FR2259092A1 - Anthelmintic tetramisoles prodn - by reacting an N-acylmethylaziridine with thiocyanic acid, conversion to oxime then reductive cyclisation - Google Patents
Anthelmintic tetramisoles prodn - by reacting an N-acylmethylaziridine with thiocyanic acid, conversion to oxime then reductive cyclisationInfo
- Publication number
- FR2259092A1 FR2259092A1 FR7402930A FR7402930A FR2259092A1 FR 2259092 A1 FR2259092 A1 FR 2259092A1 FR 7402930 A FR7402930 A FR 7402930A FR 7402930 A FR7402930 A FR 7402930A FR 2259092 A1 FR2259092 A1 FR 2259092A1
- Authority
- FR
- France
- Prior art keywords
- tetramisoles
- thiocyanic acid
- reacting
- acylmethylaziridine
- prodn
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- ZMZDMBWJUHKJPS-UHFFFAOYSA-N thiocyanic acid Chemical compound SC#N ZMZDMBWJUHKJPS-UHFFFAOYSA-N 0.000 title abstract 4
- 230000000507 anthelmentic effect Effects 0.000 title abstract 2
- 230000002829 reductive effect Effects 0.000 title abstract 2
- 238000006243 chemical reaction Methods 0.000 title 1
- 150000002923 oximes Chemical class 0.000 title 1
- 238000000034 method Methods 0.000 abstract 2
- REGFWZVTTFGQOJ-UHFFFAOYSA-N 4,5-dihydro-1,3-thiazol-2-amine Chemical class NC1=NCCS1 REGFWZVTTFGQOJ-UHFFFAOYSA-N 0.000 abstract 1
- AVXURJPOCDRRFD-UHFFFAOYSA-N Hydroxylamine Chemical compound ON AVXURJPOCDRRFD-UHFFFAOYSA-N 0.000 abstract 1
- 229910017912 NH2OH Inorganic materials 0.000 abstract 1
- 229940124339 anthelmintic agent Drugs 0.000 abstract 1
- 239000000921 anthelmintic agent Substances 0.000 abstract 1
- 150000001541 aziridines Chemical class 0.000 abstract 1
- 239000003638 chemical reducing agent Substances 0.000 abstract 1
- 125000002541 furyl group Chemical group 0.000 abstract 1
- 238000010438 heat treatment Methods 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- -1 picolyl Chemical group 0.000 abstract 1
- 125000004076 pyridyl group Chemical group 0.000 abstract 1
- 125000000335 thiazolyl group Chemical group 0.000 abstract 1
- 125000001544 thienyl group Chemical group 0.000 abstract 1
- 125000003944 tolyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7402930A FR2259092A1 (en) | 1974-01-29 | 1974-01-29 | Anthelmintic tetramisoles prodn - by reacting an N-acylmethylaziridine with thiocyanic acid, conversion to oxime then reductive cyclisation |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7402930A FR2259092A1 (en) | 1974-01-29 | 1974-01-29 | Anthelmintic tetramisoles prodn - by reacting an N-acylmethylaziridine with thiocyanic acid, conversion to oxime then reductive cyclisation |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2259092A1 true FR2259092A1 (en) | 1975-08-22 |
FR2259092B3 FR2259092B3 (enrdf_load_html_response) | 1976-11-19 |
Family
ID=9134150
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7402930A Granted FR2259092A1 (en) | 1974-01-29 | 1974-01-29 | Anthelmintic tetramisoles prodn - by reacting an N-acylmethylaziridine with thiocyanic acid, conversion to oxime then reductive cyclisation |
Country Status (1)
Country | Link |
---|---|
FR (1) | FR2259092A1 (enrdf_load_html_response) |
-
1974
- 1974-01-29 FR FR7402930A patent/FR2259092A1/fr active Granted
Also Published As
Publication number | Publication date |
---|---|
FR2259092B3 (enrdf_load_html_response) | 1976-11-19 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |