FR2359830A1 - 6-alcoyl-pyrimidines utilisables comme medicament, notamment contre la malaria - Google Patents

6-alcoyl-pyrimidines utilisables comme medicament, notamment contre la malaria

Info

Publication number
FR2359830A1
FR2359830A1 FR7723049A FR7723049A FR2359830A1 FR 2359830 A1 FR2359830 A1 FR 2359830A1 FR 7723049 A FR7723049 A FR 7723049A FR 7723049 A FR7723049 A FR 7723049A FR 2359830 A1 FR2359830 A1 FR 2359830A1
Authority
FR
France
Prior art keywords
alcoyl
medicinal product
especially against
against malaria
pyrimidines used
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7723049A
Other languages
English (en)
French (fr)
Other versions
FR2359830B1 (show.php
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Beecham Group PLC
Original Assignee
Beecham Group PLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beecham Group PLC filed Critical Beecham Group PLC
Publication of FR2359830A1 publication Critical patent/FR2359830A1/fr
Application granted granted Critical
Publication of FR2359830B1 publication Critical patent/FR2359830B1/fr
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FR7723049A 1976-07-29 1977-07-27 6-alcoyl-pyrimidines utilisables comme medicament, notamment contre la malaria Granted FR2359830A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB31582/76A GB1546937A (en) 1976-07-29 1976-07-29 2,4-diaminopyrimidine derivatives
BE184637A BE863314A (fr) 1976-07-29 1978-01-25 Derives enti-paludeens de la pyrimidine

Publications (2)

Publication Number Publication Date
FR2359830A1 true FR2359830A1 (fr) 1978-02-24
FR2359830B1 FR2359830B1 (show.php) 1980-06-06

Family

ID=25650545

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7723049A Granted FR2359830A1 (fr) 1976-07-29 1977-07-27 6-alcoyl-pyrimidines utilisables comme medicament, notamment contre la malaria

Country Status (7)

Country Link
US (2) US4179562A (show.php)
JP (1) JPS5318588A (show.php)
BE (1) BE863314A (show.php)
CH (1) CH637385A5 (show.php)
DE (1) DE2733001A1 (show.php)
FR (1) FR2359830A1 (show.php)
GB (1) GB1546937A (show.php)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2492821A1 (fr) * 1980-10-27 1982-04-30 May & Baker Ltd Derives de la pyrimidine, leur procede de preparation et les compositions pharmaceutiques les contenant

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5836121U (ja) * 1981-09-02 1983-03-09 株式会社吉野工業所 2軸延伸ブロ−成形壜体成形用1次成形品
PH22520A (en) * 1984-11-12 1988-10-17 Yamanouchi Pharma Co Ltd Heterocyclic compounds having 4-lover alkyl-3-hydroxy-2-lower alkyl phenoxy-lower alkylene-y-group, and process of producing them
DE4120698A1 (de) * 1991-06-22 1992-12-24 Gruenenthal Gmbh Substituierte phenoxyalkanole und deren ester, diese verbindungen enthaltende arzneimittel und verfahren zur herstellung dieser verbindungen und arzneimittel
US5322858A (en) * 1992-02-14 1994-06-21 Jacobus Pharmaceutical Co. Inc. N,N'-substituted imidodicarbonimidic diamides derived from hydroxylamines
RU95113597A (ru) * 1992-12-02 1997-06-10 ФМК Корпорейшн (US) Инсектицидная композиция, способы борьбы с насекомыми
RU2341296C2 (ru) 2002-05-24 2008-12-20 Энджиотек Интернэшнл Аг Композиции и способы покрытия медицинских имплантатов
US8313760B2 (en) 2002-05-24 2012-11-20 Angiotech International Ag Compositions and methods for coating medical implants
US7256218B2 (en) * 2002-11-22 2007-08-14 Jacobus Pharmaceutical Company, Inc. Biguanide and dihydrotriazine derivatives
TWI392678B (zh) 2004-03-26 2013-04-11 Dainippon Sumitomo Pharma Co 9-取代-8-氧基腺嘌呤化合物
JP2009542645A (ja) * 2006-07-05 2009-12-03 アストラゼネカ・アクチエボラーグ Tlr7のモジュレーターとして作用する8−オキソアデニン誘導体
TW200831105A (en) * 2006-12-14 2008-08-01 Astrazeneca Ab Novel compounds
EP2139894B1 (en) * 2007-03-19 2011-10-26 AstraZeneca AB 9-substituted-8-oxo-adenine compounds as toll-like receptor (tlr7) modulators
EP2132209B8 (en) * 2007-03-19 2014-04-16 AstraZeneca AB 9-substituted-8-oxo-adenine compounds as toll-like receptor (tlr7 ) modulators
WO2008114819A1 (ja) * 2007-03-20 2008-09-25 Dainippon Sumitomo Pharma Co., Ltd. 新規アデニン化合物
AU2008310898B2 (en) * 2007-10-08 2014-05-08 National Science and Technology Development Agency acting through National Center for Genetic Engineering and Biotechnology Antimalarial compounds with flexible side-chains
PE20091236A1 (es) * 2007-11-22 2009-09-16 Astrazeneca Ab Derivados de pirimidina como immunomoduladores de tlr7
PE20091156A1 (es) 2007-12-17 2009-09-03 Astrazeneca Ab Sales de (3-{[[3-(6-amino-2-butoxi-8-oxo-7,8-dihidro-9h-purin-9-il)propil](3-morfolin-4-ilpropil)amino]metil}fenil)acetato de metilo
BRPI1010937A2 (pt) 2009-05-21 2019-09-24 Astrazeneca Ab composto, uso de um composto, e, método para tratar câncer
GB0908772D0 (en) * 2009-05-21 2009-07-01 Astrazeneca Ab New salts 756
WO2012080728A1 (en) 2010-12-16 2012-06-21 Astrazeneca Ab Imidazo [4, 5 -c] quinolin- 1 -yl derivative useful in therapy
US8895570B2 (en) 2010-12-17 2014-11-25 Astrazeneca Ab Purine derivatives
WO2013172479A1 (en) 2012-05-18 2013-11-21 Dainippon Sumitomo Pharma Co., Ltd. Carboxylic acid compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB945160A (en) * 1960-11-29 1963-12-23 Vitamins Ltd New dihydrotriazine derivatives and a process for their manufacture
US3723429A (en) * 1969-11-06 1973-03-27 Beecham Group Ltd Di-hydro triazine derivatives

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2492821A1 (fr) * 1980-10-27 1982-04-30 May & Baker Ltd Derives de la pyrimidine, leur procede de preparation et les compositions pharmaceutiques les contenant

Also Published As

Publication number Publication date
US4232022A (en) 1980-11-04
JPS5318588A (en) 1978-02-20
US4179562A (en) 1979-12-18
BE863314A (fr) 1978-07-25
GB1546937A (en) 1979-05-31
DE2733001A1 (de) 1978-02-09
CH637385A5 (de) 1983-07-29
FR2359830B1 (show.php) 1980-06-06

Similar Documents

Publication Publication Date Title
FR2359830A1 (fr) 6-alcoyl-pyrimidines utilisables comme medicament, notamment contre la malaria
FR2370051A1 (fr) Nouveaux benzamides substitues utilisables comme medicaments
FR2360587A1 (fr) Nouveaux derives d'amino-alcoyl-furannes utiles comme medicaments
FR2387954A1 (fr) Derives de mercaptoalkylsulfonylproline et composes apparentes, et leur utilisation comme medicaments
FR2361340A1 (fr) Nouvelles anilines substituees utilisables comme medicament
FR2361868A1 (fr) Composes polycycliques
FR2387955A1 (fr) Derives de l'aniline utilisables comme medicament
FR2387986A1 (fr) Composes a cycle b-lactame, utilisables comme medicament
FR2383950A1 (fr) Penicillines utilisables comme medicament
FR2361366A1 (fr) Derives heterocycliques de la guanidine
FR2374309A1 (fr) Compose a cycle diazole utilisable comme medicament
FR2367742A1 (fr) Derives d'a-thio-alcanoiques, leur preparation et leur utilisation
FR2377997A1 (fr) Aralcoylanilines utilisables comme medicament
FR2401167A1 (fr) Derives de thienothiazine utiles comme medicaments
FR2391189A1 (fr) Derives de la 2-aminotetraline, leur preparation et leurs utilisations therapeutiques
FR2446279A1 (fr) Cis- et trans-3-aryloxy-4-hydroxypyrrolidines et leurs derives, utiles notamment en medecine veterinaire comme antidepresseurs
FR2384771A1 (fr) Derives de quinazoline utiles comme medicament
FR2374313A1 (fr) Compose a cycle triazole utilisable comme medicament
FR2355846A1 (fr) Esters de penicillines utilisables comme medicaments
FR2400005A1 (fr) Derives de l'alcool benzylique, leur procede de fabrication et leur application comme medicaments
FR2431497A1 (fr) Nouveaux derives de l'acide clavulanique, utilisables comme medicament
FR2380281A1 (fr) Nouvelles imidazo(1,5-b)-pyridazines utiles comme medicaments
FR2373537A1 (fr) Derives de la piperazine utilisables comme medicaments
FR2380272A1 (fr) Derives de la coumarine et d'indane-diode, utilisables comme medicament
FR2366289A1 (fr) Nouveaux derives de l'imidazo(5,1-a)isoquinoleine, leur preparation et leur application comme medicaments

Legal Events

Date Code Title Description
ST Notification of lapse