FR2803849B1 - CHIMERIC MOLECULES FORMED FROM PSORALENE AND RETINOIDE, THEIR PREPARATION PROCESS, AND THEIR APPLICATIONS IN THE TREATMENT OF CELL HYPERPROLIFERATION CONDITIONS, ESPECIALLY PSORIASIS - Google Patents

CHIMERIC MOLECULES FORMED FROM PSORALENE AND RETINOIDE, THEIR PREPARATION PROCESS, AND THEIR APPLICATIONS IN THE TREATMENT OF CELL HYPERPROLIFERATION CONDITIONS, ESPECIALLY PSORIASIS

Info

Publication number
FR2803849B1
FR2803849B1 FR0000655A FR0000655A FR2803849B1 FR 2803849 B1 FR2803849 B1 FR 2803849B1 FR 0000655 A FR0000655 A FR 0000655A FR 0000655 A FR0000655 A FR 0000655A FR 2803849 B1 FR2803849 B1 FR 2803849B1
Authority
FR
France
Prior art keywords
retinoide
psoralene
applications
treatment
preparation process
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR0000655A
Other languages
French (fr)
Other versions
FR2803849A1 (en
Inventor
Michel Giraud
Zo Andriamialisoa
Rene Santus
E Melo Teresa Sa
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Centre National de la Recherche Scientifique CNRS
Original Assignee
Centre National de la Recherche Scientifique CNRS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Centre National de la Recherche Scientifique CNRS filed Critical Centre National de la Recherche Scientifique CNRS
Priority to FR0000655A priority Critical patent/FR2803849B1/en
Priority to PCT/FR2001/000153 priority patent/WO2001053301A1/en
Publication of FR2803849A1 publication Critical patent/FR2803849A1/en
Application granted granted Critical
Publication of FR2803849B1 publication Critical patent/FR2803849B1/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D493/00Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/16Emollients or protectives, e.g. against radiation

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Dermatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Toxicology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR0000655A 2000-01-19 2000-01-19 CHIMERIC MOLECULES FORMED FROM PSORALENE AND RETINOIDE, THEIR PREPARATION PROCESS, AND THEIR APPLICATIONS IN THE TREATMENT OF CELL HYPERPROLIFERATION CONDITIONS, ESPECIALLY PSORIASIS Expired - Fee Related FR2803849B1 (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
FR0000655A FR2803849B1 (en) 2000-01-19 2000-01-19 CHIMERIC MOLECULES FORMED FROM PSORALENE AND RETINOIDE, THEIR PREPARATION PROCESS, AND THEIR APPLICATIONS IN THE TREATMENT OF CELL HYPERPROLIFERATION CONDITIONS, ESPECIALLY PSORIASIS
PCT/FR2001/000153 WO2001053301A1 (en) 2000-01-19 2001-01-18 Chimeric molecules consisting of psoralen and retinoid, preparation method, uses thereof for treating cell hyperproliferation pathologies and in particular psoriasis

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0000655A FR2803849B1 (en) 2000-01-19 2000-01-19 CHIMERIC MOLECULES FORMED FROM PSORALENE AND RETINOIDE, THEIR PREPARATION PROCESS, AND THEIR APPLICATIONS IN THE TREATMENT OF CELL HYPERPROLIFERATION CONDITIONS, ESPECIALLY PSORIASIS

Publications (2)

Publication Number Publication Date
FR2803849A1 FR2803849A1 (en) 2001-07-20
FR2803849B1 true FR2803849B1 (en) 2002-04-19

Family

ID=8846069

Family Applications (1)

Application Number Title Priority Date Filing Date
FR0000655A Expired - Fee Related FR2803849B1 (en) 2000-01-19 2000-01-19 CHIMERIC MOLECULES FORMED FROM PSORALENE AND RETINOIDE, THEIR PREPARATION PROCESS, AND THEIR APPLICATIONS IN THE TREATMENT OF CELL HYPERPROLIFERATION CONDITIONS, ESPECIALLY PSORIASIS

Country Status (2)

Country Link
FR (1) FR2803849B1 (en)
WO (1) WO2001053301A1 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005518354A (en) * 2001-11-19 2005-06-23 コントロール・デリバリー・システムズ・インコーポレイテッド Pharmaceutical composition containing a codrug
US8383836B2 (en) * 2009-04-21 2013-02-26 Duke University Methods and systems for treating cell proliferation disorders with psoralen derivatives

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4124598A (en) * 1976-10-20 1978-11-07 Hoffmann-La Roche Inc. Psoralens
LU80347A1 (en) * 1977-10-21 1979-03-16 Goupil J 5-METHOXY-PSORALENE AS A NEW MEDICINAL PRODUCT AND SYNTHESIS
US4328239A (en) * 1979-09-10 1982-05-04 Elder Pharmaceuticals, Inc. 8-Aminoalkylpsoralens
US4294822A (en) * 1980-07-29 1981-10-13 Thomas C. Elder, Inc. 5-Aminoalkyl-4,4,8-trialkylpsoralens

Also Published As

Publication number Publication date
WO2001053301A1 (en) 2001-07-26
FR2803849A1 (en) 2001-07-20

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Legal Events

Date Code Title Description
ST Notification of lapse