FR2381037A2 - NEW HYDROXYMETHYL-5 OXAZOLIDINONES-2, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION - Google Patents

NEW HYDROXYMETHYL-5 OXAZOLIDINONES-2, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION

Info

Publication number
FR2381037A2
FR2381037A2 FR7726105A FR7726105A FR2381037A2 FR 2381037 A2 FR2381037 A2 FR 2381037A2 FR 7726105 A FR7726105 A FR 7726105A FR 7726105 A FR7726105 A FR 7726105A FR 2381037 A2 FR2381037 A2 FR 2381037A2
Authority
FR
France
Prior art keywords
oxazolidinones
preparation process
therapeutic application
new
hydroxymethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7726105A
Other languages
French (fr)
Other versions
FR2381037B2 (en
Inventor
Philippe Dostert
Colette Douzon
Guy Bourgery
Claude Gouret
Gisele Mocquet
Jean-Alain Coston
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Delalande SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from CH219177A external-priority patent/CH618975A5/fr
Application filed by Delalande SA filed Critical Delalande SA
Priority to BE78189699A priority Critical patent/BE869521R/en
Priority to LU80081A priority patent/LU80081A1/en
Priority to GR56962A priority patent/GR64146B/en
Priority to US05/932,212 priority patent/US4250318A/en
Priority to CH861378A priority patent/CH634836A5/en
Priority to GB7833478A priority patent/GB2003151B/en
Priority to ZA00784685A priority patent/ZA784685B/en
Priority to JP10082478A priority patent/JPS5441871A/en
Priority to DE19782836305 priority patent/DE2836305A1/en
Priority to SE7808804A priority patent/SE444813B/en
Priority to AU39249/78A priority patent/AU526714B2/en
Priority to CA310,018A priority patent/CA1113093A/en
Priority to ES472825A priority patent/ES472825A1/en
Priority to IT68979/78A priority patent/IT1118099B/en
Priority to MX10092378U priority patent/MX5086E/en
Priority to NL7808817A priority patent/NL7808817A/en
Publication of FR2381037A2 publication Critical patent/FR2381037A2/en
Priority to US06/174,415 priority patent/US4338451A/en
Publication of FR2381037B2 publication Critical patent/FR2381037B2/fr
Application granted granted Critical
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/18—Oxygen atoms
    • C07D263/20—Oxygen atoms attached in position 2
    • C07D263/24—Oxygen atoms attached in position 2 with hydrocarbon radicals, substituted by oxygen atoms, attached to other ring carbon atoms

Abstract

a. Nouvelles hydroxyméthyl-5 oxazolidinones-2. b. Elles répondent à la formule :at. New 5-hydroxymethyl oxazolidinones-2. b. They respond to the formula:

FR7726105A 1977-02-22 1977-08-26 NEW HYDROXYMETHYL-5 OXAZOLIDINONES-2, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION Granted FR2381037A2 (en)

Priority Applications (17)

Application Number Priority Date Filing Date Title
BE78189699A BE869521R (en) 1977-08-26 1978-08-04 NEW ARYL-3 OXAZOLIDINONES-2, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION
LU80081A LU80081A1 (en) 1977-08-26 1978-08-04 NEW HYDROXYMETHYL-5 OXAZOLIDINONES-2, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION
GR56962A GR64146B (en) 1977-08-26 1978-08-08 Method for the preparation of new hydroxymethyl-5 oxazolidinones-2
US05/932,212 US4250318A (en) 1977-08-26 1978-08-09 Novel 5-hydroxymethyl oxazolidinones, the method of preparing them and their application in therapeutics
CH861378A CH634836A5 (en) 1977-08-26 1978-08-14 HYDROXYMETHYL-5 OXAZOLIDINONES-2, MEDICINAL PRODUCT AND METHOD OF PREPARATION.
GB7833478A GB2003151B (en) 1977-08-26 1978-08-16 5-hydroxymethyl ozazolidinones the method of preparing them and their application in therapeutics
ZA00784685A ZA784685B (en) 1977-08-26 1978-08-17 Novel 5-hydroxymethyl oxazolidinones,the method of preparing them and their application in therapeutics
DE19782836305 DE2836305A1 (en) 1977-08-26 1978-08-18 5-HYDROXYMETHYL-2-OXAZOLIDINONE, METHOD OF MANUFACTURING AND MEDICINAL PRODUCTS CONTAINING IT
JP10082478A JPS5441871A (en) 1977-08-26 1978-08-18 Novel 55hydroxymethyloxazolidinons and its manufacture
SE7808804A SE444813B (en) 1977-08-26 1978-08-21 NEW 5-HYDROXIMETHYL-2-OXAZOLIDINONES
AU39249/78A AU526714B2 (en) 1977-08-26 1978-08-24 Novel 5-hydroxymethyl oxazolidinones, the method of preparing them and their application in therapeutics
CA310,018A CA1113093A (en) 1977-08-26 1978-08-24 5-hydroxymethyl 2-oxazolidinones, process for preparing same and therapeutic use thereof
ES472825A ES472825A1 (en) 1977-08-26 1978-08-24 Novel 5-hydroxymethyl oxazolidinones, the method of preparing them and their application in therapeutics
MX10092378U MX5086E (en) 1977-08-26 1978-08-25 HYDROXIMETIL-5-OXAZOLIDINONAS-2 PREPARATION PROCEDURE
IT68979/78A IT1118099B (en) 1977-08-26 1978-08-25 ORIGINAL HYDROXYMETHYL 5 OSSAZOLI DINONI 2 THEIR PREPARATION PROCEDURE AND THEIR APPLICATION IN THERAPY
NL7808817A NL7808817A (en) 1977-08-26 1978-08-25 NEW 5-HYDROXYMETHYL OXAZOLIDINONES-2, METHOD FOR THEIR PREPARATION AND THEIR USE AS A MEDICINAL PRODUCT.
US06/174,415 US4338451A (en) 1977-08-26 1980-08-01 5-Hydroxymethyl oxazolidinones

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH219177A CH618975A5 (en) 1976-03-01 1977-02-22

Publications (2)

Publication Number Publication Date
FR2381037A2 true FR2381037A2 (en) 1978-09-15
FR2381037B2 FR2381037B2 (en) 1981-05-29

Family

ID=4228019

Family Applications (3)

Application Number Title Priority Date Filing Date
FR7718075A Granted FR2380780A2 (en) 1977-02-22 1977-06-13 Psychotropic medicaments - comprising 5-hydroxymethyl-3-phenyl-2-oxazolidone derivs.
FR7726104A Granted FR2381038A2 (en) 1977-02-22 1977-08-26 NEW DERIVATIVES OF CARBAMOYLOXYMETHYL-5 OXAZOLIDINONE-2, THEIR PREPARATION PROCESS AND THEIR APPLICATION IN THERAPEUTICS
FR7726105A Granted FR2381037A2 (en) 1977-02-22 1977-08-26 NEW HYDROXYMETHYL-5 OXAZOLIDINONES-2, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION

Family Applications Before (2)

Application Number Title Priority Date Filing Date
FR7718075A Granted FR2380780A2 (en) 1977-02-22 1977-06-13 Psychotropic medicaments - comprising 5-hydroxymethyl-3-phenyl-2-oxazolidone derivs.
FR7726104A Granted FR2381038A2 (en) 1977-02-22 1977-08-26 NEW DERIVATIVES OF CARBAMOYLOXYMETHYL-5 OXAZOLIDINONE-2, THEIR PREPARATION PROCESS AND THEIR APPLICATION IN THERAPEUTICS

Country Status (1)

Country Link
FR (3) FR2380780A2 (en)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4413001A (en) * 1978-06-09 1983-11-01 Delalande S.A. N-Aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones
DE3320394A1 (en) * 1982-06-08 1983-12-08 Delalande S.A., 92400 Courbevoie, Hauts-de-Seine OPTICALLY ACTIVE N-ARYLATED OXAZOLIDINONE (2) DERIVATIVES, THE USE THEREOF AS SPECIFIC AND REVERSIBLE INHIBITORS OF MONOAMINOOXYDASE OF THE B-TYPE AND METHOD FOR THE PRODUCTION THEREOF
EP0657440A1 (en) * 1993-12-13 1995-06-14 F. Hoffmann-La Roche Ag Oxazolidine-2-one derivatives
US6166056A (en) * 1995-09-01 2000-12-26 Pharmacia Phenyloxazolidinones having a C-C bond to 4-8 membered heterocyclic rings

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4340606A (en) 1980-10-23 1982-07-20 E. I. Du Pont De Nemours And Company 3-(p-Alkylsulfonylphenyl)oxazolidinone derivatives as antibacterial agents

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2035024A1 (en) * 1969-03-18 1970-12-18 Delalande Sa

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2035024A1 (en) * 1969-03-18 1970-12-18 Delalande Sa

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4413001A (en) * 1978-06-09 1983-11-01 Delalande S.A. N-Aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones
DE3320394A1 (en) * 1982-06-08 1983-12-08 Delalande S.A., 92400 Courbevoie, Hauts-de-Seine OPTICALLY ACTIVE N-ARYLATED OXAZOLIDINONE (2) DERIVATIVES, THE USE THEREOF AS SPECIFIC AND REVERSIBLE INHIBITORS OF MONOAMINOOXYDASE OF THE B-TYPE AND METHOD FOR THE PRODUCTION THEREOF
EP0657440A1 (en) * 1993-12-13 1995-06-14 F. Hoffmann-La Roche Ag Oxazolidine-2-one derivatives
US5574055A (en) * 1993-12-13 1996-11-12 Hoffmann-La Roche Inc. Oxazolidinone derivatives
AU684319B2 (en) * 1993-12-13 1997-12-11 F. Hoffmann-La Roche Ag Oxazolidin-2-one derivatives
CN1051308C (en) * 1993-12-13 2000-04-12 弗·哈夫曼-拉罗切有限公司 Oxazolidin-2-one derivatives
US6166056A (en) * 1995-09-01 2000-12-26 Pharmacia Phenyloxazolidinones having a C-C bond to 4-8 membered heterocyclic rings
US6358942B1 (en) 1995-09-01 2002-03-19 Pharmacia & Upjohn Company Phenyloxazolidinones having a c-c bond 4-8 membered heterocyclic rings

Also Published As

Publication number Publication date
FR2380780B2 (en) 1981-05-29
FR2381038A2 (en) 1978-09-15
FR2380780A2 (en) 1978-09-15
FR2381037B2 (en) 1981-05-29
FR2381038B2 (en) 1980-07-18

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