FI942963A0 - Imidazoquinazoline compounds and their preparation and use - Google Patents

Imidazoquinazoline compounds and their preparation and use

Info

Publication number
FI942963A0
FI942963A0 FI942963A FI942963A FI942963A0 FI 942963 A0 FI942963 A0 FI 942963A0 FI 942963 A FI942963 A FI 942963A FI 942963 A FI942963 A FI 942963A FI 942963 A0 FI942963 A0 FI 942963A0
Authority
FI
Finland
Prior art keywords
preparation
imidazoquinazoline
compounds
imidazoquinazoline compounds
Prior art date
Application number
FI942963A
Other languages
Finnish (fi)
Swedish (sv)
Other versions
FI942963A (en
Inventor
Holger Claus Hansen
Marit Gustav Kristiansen
Original Assignee
Novo Nordisk As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novo Nordisk As filed Critical Novo Nordisk As
Publication of FI942963A publication Critical patent/FI942963A/en
Publication of FI942963A0 publication Critical patent/FI942963A0/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
FI942963A 1991-12-20 1994-06-20 Imidazoquinazoline compounds and their preparation and use FI942963A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DK912042A DK204291D0 (en) 1991-12-20 1991-12-20 HETEROCYCLIC RELATIONSHIPS OF THEIR PREPARATION AND USE
PCT/DK1992/000385 WO1993013103A1 (en) 1991-12-20 1992-12-18 Imidazoquinazoline compounds and their preparation and use

Publications (2)

Publication Number Publication Date
FI942963A FI942963A (en) 1994-06-20
FI942963A0 true FI942963A0 (en) 1994-06-20

Family

ID=8109668

Family Applications (1)

Application Number Title Priority Date Filing Date
FI942963A FI942963A0 (en) 1991-12-20 1994-06-20 Imidazoquinazoline compounds and their preparation and use

Country Status (12)

Country Link
EP (1) EP0619820A1 (en)
JP (1) JPH07502278A (en)
AU (1) AU673814B2 (en)
CA (1) CA2125854A1 (en)
DK (1) DK204291D0 (en)
FI (1) FI942963A0 (en)
IL (1) IL104099A (en)
NO (1) NO942301L (en)
NZ (1) NZ246558A (en)
TW (1) TW211568B (en)
WO (1) WO1993013103A1 (en)
ZA (1) ZA929770B (en)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK151890D0 (en) * 1990-06-22 1990-06-22 Ferrosan As HETEROCYCLIC RELATIONSHIPS OF THEIR PREPARATION AND USE
CN1052724C (en) * 1996-07-01 2000-05-24 瑞安大药厂股份有限公司 Optical active 2, 3-dihydro-imidazole and [1, 2-c] quinazoline derivative, preparation method and use thereof
US8053762B2 (en) 2005-12-13 2011-11-08 Lg Chem, Ltd. Imidazoquinazoline derivative, process for preparing the same, and organic electronic device using the same
US8835426B2 (en) 2007-02-26 2014-09-16 Vitae Pharmaceuticals, Inc. Cyclic urea and carbamate inhibitors of 11β-hydroxysteroid dehydrogenase 1
AR069207A1 (en) 2007-11-07 2010-01-06 Vitae Pharmaceuticals Inc CYCLIC UREAS AS INHIBITORS OF THE 11 BETA - HIDROXI-ESTEROIDE DESHIDROGENASA 1
EP2229368A1 (en) 2007-12-11 2010-09-22 Vitae Pharmaceuticals, Inc. Cyclic urea inhibitors of 11beta-hydroxysteroid dehydrogenase 1
EP2324017B1 (en) 2008-07-25 2014-12-31 Boehringer Ingelheim International GmbH INHIBITORS OF 11beta-HYDROXYSTEROID DEHYDROGENASE 1
NZ590495A (en) 2008-07-25 2012-10-26 Vitae Pharmaceuticals Inc Dihydropyridin-phenyl-3-oxazinan-2-ones as inhibitors of 11beta-hydroxysteroid dehydrogenase 1
US8637505B2 (en) 2009-02-04 2014-01-28 Boehringer Ingelheim International Gmbh Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
UA109255C2 (en) 2009-04-30 2015-08-10 Берінгер Інгельхайм Інтернешнл Гмбх Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
JP5656986B2 (en) 2009-06-11 2015-01-21 ヴァイティー ファーマシューティカルズ,インコーポレイテッド Cyclic inhibitor of 11β-hydroxysteroid dehydrogenase 1 based on 1,3-oxazinan-2-one structure
US8883778B2 (en) 2009-07-01 2014-11-11 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11 beta-hydroxysteroid dehydrogenase 1
JP5860042B2 (en) 2010-06-16 2016-02-16 ヴァイティー ファーマシューティカルズ,インコーポレイテッド Substituted 5, 6 and 7 membered heterocycles, medicaments containing such compounds and their use
WO2011161128A1 (en) 2010-06-25 2011-12-29 Boehringer Ingelheim International Gmbh Azaspirohexanones as inhibitors of 11-beta-hsd1 for the treatment of metabolic disorders
EA201300522A1 (en) 2010-11-02 2013-11-29 Бёрингер Ингельхайм Интернациональ Гмбх PHARMACEUTICAL COMBINATIONS FOR THE TREATMENT OF METABOLIC DISORDERS

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE44381T1 (en) * 1985-10-17 1989-07-15 Ferrosan As HETEROCYCLIC COMPOUNDS AND THEIR PRODUCTION AND USE.
DK155524C (en) * 1987-03-18 1989-09-11 Ferrosan As CONDENSED IMIDAZOLD DERIVATIVES AND PHARMACEUTICAL PREPARATIONS CONTAINING THESE
DK443589D0 (en) * 1989-09-08 1989-09-08 Ferrosan As HETEROCYCLIC COMPOUNDS, THEIR PREPARATION AND USE
DK151890D0 (en) * 1990-06-22 1990-06-22 Ferrosan As HETEROCYCLIC RELATIONSHIPS OF THEIR PREPARATION AND USE

Also Published As

Publication number Publication date
NZ246558A (en) 1995-07-26
ZA929770B (en) 1994-06-17
EP0619820A1 (en) 1994-10-19
NO942301D0 (en) 1994-06-17
WO1993013103A1 (en) 1993-07-08
IL104099A (en) 1996-07-23
AU3344893A (en) 1993-07-28
FI942963A (en) 1994-06-20
NO942301L (en) 1994-08-19
JPH07502278A (en) 1995-03-09
AU673814B2 (en) 1996-11-28
IL104099A0 (en) 1993-05-13
CA2125854A1 (en) 1993-07-08
DK204291D0 (en) 1991-12-20
TW211568B (en) 1993-08-21

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