FR2243195A1 - 2,4-Diamino-6-sulphamoyl quinazolines - with antibacterial and antiparasitic activity - Google Patents
2,4-Diamino-6-sulphamoyl quinazolines - with antibacterial and antiparasitic activityInfo
- Publication number
- FR2243195A1 FR2243195A1 FR7430042A FR7430042A FR2243195A1 FR 2243195 A1 FR2243195 A1 FR 2243195A1 FR 7430042 A FR7430042 A FR 7430042A FR 7430042 A FR7430042 A FR 7430042A FR 2243195 A1 FR2243195 A1 FR 2243195A1
- Authority
- FR
- France
- Prior art keywords
- opt
- antibacterial
- sulphamoyl
- quinazolines
- diamino
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 230000000844 anti-bacterial effect Effects 0.000 title abstract 2
- 230000002141 anti-parasite Effects 0.000 title abstract 2
- UCZFGQIYPGPGAX-UHFFFAOYSA-N 2,4-diaminoquinazoline-6-sulfonamide Chemical class C1=C(S(N)(=O)=O)C=CC2=NC(N)=NC(N)=C21 UCZFGQIYPGPGAX-UHFFFAOYSA-N 0.000 title 1
- 125000004450 alkenylene group Chemical group 0.000 abstract 2
- 241000224017 Plasmodium berghei Species 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000002947 alkylene group Chemical group 0.000 abstract 1
- 230000036772 blood pressure Effects 0.000 abstract 1
- WHTVZRBIWZFKQO-UHFFFAOYSA-N chloroquine Chemical compound ClC1=CC=C2C(NC(C)CCCN(CC)CC)=CC=NC2=C1 WHTVZRBIWZFKQO-UHFFFAOYSA-N 0.000 abstract 1
- 230000003247 decreasing effect Effects 0.000 abstract 1
- 230000001882 diuretic effect Effects 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 125000005842 heteroatom Chemical group 0.000 abstract 1
- 201000004792 malaria Diseases 0.000 abstract 1
- 239000000463 material Substances 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
- C07D295/26—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH1281673 | 1973-09-06 | ||
| CH983974 | 1974-07-17 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2243195A1 true FR2243195A1 (en) | 1975-04-04 |
| FR2243195B1 FR2243195B1 (https=) | 1977-03-25 |
Family
ID=25705395
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7430042A Granted FR2243195A1 (en) | 1973-09-06 | 1974-09-04 | 2,4-Diamino-6-sulphamoyl quinazolines - with antibacterial and antiparasitic activity |
Country Status (7)
| Country | Link |
|---|---|
| AU (1) | AU7296174A (https=) |
| DE (1) | DE2441959A1 (https=) |
| DK (1) | DK408574A (https=) |
| FR (1) | FR2243195A1 (https=) |
| NL (1) | NL7411179A (https=) |
| OA (1) | OA04773A (https=) |
| SE (1) | SE7410216L (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2002012189A1 (en) * | 2000-08-09 | 2002-02-14 | Mitsubishi Pharma Corporation | Fused bicyclic amide compounds and medicinal use thereof |
| PA8539401A1 (es) * | 2001-02-14 | 2002-10-28 | Warner Lambert Co | Quinazolinas como inhibidores de mmp-13 |
-
1974
- 1974-07-31 DK DK408574*A patent/DK408574A/da unknown
- 1974-08-09 SE SE7410216A patent/SE7410216L/xx unknown
- 1974-08-21 NL NL7411179A patent/NL7411179A/xx unknown
- 1974-09-02 DE DE2441959A patent/DE2441959A1/de active Pending
- 1974-09-04 FR FR7430042A patent/FR2243195A1/fr active Granted
- 1974-09-04 AU AU72961/74A patent/AU7296174A/en not_active Expired
- 1974-09-05 OA OA55288A patent/OA04773A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NL7411179A (nl) | 1975-03-10 |
| FR2243195B1 (https=) | 1977-03-25 |
| OA04773A (fr) | 1980-08-31 |
| AU7296174A (en) | 1976-03-11 |
| DK408574A (https=) | 1975-05-05 |
| SE7410216L (https=) | 1975-03-07 |
| DE2441959A1 (de) | 1975-03-13 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ST | Notification of lapse |