FR2351957A1 - Aldehyde a-cyano-cinnamique et ses derives, procede pour preparer ces composes et application a la preparation des 5-benzyl-2,4-diamino-pyrimidines - Google Patents
Aldehyde a-cyano-cinnamique et ses derives, procede pour preparer ces composes et application a la preparation des 5-benzyl-2,4-diamino-pyrimidinesInfo
- Publication number
- FR2351957A1 FR2351957A1 FR7715410A FR7715410A FR2351957A1 FR 2351957 A1 FR2351957 A1 FR 2351957A1 FR 7715410 A FR7715410 A FR 7715410A FR 7715410 A FR7715410 A FR 7715410A FR 2351957 A1 FR2351957 A1 FR 2351957A1
- Authority
- FR
- France
- Prior art keywords
- pyrimidines
- diamino
- cyano
- benzyl
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 229940058936 antimalarials diaminopyrimidines Drugs 0.000 title 1
- 229940117916 cinnamic aldehyde Drugs 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
- C07D239/49—Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
- C07D317/50—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring
- C07D317/60—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19762623169 DE2623169A1 (de) | 1976-05-22 | 1976-05-22 | Verfahren zur herstellung von 2,4- diaminopyrimidinen |
| DE19762623170 DE2623170C2 (de) | 1976-05-22 | 1976-05-22 | Verfahren zur Herstellung von α-Cyanzimtaldehyd-Derivaten und 3,4,5-Trimethoxy-α-Cyanzimtaldehyd |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2351957A1 true FR2351957A1 (fr) | 1977-12-16 |
| FR2351957B3 FR2351957B3 (OSRAM) | 1980-02-15 |
Family
ID=25770492
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7715410A Granted FR2351957A1 (fr) | 1976-05-22 | 1977-05-18 | Aldehyde a-cyano-cinnamique et ses derives, procede pour preparer ces composes et application a la preparation des 5-benzyl-2,4-diamino-pyrimidines |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US4172090A (OSRAM) |
| JP (1) | JPS52142042A (OSRAM) |
| FR (1) | FR2351957A1 (OSRAM) |
| GB (1) | GB1578265A (OSRAM) |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA617233A (en) * | 1961-03-28 | Melone Gaetano | Derivatives of cinnamaldehyde and 2-thienyl-acrolein and method of preparation thereof | |
| US3855265A (en) * | 1969-03-06 | 1974-12-17 | Burroughs Wellcome Co | 5-benzyl pyrimidines intermediates therefore, and method |
| US3833637A (en) * | 1971-11-22 | 1974-09-03 | Phillips Petroleum Co | Preparation of unsaturated nitriles |
-
1977
- 1977-05-12 US US05/796,063 patent/US4172090A/en not_active Expired - Lifetime
- 1977-05-18 FR FR7715410A patent/FR2351957A1/fr active Granted
- 1977-05-20 GB GB21261/77A patent/GB1578265A/en not_active Expired
- 1977-05-20 JP JP5777577A patent/JPS52142042A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| GB1578265A (en) | 1980-11-05 |
| JPS52142042A (en) | 1977-11-26 |
| US4172090A (en) | 1979-10-23 |
| FR2351957B3 (OSRAM) | 1980-02-15 |
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