FR2229415A1 - 5-Benzoyl-4-alkylamino-pyrazolo(3,4-b)-pyridines - as anti inflammatory agents with low diuretic activity - Google Patents

5-Benzoyl-4-alkylamino-pyrazolo(3,4-b)-pyridines - as anti inflammatory agents with low diuretic activity

Info

Publication number
FR2229415A1
FR2229415A1 FR7417292A FR7417292A FR2229415A1 FR 2229415 A1 FR2229415 A1 FR 2229415A1 FR 7417292 A FR7417292 A FR 7417292A FR 7417292 A FR7417292 A FR 7417292A FR 2229415 A1 FR2229415 A1 FR 2229415A1
Authority
FR
France
Prior art keywords
benzoyl
pyrazolo
pyridines
alkylamino
inflammatory agents
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7417292A
Other languages
French (fr)
Other versions
FR2229415B1 (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ER Squibb and Sons LLC
Original Assignee
ER Squibb and Sons LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ER Squibb and Sons LLC filed Critical ER Squibb and Sons LLC
Publication of FR2229415A1 publication Critical patent/FR2229415A1/en
Application granted granted Critical
Publication of FR2229415B1 publication Critical patent/FR2229415B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10—Antioedematous agents; Diuretics

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Cpds. (I): (where R' and R" are H or Me; R"' is H, halogen, 1-4 C-alkyl or -alkoxy and the dotted line represent a bond or 2 H atoms) are prepd. by reacting a 4-X-5-benzoylpyrazolopipidine (where X is Cl, Br or alkoxy) with an amine. Thus (I, R' = Me, R" = Et, R"' = H) is prepd. from 5-benzoyl-4-ethoxy-1H-pipazolo 3,4-b pyridine and sec.-butylamine.
FR7417292A 1973-05-17 1974-05-17 5-Benzoyl-4-alkylamino-pyrazolo(3,4-b)-pyridines - as anti inflammatory agents with low diuretic activity Granted FR2229415A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US36112073A 1973-05-17 1973-05-17

Publications (2)

Publication Number Publication Date
FR2229415A1 true FR2229415A1 (en) 1974-12-13
FR2229415B1 FR2229415B1 (en) 1977-07-08

Family

ID=23420728

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7417292A Granted FR2229415A1 (en) 1973-05-17 1974-05-17 5-Benzoyl-4-alkylamino-pyrazolo(3,4-b)-pyridines - as anti inflammatory agents with low diuretic activity

Country Status (19)

Country Link
JP (1) JPS5714674B2 (en)
AR (1) AR201145A1 (en)
AT (1) AT336015B (en)
BE (1) BE815200A (en)
CA (1) CA997351A (en)
CH (1) CH594666A5 (en)
DD (1) DD111379A5 (en)
DE (1) DE2423060A1 (en)
ES (1) ES426359A1 (en)
FI (1) FI55660C (en)
FR (1) FR2229415A1 (en)
HU (1) HU168565B (en)
IL (1) IL44744A (en)
NL (1) NL7406559A (en)
NO (1) NO140062C (en)
PL (1) PL91641B1 (en)
SE (1) SE395150B (en)
SU (1) SU501675A3 (en)
YU (1) YU136874A (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5030665B1 (en) * 1971-04-19 1975-10-02
JPS5539378B1 (en) * 1971-11-22 1980-10-11
JPS5199554U (en) * 1975-02-07 1976-08-10
JPS53130740A (en) * 1977-04-20 1978-11-15 Matsushita Electronics Corp Electrostatic coating apparatus for fluorecent substance
CH623489A5 (en) * 1977-12-08 1981-06-15 Gema Ag
JPS5719051A (en) * 1980-07-07 1982-02-01 Nippon Wagner Supureetec Kk Static painting apparatus
US4811898A (en) * 1987-09-21 1989-03-14 Nordson Corporation Electrostatic powder spray gun with adjustable deflector and electrostatic shield

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2225433A1 (en) * 1971-05-25 1972-12-07 Chemische Fabrik von Heyden GmbH, 8000 München Aminopyrazolo (3,4-b) pyridine-5-ketones with their salts, manufacturing processes therefor and pharmaceuticals therefrom

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2225433A1 (en) * 1971-05-25 1972-12-07 Chemische Fabrik von Heyden GmbH, 8000 München Aminopyrazolo (3,4-b) pyridine-5-ketones with their salts, manufacturing processes therefor and pharmaceuticals therefrom

Also Published As

Publication number Publication date
NO741752L (en) 1974-11-19
DE2423060A1 (en) 1974-12-05
JPS5018495A (en) 1975-02-26
AT336015B (en) 1977-04-12
FR2229415B1 (en) 1977-07-08
HU168565B (en) 1976-05-28
ATA413774A (en) 1976-08-15
NO140062B (en) 1979-03-19
PL91641B1 (en) 1977-03-31
CA997351A (en) 1976-09-21
BE815200A (en) 1974-11-18
NL7406559A (en) 1974-11-19
AU6861574A (en) 1975-11-06
CH594666A5 (en) 1978-01-13
YU136874A (en) 1982-06-18
IL44744A (en) 1978-06-15
SE395150B (en) 1977-08-01
NO140062C (en) 1979-07-04
IL44744A0 (en) 1974-07-31
FI150274A (en) 1974-11-18
FI55660C (en) 1979-09-10
JPS5714674B2 (en) 1982-03-25
DD111379A5 (en) 1975-02-12
FI55660B (en) 1979-05-31
ES426359A1 (en) 1976-07-01
SU501675A3 (en) 1976-01-30
AR201145A1 (en) 1975-02-14

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Legal Events

Date Code Title Description
ST Notification of lapse