FR2780971B1 - Nouveaux derives de 2-aminopyridines, leur application en tant que medicaments et compositions pharmaceutiques les contenant - Google Patents

Nouveaux derives de 2-aminopyridines, leur application en tant que medicaments et compositions pharmaceutiques les contenant

Info

Publication number
FR2780971B1
FR2780971B1 FR9808732A FR9808732A FR2780971B1 FR 2780971 B1 FR2780971 B1 FR 2780971B1 FR 9808732 A FR9808732 A FR 9808732A FR 9808732 A FR9808732 A FR 9808732A FR 2780971 B1 FR2780971 B1 FR 2780971B1
Authority
FR
France
Prior art keywords
medicaments
novel
application
pharmaceutical compositions
compositions containing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR9808732A
Other languages
English (en)
Other versions
FR2780971A1 (fr
Inventor
De Lassauniere Pierre Chabrier
Gerard Auvin
Jerry Harnett
Dominique Pons
Gerard Ulibarri
Dennis Bigg
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Ipsen Pharma SAS
Original Assignee
Societe de Conseils de Recherches et dApplications Scientifiques SCRAS SAS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Societe de Conseils de Recherches et dApplications Scientifiques SCRAS SAS filed Critical Societe de Conseils de Recherches et dApplications Scientifiques SCRAS SAS
Priority to FR9808732A priority Critical patent/FR2780971B1/fr
Priority to ARP990103182A priority patent/AR019190A1/es
Priority to MYPI99002793A priority patent/MY128840A/en
Priority to DK99929395T priority patent/DK1095020T3/da
Priority to AU46223/99A priority patent/AU756221B2/en
Priority to RU2001103646/04A priority patent/RU2226527C2/ru
Priority to DE69927033T priority patent/DE69927033T2/de
Priority to ES99929395T priority patent/ES2249015T3/es
Priority to PL99345354A priority patent/PL345354A1/xx
Priority to AT99929395T priority patent/ATE303363T1/de
Priority to US09/743,043 priority patent/US6762176B1/en
Priority to EP99929395A priority patent/EP1095020B1/fr
Priority to CA002337258A priority patent/CA2337258A1/fr
Priority to HU0105073A priority patent/HUP0105073A3/hu
Priority to JP2000559091A priority patent/JP2002520317A/ja
Priority to IL14052599A priority patent/IL140525A0/xx
Priority to PCT/FR1999/001610 priority patent/WO2000002860A1/fr
Priority to CZ20010086A priority patent/CZ299818B6/cs
Priority to TW088111513A priority patent/TW509677B/zh
Publication of FR2780971A1 publication Critical patent/FR2780971A1/fr
Priority to IL140525A priority patent/IL140525A/en
Priority to NO20010031A priority patent/NO318383B1/no
Application granted granted Critical
Publication of FR2780971B1 publication Critical patent/FR2780971B1/fr
Priority to US10/405,828 priority patent/US6727239B1/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72Nitrogen atoms
    • C07D213/73Unsubstituted amino or imino radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
FR9808732A 1998-07-08 1998-07-08 Nouveaux derives de 2-aminopyridines, leur application en tant que medicaments et compositions pharmaceutiques les contenant Expired - Fee Related FR2780971B1 (fr)

Priority Applications (22)

Application Number Priority Date Filing Date Title
FR9808732A FR2780971B1 (fr) 1998-07-08 1998-07-08 Nouveaux derives de 2-aminopyridines, leur application en tant que medicaments et compositions pharmaceutiques les contenant
ARP990103182A AR019190A1 (es) 1998-07-08 1999-06-30 Derivados de 2-aminopiridinas, productos intermedios para su preparacion, medicamentos y composiciones farmaceuticas que los contienen y su uso para preparar medicamentos
MYPI99002793A MY128840A (en) 1998-07-08 1999-07-01 Derivatives of 2-aminopyridines, their use as medicaments and pharmaceutical compositions containing them
JP2000559091A JP2002520317A (ja) 1998-07-08 1999-07-05 2−アミノピリジン誘導体、その医薬としての使用及びそれを含有する医薬組成物
RU2001103646/04A RU2226527C2 (ru) 1998-07-08 1999-07-05 Производные 2-аминопиридинов, фармацевтические композиции на их основе и промежуточные вещества
DE69927033T DE69927033T2 (de) 1998-07-08 1999-07-05 4-aminopyridinderivate, ihre verwendung als arzneimittel und diese enthaltende pharmazeutische zusammensetzungen
ES99929395T ES2249015T3 (es) 1998-07-08 1999-07-05 Derivados de 2-aminopiridinas, su utilizacion como medicamentos y composiciones farmaceuticas que los contienen.
PL99345354A PL345354A1 (en) 1998-07-08 1999-07-05 2-aminopyridine erivatives, their use as medicines and pharmaceutical compositions containing them
AT99929395T ATE303363T1 (de) 1998-07-08 1999-07-05 4-aminopyridinderivate, ihre verwendung als arzneimittel und diese enthaltende pharmazeutische zusammensetzungen
US09/743,043 US6762176B1 (en) 1998-07-08 1999-07-05 2-aminopyridine derivatives, their use as medicines and pharmaceutical compositions containing them
EP99929395A EP1095020B1 (fr) 1998-07-08 1999-07-05 Derives de 2-aminopyridines, leur utilisation en tant que medicaments et compositions pharmaceutiques les contenant
CA002337258A CA2337258A1 (fr) 1998-07-08 1999-07-05 Derives de 2-aminopyridines, leur utilisation en tant que medicaments et compositions pharmaceutiques les contenant
DK99929395T DK1095020T3 (da) 1998-07-08 1999-07-05 2-Aminopyridinderivater, deres anvendelse som lægemidler og farmaceutiske præparater, der indeholder dem
AU46223/99A AU756221B2 (en) 1998-07-08 1999-07-05 2-aminopyridine derivatives, their use as medicines and pharmaceutical compositions containing them
IL14052599A IL140525A0 (en) 1998-07-08 1999-07-05 2-aminopyridine derivatives, their use as medicines and pharmaceutical compositions containing them
PCT/FR1999/001610 WO2000002860A1 (fr) 1998-07-08 1999-07-05 Derives de 2-aminopyridines, leur utilisation en tant que medicaments et compositions pharmaceutiques les contenant
CZ20010086A CZ299818B6 (cs) 1998-07-08 1999-07-05 Deriváty 2-aminopyridinu, farmaceutické kompozices jejich obsahem a použití derivátu jako léciva
HU0105073A HUP0105073A3 (en) 1998-07-08 1999-07-05 2-aminopyridine derivatives, their use as medicines and pharmaceutical compositions containing them
TW088111513A TW509677B (en) 1998-07-08 1999-08-18 New derivatives of 2-aminopyridines, their use as medicaments and pharmaceutical compositions containing them
IL140525A IL140525A (en) 1998-07-08 2000-12-25 2-aminopyridine derivatives, their use as medicines and pharmaceutical compositions
NO20010031A NO318383B1 (no) 1998-07-08 2001-01-03 Derivater av 2-aminopyridiner, anvendelse av dem som medikamenter og farmasoytiske preparater inneholdende dem
US10/405,828 US6727239B1 (en) 1998-07-08 2003-04-02 Derivatives of 2-aminopyridines, their use as medicaments and pharmaceutical compositions containing them

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9808732A FR2780971B1 (fr) 1998-07-08 1998-07-08 Nouveaux derives de 2-aminopyridines, leur application en tant que medicaments et compositions pharmaceutiques les contenant

Publications (2)

Publication Number Publication Date
FR2780971A1 FR2780971A1 (fr) 2000-01-14
FR2780971B1 true FR2780971B1 (fr) 2001-09-28

Family

ID=9528406

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9808732A Expired - Fee Related FR2780971B1 (fr) 1998-07-08 1998-07-08 Nouveaux derives de 2-aminopyridines, leur application en tant que medicaments et compositions pharmaceutiques les contenant

Country Status (1)

Country Link
FR (1) FR2780971B1 (fr)

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2830351A1 (de) * 1978-07-11 1980-01-24 Consortium Elektrochem Ind Acylanilide
US4180574A (en) * 1978-12-26 1979-12-25 Abbott Laboratories Certain ovicidal piperazines
JPS62223173A (ja) * 1986-03-25 1987-10-01 Otsuka Pharmaceut Factory Inc ピリジルアミノフエノ−ル誘導体及びその製造方法
AU4515696A (en) * 1994-12-12 1996-07-03 Merck & Co., Inc. Substituted 2-aminopyridines as inhibitors of nitric oxide synthase
GB9506188D0 (en) * 1995-03-27 1995-05-17 Fujisawa Pharmaceutical Co Amidine derivatives
CA2197364A1 (fr) * 1996-02-15 1997-08-16 Toshikazu Suzuki Compose phenolique et methode de preparation
HN1997000027A (es) * 1996-12-06 1997-06-05 Pfizer Prod Inc Derivados de 6-fenil piridil - 2 amina

Also Published As

Publication number Publication date
FR2780971A1 (fr) 2000-01-14

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