FR2253503A2 - Ethylenic piperonal alcohols and ketones - anxiolytics, antidepressants, hypnotics and tranquillisers - Google Patents

Ethylenic piperonal alcohols and ketones - anxiolytics, antidepressants, hypnotics and tranquillisers

Info

Publication number
FR2253503A2
FR2253503A2 FR7343938A FR7343938A FR2253503A2 FR 2253503 A2 FR2253503 A2 FR 2253503A2 FR 7343938 A FR7343938 A FR 7343938A FR 7343938 A FR7343938 A FR 7343938A FR 2253503 A2 FR2253503 A2 FR 2253503A2
Authority
FR
France
Prior art keywords
tranquillisers
piperonal
anxiolytics
hypnotics
antidepressants
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7343938A
Other languages
French (fr)
Other versions
FR2253503B2 (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Unicler
Original Assignee
Unicler
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Unicler filed Critical Unicler
Priority to FR7343938A priority Critical patent/FR2253503A2/en
Publication of FR2253503A2 publication Critical patent/FR2253503A2/en
Application granted granted Critical
Publication of FR2253503B2 publication Critical patent/FR2253503B2/fr
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D317/00Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/62Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring
    • C07D317/64Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D317/00Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/50Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring
    • C07D317/54Radicals substituted by oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D317/00Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/62Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring

Abstract

Piperonal derivs. have formula (I): (where R1=H, R2=OH, R3=H, halogen, OH, NO2 or CH3O, R4=alkyl, of 1-6C, opt. substd. by OH or phenyl which may be substd. by one or more methyl, hydroxy, methoxy or allyloxy gps., but when R3=H, R4 is not = tert. butyl). The cpds. have activity on the central nervous system, esp. as anxiolytics, antidepressants, hypnotics, and tranquillisers.
FR7343938A 1973-12-10 1973-12-10 Ethylenic piperonal alcohols and ketones - anxiolytics, antidepressants, hypnotics and tranquillisers Granted FR2253503A2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FR7343938A FR2253503A2 (en) 1973-12-10 1973-12-10 Ethylenic piperonal alcohols and ketones - anxiolytics, antidepressants, hypnotics and tranquillisers

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7343938A FR2253503A2 (en) 1973-12-10 1973-12-10 Ethylenic piperonal alcohols and ketones - anxiolytics, antidepressants, hypnotics and tranquillisers

Publications (2)

Publication Number Publication Date
FR2253503A2 true FR2253503A2 (en) 1975-07-04
FR2253503B2 FR2253503B2 (en) 1977-04-22

Family

ID=9128948

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7343938A Granted FR2253503A2 (en) 1973-12-10 1973-12-10 Ethylenic piperonal alcohols and ketones - anxiolytics, antidepressants, hypnotics and tranquillisers

Country Status (1)

Country Link
FR (1) FR2253503A2 (en)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2670781A1 (en) * 1990-12-21 1992-06-26 Roussel Uclaf New alpha -methylene-6-(styryl)phenylacrylic acid derivatives, process for their preparation and their application as pesticides
JP2016537435A (en) * 2013-11-20 2016-12-01 ビオコデ Pharmacological treatment of obsessive-compulsive disorder
JP2016540815A (en) * 2013-12-18 2016-12-28 ビオコデ Benzodioxole derivatives for use in the treatment of attention deficit and / or hyperactivity
WO2022025242A1 (en) * 2020-07-31 2022-02-03 国立大学法人 岡山大学 Novel stiripentol derivative and use thereof

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2399426A1 (en) 1977-08-04 1979-03-02 Unicler A-BENZYLIDENE-CYCLOALCANONES AND CORRESPONDING ALCOHOLS AND THEIR APPLICATION IN THERAPEUTICS

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2670781A1 (en) * 1990-12-21 1992-06-26 Roussel Uclaf New alpha -methylene-6-(styryl)phenylacrylic acid derivatives, process for their preparation and their application as pesticides
JP2016537435A (en) * 2013-11-20 2016-12-01 ビオコデ Pharmacological treatment of obsessive-compulsive disorder
US10696647B2 (en) 2013-11-20 2020-06-30 Biocodex Pharmacological treatment of obsessive-compulsive disorder
JP2016540815A (en) * 2013-12-18 2016-12-28 ビオコデ Benzodioxole derivatives for use in the treatment of attention deficit and / or hyperactivity
WO2022025242A1 (en) * 2020-07-31 2022-02-03 国立大学法人 岡山大学 Novel stiripentol derivative and use thereof

Also Published As

Publication number Publication date
FR2253503B2 (en) 1977-04-22

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