FR2081371A1 - Beta-adrenergic blocking propanolamine - derivs - Google Patents
Beta-adrenergic blocking propanolamine - derivsInfo
- Publication number
- FR2081371A1 FR2081371A1 FR7045437A FR7045437A FR2081371A1 FR 2081371 A1 FR2081371 A1 FR 2081371A1 FR 7045437 A FR7045437 A FR 7045437A FR 7045437 A FR7045437 A FR 7045437A FR 2081371 A1 FR2081371 A1 FR 2081371A1
- Authority
- FR
- France
- Prior art keywords
- beta
- adrenergic blocking
- lower alkyl
- derivs
- propanolamine
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 230000000903 blocking effect Effects 0.000 title abstract 3
- WUGQZFFCHPXWKQ-UHFFFAOYSA-N Propanolamine Chemical compound NCCCO WUGQZFFCHPXWKQ-UHFFFAOYSA-N 0.000 title abstract 2
- -1 sulphonamido Chemical group 0.000 abstract 4
- 125000000217 alkyl group Chemical group 0.000 abstract 3
- 125000000816 ethylene group Chemical group [H]C([H])([*:1])C([H])([H])[*:2] 0.000 abstract 2
- 125000000325 methylidene group Chemical group [H]C([H])=* 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 206010002383 Angina Pectoris Diseases 0.000 abstract 1
- 125000000738 acetamido group Chemical group [H]C([H])([H])C(=O)N([H])[*] 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 125000003342 alkenyl group Chemical group 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 1
- 125000004466 alkoxycarbonylamino group Chemical group 0.000 abstract 1
- 206010003119 arrhythmia Diseases 0.000 abstract 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 abstract 1
- 125000001589 carboacyl group Chemical group 0.000 abstract 1
- 230000000747 cardiac effect Effects 0.000 abstract 1
- 239000007859 condensation product Substances 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 125000002485 formyl group Chemical class [H]C(*)=O 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 238000010438 heat treatment Methods 0.000 abstract 1
- 230000002093 peripheral effect Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C233/16—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Epidemiology (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB6141469 | 1969-12-17 | ||
| GB2436070A GB1279877A (en) | 1969-12-17 | 1969-12-17 | Alkanolamine derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2081371A1 true FR2081371A1 (en) | 1971-12-03 |
| FR2081371B1 FR2081371B1 (enrdf_load_stackoverflow) | 1974-09-20 |
Family
ID=26257075
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7045437A Granted FR2081371A1 (en) | 1969-12-17 | 1970-12-16 | Beta-adrenergic blocking propanolamine - derivs |
Country Status (7)
| Country | Link |
|---|---|
| JP (1) | JPS5231858B1 (enrdf_load_stackoverflow) |
| BE (1) | BE760423A (enrdf_load_stackoverflow) |
| CH (1) | CH544064A (enrdf_load_stackoverflow) |
| DE (1) | DE2062055C3 (enrdf_load_stackoverflow) |
| ES (1) | ES386554A1 (enrdf_load_stackoverflow) |
| FR (1) | FR2081371A1 (enrdf_load_stackoverflow) |
| SE (1) | SE382324B (enrdf_load_stackoverflow) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1540463A (en) * | 1976-10-07 | 1979-02-14 | Ici Ltd | Alkanolamine derivatives |
| PT71175A (fr) * | 1979-05-04 | 1980-05-01 | Continental Pharma | Procede pour preparer derives de benzimidazoles |
| DE3423429A1 (de) * | 1984-06-26 | 1986-01-02 | Beiersdorf Ag, 2000 Hamburg | Substituierte phenoxyalkylaminopropanole, verfahren zu ihrer herstellung und ihre verwendung sowie diese verbindungen enthaltende zubereitungen |
| US6451814B1 (en) * | 2000-07-17 | 2002-09-17 | Wyeth | Heterocyclic β-3 adrenergic receptor agonists |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1458635A (fr) * | 1964-09-30 | 1966-03-04 | Ici Ltd | Procédé de fabrication de nouvelles alcanolamines et de leurs dérivés |
| FR2013209A1 (enrdf_load_stackoverflow) * | 1968-07-18 | 1970-03-27 | Ici Ltd | |
| NL7007861A (enrdf_load_stackoverflow) * | 1969-05-30 | 1970-12-02 |
-
1970
- 1970-12-11 JP JP45109592A patent/JPS5231858B1/ja active Pending
- 1970-12-14 SE SE7016903A patent/SE382324B/xx unknown
- 1970-12-16 BE BE760423A patent/BE760423A/xx unknown
- 1970-12-16 FR FR7045437A patent/FR2081371A1/fr active Granted
- 1970-12-16 DE DE2062055A patent/DE2062055C3/de not_active Expired
- 1970-12-16 CH CH1866270A patent/CH544064A/fr not_active IP Right Cessation
- 1970-12-17 ES ES386554A patent/ES386554A1/es not_active Expired
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1458635A (fr) * | 1964-09-30 | 1966-03-04 | Ici Ltd | Procédé de fabrication de nouvelles alcanolamines et de leurs dérivés |
| FR2013209A1 (enrdf_load_stackoverflow) * | 1968-07-18 | 1970-03-27 | Ici Ltd | |
| NL7007861A (enrdf_load_stackoverflow) * | 1969-05-30 | 1970-12-02 |
Also Published As
| Publication number | Publication date |
|---|---|
| FR2081371B1 (enrdf_load_stackoverflow) | 1974-09-20 |
| DE2062055B2 (de) | 1978-05-24 |
| CH544064A (fr) | 1973-11-15 |
| ES386554A1 (es) | 1974-02-16 |
| DE2062055C3 (de) | 1979-01-18 |
| JPS5231858B1 (enrdf_load_stackoverflow) | 1977-08-17 |
| SE382324B (sv) | 1976-01-26 |
| BE760423A (fr) | 1971-06-16 |
| DE2062055A1 (de) | 1971-06-24 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ST | Notification of lapse |