FR2645864B1 - NOVEL 17/21 ALKYL DERIVATIVES OF 19-NOR PROGESTERONE, PROCESSES FOR OBTAINING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME - Google Patents
NOVEL 17/21 ALKYL DERIVATIVES OF 19-NOR PROGESTERONE, PROCESSES FOR OBTAINING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAMEInfo
- Publication number
- FR2645864B1 FR2645864B1 FR8904910A FR8904910A FR2645864B1 FR 2645864 B1 FR2645864 B1 FR 2645864B1 FR 8904910 A FR8904910 A FR 8904910A FR 8904910 A FR8904910 A FR 8904910A FR 2645864 B1 FR2645864 B1 FR 2645864B1
- Authority
- FR
- France
- Prior art keywords
- same
- progesterone
- novel
- processes
- pharmaceutical compositions
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
- C07J7/0005—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21
- C07J7/001—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group
- C07J7/004—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group substituted in position 17 alfa
Priority Applications (12)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR8904910A FR2645864B1 (en) | 1989-04-13 | 1989-04-13 | NOVEL 17/21 ALKYL DERIVATIVES OF 19-NOR PROGESTERONE, PROCESSES FOR OBTAINING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME |
AU55525/90A AU635739B2 (en) | 1989-04-13 | 1990-04-13 | Alkyl derivates in 17/21 of 19-nor progesterone |
KR1019900702623A KR920700219A (en) | 1989-04-13 | 1990-04-13 | 17/21 alkylated derivatives of 19-norprogesterone, their preparation and pharmaceutical compositions containing them |
TNTNSN90053A TNSN90053A1 (en) | 1989-04-13 | 1990-04-13 | PROCESS FOR OBTAINING NEW 17/21 ALKYL DERIVATIVES OF 19- NOR PROGESTERONE |
JP2506960A JPH04500523A (en) | 1989-04-13 | 1990-04-13 | Novel 17/21 alkylated derivatives of 19-norprogesterone, processes for their preparation and pharmaceutical compositions containing them |
PCT/FR1990/000270 WO1990012027A1 (en) | 1989-04-13 | 1990-04-13 | Alkyl derivates in 17/21 of 19-nor progesterone |
EP90907142A EP0437552A1 (en) | 1989-04-13 | 1990-04-13 | Alkyl derivates in 17/21 of 19-nor progesterone |
HU904373A HU208152B (en) | 1989-04-13 | 1990-04-13 | Process for producing 19-norprogesterone derivatives alkylated in 17/21-position and pharmaceutical compositions comprising such compounds |
NO905344A NO174393C (en) | 1989-04-13 | 1990-12-11 | Analogous process for the preparation of therapeutically active 6-methyl-19-nor-pregna-4,6-dienes which are 17 optionally 21-alkylated |
SU904894526A RU1836379C (en) | 1989-04-13 | 1990-12-12 | Method for obtaining 17- alkylated 6-methyl-19-norpregna-4,6-dienes and intermediate compounds of this synthesis |
FI906116A FI906116A0 (en) | 1989-04-13 | 1990-12-12 | 17/21-ALKYLERADE 19-NORPROGESTERONDERIVAT. |
OA59916A OA09632A (en) | 1989-04-13 | 1990-12-13 | New 17/21 alkyl derivatives of 19-nor progesterone, their production processes and pharmaceutical compositions containing |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR8904910A FR2645864B1 (en) | 1989-04-13 | 1989-04-13 | NOVEL 17/21 ALKYL DERIVATIVES OF 19-NOR PROGESTERONE, PROCESSES FOR OBTAINING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2645864A1 FR2645864A1 (en) | 1990-10-19 |
FR2645864B1 true FR2645864B1 (en) | 1991-07-12 |
Family
ID=9380699
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR8904910A Expired - Fee Related FR2645864B1 (en) | 1989-04-13 | 1989-04-13 | NOVEL 17/21 ALKYL DERIVATIVES OF 19-NOR PROGESTERONE, PROCESSES FOR OBTAINING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME |
Country Status (12)
Country | Link |
---|---|
EP (1) | EP0437552A1 (en) |
JP (1) | JPH04500523A (en) |
KR (1) | KR920700219A (en) |
AU (1) | AU635739B2 (en) |
FI (1) | FI906116A0 (en) |
FR (1) | FR2645864B1 (en) |
HU (1) | HU208152B (en) |
NO (1) | NO174393C (en) |
OA (1) | OA09632A (en) |
RU (1) | RU1836379C (en) |
TN (1) | TNSN90053A1 (en) |
WO (1) | WO1990012027A1 (en) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2675047B1 (en) * | 1991-04-09 | 1995-05-12 | Theramex | NOVEL ANTI-GLAUCOMATORY PHARMACEUTICAL COMPOSITIONS AND THEIR PROCESS FOR OBTAINING SAME. |
DK0593520T3 (en) * | 1991-06-18 | 2000-04-03 | Theramex | Compounds containing steroids content and their use in the treatment of glaucoma |
FR2679236B1 (en) * | 1991-07-18 | 1997-01-24 | Theramex | NOVEL STEROUIDES SUBSTITUTED IN POSITION 6, PROCESSES FOR OBTAINING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME. |
HU231125B1 (en) | 2016-12-16 | 2020-12-28 | Richter Gedeon Nyrt. | Industrial process for the preparation of nomegestrol acetate |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3361744A (en) * | 1962-07-18 | 1968-01-02 | American Cyanamid Co | Novel 17-hydrocarbon substituted progesterones, intermediates and methods of preparing the same |
FR2077877B1 (en) * | 1970-02-20 | 1974-02-01 | Roussel Uclaf | |
FR2552766B1 (en) * | 1983-10-04 | 1987-06-26 | Theramex | NEW PROCESS FOR THE PREPARATION OF DERIVATIVES FROM THE 17 A-HYDROXY 19-NOR PROGESTERONE SERIES |
AU624096B2 (en) * | 1987-10-27 | 1992-06-04 | Laboratoire Theramex S.A. | Derivatives of 19-norprogesterone, their preparation and their use |
-
1989
- 1989-04-13 FR FR8904910A patent/FR2645864B1/en not_active Expired - Fee Related
-
1990
- 1990-04-13 JP JP2506960A patent/JPH04500523A/en active Pending
- 1990-04-13 AU AU55525/90A patent/AU635739B2/en not_active Ceased
- 1990-04-13 WO PCT/FR1990/000270 patent/WO1990012027A1/en not_active Application Discontinuation
- 1990-04-13 KR KR1019900702623A patent/KR920700219A/en not_active Application Discontinuation
- 1990-04-13 TN TNTNSN90053A patent/TNSN90053A1/en unknown
- 1990-04-13 EP EP90907142A patent/EP0437552A1/en not_active Withdrawn
- 1990-04-13 HU HU904373A patent/HU208152B/en not_active IP Right Cessation
- 1990-12-11 NO NO905344A patent/NO174393C/en unknown
- 1990-12-12 RU SU904894526A patent/RU1836379C/en active
- 1990-12-12 FI FI906116A patent/FI906116A0/en not_active Application Discontinuation
- 1990-12-13 OA OA59916A patent/OA09632A/en unknown
Also Published As
Publication number | Publication date |
---|---|
AU5552590A (en) | 1990-11-05 |
RU1836379C (en) | 1993-08-23 |
FR2645864A1 (en) | 1990-10-19 |
WO1990012027A1 (en) | 1990-10-18 |
HU904373D0 (en) | 1991-06-28 |
TNSN90053A1 (en) | 1991-03-05 |
NO905344L (en) | 1991-02-01 |
KR920700219A (en) | 1992-02-19 |
EP0437552A1 (en) | 1991-07-24 |
NO174393B (en) | 1994-01-17 |
NO174393C (en) | 1994-04-27 |
HUT56579A (en) | 1991-09-30 |
AU635739B2 (en) | 1993-04-01 |
FI906116A0 (en) | 1990-12-12 |
JPH04500523A (en) | 1992-01-30 |
NO905344D0 (en) | 1990-12-11 |
HU208152B (en) | 1993-08-30 |
OA09632A (en) | 1993-04-30 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |