FR2430935A1 - Procede d'activation d'acides carboxyliques - Google Patents

Procede d'activation d'acides carboxyliques

Info

Publication number
FR2430935A1
FR2430935A1 FR7918215A FR7918215A FR2430935A1 FR 2430935 A1 FR2430935 A1 FR 2430935A1 FR 7918215 A FR7918215 A FR 7918215A FR 7918215 A FR7918215 A FR 7918215A FR 2430935 A1 FR2430935 A1 FR 2430935A1
Authority
FR
France
Prior art keywords
carboxylic acid
activation process
acid activation
carboxylic acids
oxazolidinone
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
FR7918215A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Antibioticos SA
Original Assignee
Antibioticos SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Antibioticos SA filed Critical Antibioticos SA
Publication of FR2430935A1 publication Critical patent/FR2430935A1/fr
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C07D213/82—Amides; Imides in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C201/00—Preparation of esters of nitric or nitrous acid or of compounds containing nitro or nitroso groups bound to a carbon skeleton
    • C07C201/06—Preparation of nitro compounds
    • C07C201/12—Preparation of nitro compounds by reactions not involving the formation of nitro groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/49—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups
    • C07C205/57—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/02—Preparation of carboxylic acid amides from carboxylic acids or from esters, anhydrides, or halides thereof by reaction with ammonia or amines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C253/00—Preparation of carboxylic acid nitriles
    • C07C253/30—Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00—Preparation of carboxylic acid esters
    • C07C67/08—Preparation of carboxylic acid esters by reacting carboxylic acids or symmetrical anhydrides with the hydroxy or O-metal group of organic compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04—Five-membered rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/24—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6527—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07F9/653—Five-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Cephalosporin Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)

Abstract

Procédé d'activation d'acides carboxyliques, utile pour la transformation ultérieure desdits acides carboxyliques en leurs esters ou amides correspondants, caractérisé par les étapes suivantes : a. On fait réagir un équivalent d'une 2-oxazolidinone de formule générale :
FR7918215A 1978-07-15 1979-07-13 Procede d'activation d'acides carboxyliques Pending FR2430935A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES471783A ES471783A1 (es) 1978-07-15 1978-07-15 Procedimiento de preparacion de n,n-bis-(3-oxazolidinil-2- ona) fosforanos-p-triclorados para su aplicacion a la obten-cion de amidas y esteres

Publications (1)

Publication Number Publication Date
FR2430935A1 true FR2430935A1 (fr) 1980-02-08

Family

ID=8476492

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7918215A Pending FR2430935A1 (fr) 1978-07-15 1979-07-13 Procede d'activation d'acides carboxyliques

Country Status (5)

Country Link
JP (1) JPS5533470A (fr)
DE (1) DE2927536A1 (fr)
ES (1) ES471783A1 (fr)
FR (1) FR2430935A1 (fr)
GB (1) GB2028331A (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3140141A1 (de) * 1981-10-09 1983-04-28 Hoechst Ag, 6230 Frankfurt Verfahren zur herstellung eines azopigments
JPS61159451A (ja) * 1985-01-08 1986-07-19 Toshiba Silicone Co Ltd ポリオルガノシロキサン組成物

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2234310A1 (en) * 1973-06-21 1975-01-17 Castro Bernard Azido-tris (dialkylamino) phosphonium salts - as peptide-coupling agents giving high yields
DE2701751A1 (de) * 1976-01-20 1977-07-21 Antibioticos Sa Verfahren zur acylierung von 6-aminopenicillansaeure, 7-aminocephalosporansaeure und 7-aminodesacetoxycephalosporansaeure sowie deren derivaten
FR2400031A1 (fr) * 1977-08-11 1979-03-09 Antibioticos Sa N,n'-bis-(3-oxalidinyl-2-one)-phosphoramides p-substitues et procede pour leur obtention

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2234310A1 (en) * 1973-06-21 1975-01-17 Castro Bernard Azido-tris (dialkylamino) phosphonium salts - as peptide-coupling agents giving high yields
DE2701751A1 (de) * 1976-01-20 1977-07-21 Antibioticos Sa Verfahren zur acylierung von 6-aminopenicillansaeure, 7-aminocephalosporansaeure und 7-aminodesacetoxycephalosporansaeure sowie deren derivaten
FR2400031A1 (fr) * 1977-08-11 1979-03-09 Antibioticos Sa N,n'-bis-(3-oxalidinyl-2-one)-phosphoramides p-substitues et procede pour leur obtention

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
CA1979 *

Also Published As

Publication number Publication date
ES471783A1 (es) 1979-10-16
DE2927536A1 (de) 1980-01-31
JPH0129775B2 (fr) 1989-06-14
JPS5533470A (en) 1980-03-08
GB2028331A (en) 1980-03-05

Similar Documents

Publication Publication Date Title
BE830297A (fr) Procede de production d'acides insatures a partir des aldehydes correspondants
FR2442227A1 (fr) Procede de production d'acides threo-3-amino-2-hydroxybutanoylaminoacetiques
FR2274595A1 (fr) Procede pour la preparation d'acides carboxyliques a partir d'halogenures organiques
FR2405245A1 (fr) Insecticides et acaricides a base de carboxylates de benzyl-pyrrolyl-methyle
FR2398713A1 (fr) Procede pour la preparation d'acides a-hydroxycarboxyliques optiquement actifs
FR2327215A1 (fr) Procede d'obtention d'acides carboxyliques a partir de leurs solutions aqueuses
FR2383907A1 (fr) Procede de preparation de derives de l'acide acetique et derives obtenus par ce procede
FR2368488A1 (fr) Procede pour la preparation de methoxypsoralene
FR2369287A1 (fr) Procede de preparation de derives organiques d'etain d'esters mercaptoalcooliques
FR2386502A1 (fr) Procede pour conferer a un produit en vermiculite de la stabilite a l'egard de l'eau
FR2376120A1 (fr) Procede de preparation d'esters d'alcoyle inferieur d'acides cis ou trans 3-formyl cyclopropane 1-carboxyliques 2,2-disubstitues racemiques
PT73314A (fr) Procede pour la fabrication de l'acide beta-hydroxybutyrique etde ses oligocondensats
NO873248L (no) FremgangsmŸte for fremstilling av kinolincarboxylsyrer.
FR2430935A1 (fr) Procede d'activation d'acides carboxyliques
FR2368479A1 (fr) Procede pour monoacyler des acides aminohydroxynaphtalene-sulfoniques avec une 2,4,6-trifluoro-s-triazine
FR2432015A1 (fr) Composes derives de l'acide cyclohexylcarboxylique et leur procede de preparation
BE821703A (fr) Procede de production d'acide acetique par oxydation en phase gazeuse
FR2354339A1 (fr) Procede de preparation d'acides 1-aminoalcane-1,1-diphosphoniques
FR2400020A1 (fr) Procede pour la preparation de furannones
FR2361341A1 (fr) Procede de preparation d'esters de l'acide anthranilique
FR2444678A2 (fr) Nouveau procede de preparation de derives du piperidyl-indole et de leurs sels
FR2395258A1 (fr) Procede pour la preparation de phenylalkylsulfones
FR2376119A1 (fr) Procede de preparation d'esters d'alcoyle inferieur d'acides trans cyclopropane-1,3-dicarboxyliques 2,2-disubstitues racemiques et nouveaux esters desdits acides
BE861207A (fr) Procede de preparation d'acide 6-aminopenicillanique par transformation enzymatique d'une penicilline
FR2359133A1 (fr) Procede de preparation de (vinyl 2,2-disubstitue)-g-butyrolactones