un groupement aryle, arylalkyle ou aroyle,Médicaments.Compounds of formula (I): in which: • A represents a group -NHCOR1 or -CONHR1 in which R1 is as defined in the description, • R2 represents an alkoxy group, • R3 represents an aryl, arylalkyl or aroyl group, Drugs .

FR0409202A 2004-08-31 2004-08-31 NOVEL IMIDAZOPYRIDINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Expired - Fee Related FR2874611B1 (en)

Priority Applications (3)

Application Number Priority Date Filing Date Title
FR0409202A FR2874611B1 (en) 2004-08-31 2004-08-31 NOVEL IMIDAZOPYRIDINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
PCT/FR2005/002162 WO2006027474A2 (en) 2004-08-31 2005-08-30 Novel imidazopyridine derivatives having an affinity with respect to melatonin receptors, method for the preparation thereof and pharmaceutical compositions containing said derivatives
ARP050103619A AR050542A1 (en) 2004-08-31 2005-08-30 IMIDAZOPIRIDINE COMPOUNDS PROCEDURE FOR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0409202A FR2874611B1 (en) 2004-08-31 2004-08-31 NOVEL IMIDAZOPYRIDINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Publications (2)

Publication Number Publication Date
FR2874611A1 true FR2874611A1 (en) 2006-03-03
FR2874611B1 FR2874611B1 (en) 2006-11-17

Family

ID=34947773

Family Applications (1)

Application Number Title Priority Date Filing Date
FR0409202A Expired - Fee Related FR2874611B1 (en) 2004-08-31 2004-08-31 NOVEL IMIDAZOPYRIDINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Country Status (3)

Country Link
AR (1) AR050542A1 (en)
FR (1) FR2874611B1 (en)
WO (1) WO2006027474A2 (en)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2388001A2 (en) * 2006-10-13 2011-11-23 Zenyaku Kogyo Kabushikikaisha Age retardant containing heterocyclic compound having specific structure
US9241942B2 (en) 2007-06-08 2016-01-26 Mannkind Corporation IRE-1α inhibitors

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20090086641A (en) * 2006-12-08 2009-08-13 다케다 야쿠힌 고교 가부시키가이샤 Tricyclic compound and medical use thereof
EP2072516A1 (en) * 2007-12-21 2009-06-24 Santhera Pharmaceuticals (Schweiz) AG Substituted imidazopyridine derivates as Melancortin-4 receptor antagonists

Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0050563A1 (en) * 1980-10-22 1982-04-28 Synthelabo Imidazo(1,2-a)pyridine derivatives, process for their preparation and their therapeutical use
EP0092458A2 (en) * 1982-04-21 1983-10-26 Synthelabo Imidazo(1,2-a)pyridine derivatives, their preparation and use in therapeutical products
EP0172096A1 (en) * 1984-08-07 1986-02-19 Synthelabo 3-Acylaminomethylimidazo [1,2-a] pyridines, their preparation and therapeutical use
WO1989001472A1 (en) * 1987-08-17 1989-02-23 Nelson Research & Development Co. Melatonin analogues
EP0527687A2 (en) * 1991-08-13 1993-02-17 Adir Et Compagnie Novel arylethylamin derivatives, processes for their preparation and pharmaceutical compositions containing them
WO2002066478A1 (en) * 2001-02-20 2002-08-29 Astrazeneca Ab Antagonists of gonadotropin releasing hormone

Patent Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0050563A1 (en) * 1980-10-22 1982-04-28 Synthelabo Imidazo(1,2-a)pyridine derivatives, process for their preparation and their therapeutical use
EP0092458A2 (en) * 1982-04-21 1983-10-26 Synthelabo Imidazo(1,2-a)pyridine derivatives, their preparation and use in therapeutical products
EP0172096A1 (en) * 1984-08-07 1986-02-19 Synthelabo 3-Acylaminomethylimidazo [1,2-a] pyridines, their preparation and therapeutical use
WO1989001472A1 (en) * 1987-08-17 1989-02-23 Nelson Research & Development Co. Melatonin analogues
EP0527687A2 (en) * 1991-08-13 1993-02-17 Adir Et Compagnie Novel arylethylamin derivatives, processes for their preparation and pharmaceutical compositions containing them
WO2002066478A1 (en) * 2001-02-20 2002-08-29 Astrazeneca Ab Antagonists of gonadotropin releasing hormone

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
TRAPANI G ET AL: "Synthesis and Binding Affinity of 2-Phenylimidazo[1,2-alpha]pyridine Derivatives for both Central and Peripheral Benzodiazepine Receptors. A New Series of High-Affinity and Selective Ligands for the Peripheral Type", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY. WASHINGTON, US, vol. 40, 1997, pages 3109 - 3118, XP002900938, ISSN: 0022-2623 *

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2388001A2 (en) * 2006-10-13 2011-11-23 Zenyaku Kogyo Kabushikikaisha Age retardant containing heterocyclic compound having specific structure
EP2388001A3 (en) * 2006-10-13 2012-01-11 Zenyaku Kogyo Kabushikikaisha Age retardant containing heterocyclic compound having specific structure
US9089561B2 (en) 2006-10-13 2015-07-28 Zenyaku Kogyo Kabushiki Kaisha Methods for treating depression, neurodegeneration, inhibiting amyloid β deposition, delaying senescence, and extending life spans with heterocyclic compounds
US9241942B2 (en) 2007-06-08 2016-01-26 Mannkind Corporation IRE-1α inhibitors
US9546149B2 (en) 2007-06-08 2017-01-17 Mannkind Corporation IRE-1α inhibitors
US9981901B2 (en) 2007-06-08 2018-05-29 Fosun Orinove Pharmatech, Inc. IRE-1α inhibitors

Also Published As

Publication number Publication date
WO2006027474A2 (en) 2006-03-16
AR050542A1 (en) 2006-11-01
WO2006027474A3 (en) 2006-06-08
FR2874611B1 (en) 2006-11-17

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Legal Events

Date Code Title Description
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Effective date: 20080430