FR2470126A1 - Fortimicines 6'-modifiees utiles notamment comme medicaments antibiotiques, et leur procede de preparation - Google Patents

Fortimicines 6'-modifiees utiles notamment comme medicaments antibiotiques, et leur procede de preparation Download PDF

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Publication number
FR2470126A1
FR2470126A1 FR8020598A FR8020598A FR2470126A1 FR 2470126 A1 FR2470126 A1 FR 2470126A1 FR 8020598 A FR8020598 A FR 8020598A FR 8020598 A FR8020598 A FR 8020598A FR 2470126 A1 FR2470126 A1 FR 2470126A1
Authority
FR
France
Prior art keywords
fortimicin
benzyloxycarbonyl
carbamate
radical
chloroform
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
FR8020598A
Other languages
English (en)
French (fr)
Inventor
John Soloman Tadanier
Robert Hallas
Jerry Roy Martin
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Abbott Laboratories
Original Assignee
Abbott Laboratories
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Laboratories filed Critical Abbott Laboratories
Publication of FR2470126A1 publication Critical patent/FR2470126A1/fr
Pending legal-status Critical Current

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/22Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/224Cyclohexane rings substituted by at least two nitrogen atoms with only one saccharide radical directly attached to the cyclohexyl radical, e.g. destomycin, fortimicin, neamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FR8020598A 1979-09-26 1980-09-25 Fortimicines 6'-modifiees utiles notamment comme medicaments antibiotiques, et leur procede de preparation Pending FR2470126A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/079,129 US4431799A (en) 1979-09-26 1979-09-26 6'-Modified fortimicin compounds

Publications (1)

Publication Number Publication Date
FR2470126A1 true FR2470126A1 (fr) 1981-05-29

Family

ID=22148618

Family Applications (1)

Application Number Title Priority Date Filing Date
FR8020598A Pending FR2470126A1 (fr) 1979-09-26 1980-09-25 Fortimicines 6'-modifiees utiles notamment comme medicaments antibiotiques, et leur procede de preparation

Country Status (8)

Country Link
US (1) US4431799A (enExample)
JP (1) JPS5646898A (enExample)
BE (1) BE885399A (enExample)
DE (1) DE3036173A1 (enExample)
ES (1) ES8200117A1 (enExample)
FR (1) FR2470126A1 (enExample)
GB (1) GB2061265A (enExample)
GR (1) GR70195B (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6042394A (ja) * 1983-08-18 1985-03-06 Kowa Co 新規なアミノグリコシド及びその製法

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2010805A (en) * 1977-12-21 1979-07-04 Abbott Lab 6'-epi-fortimicin a and b derivatives
GB2010838A (en) * 1977-12-21 1979-07-04 Abbott Lab 2-deoxyfortimicin b and intermediates therefor

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4091032A (en) * 1976-09-23 1978-05-23 Abbott Laboratories 4-N-acylfortimicin B derivatives and the chemical conversion of fortimicin B to fortimicin A

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2010805A (en) * 1977-12-21 1979-07-04 Abbott Lab 6'-epi-fortimicin a and b derivatives
GB2010838A (en) * 1977-12-21 1979-07-04 Abbott Lab 2-deoxyfortimicin b and intermediates therefor

Also Published As

Publication number Publication date
DE3036173A1 (de) 1981-04-16
ES495310A0 (es) 1981-10-16
ES8200117A1 (es) 1981-10-16
GR70195B (enExample) 1982-08-31
GB2061265A (en) 1981-05-13
BE885399A (fr) 1981-03-25
JPS5646898A (en) 1981-04-28
US4431799A (en) 1984-02-14

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