FI940775A0 - process for the preparation of alpha-phenylisoserine derivatives and their use - Google Patents
process for the preparation of alpha-phenylisoserine derivatives and their useInfo
- Publication number
- FI940775A0 FI940775A0 FI940775A FI940775A FI940775A0 FI 940775 A0 FI940775 A0 FI 940775A0 FI 940775 A FI940775 A FI 940775A FI 940775 A FI940775 A FI 940775A FI 940775 A0 FI940775 A0 FI 940775A0
- Authority
- FI
- Finland
- Prior art keywords
- alpha
- preparation
- phenylisoserine derivatives
- phenylisoserine
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C231/00—Preparation of carboxylic acid amides
- C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C269/06—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups by reactions not involving the formation of carbamate groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Epoxy Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR919110398A FR2680506B1 (en) | 1991-08-19 | 1991-08-19 | PROCESS FOR THE PREPARATION OF BETA-PHENYLISOSERIN DERIVATIVES AND THEIR USE. |
PCT/FR1992/000795 WO1993004038A1 (en) | 1991-08-19 | 1992-08-17 | Process for the preparation of beta-phenylisoserine derivatives and use thereof |
Publications (2)
Publication Number | Publication Date |
---|---|
FI940775A0 true FI940775A0 (en) | 1994-02-18 |
FI940775A FI940775A (en) | 1994-02-18 |
Family
ID=9416254
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI940775A FI940775A (en) | 1991-08-19 | 1994-02-18 | Process for the preparation and use of alpha-phenylisoserine derivatives |
Country Status (16)
Country | Link |
---|---|
EP (2) | EP0599973A1 (en) |
JP (1) | JPH06510033A (en) |
AU (1) | AU2490492A (en) |
CA (1) | CA2113827A1 (en) |
CZ (1) | CZ35494A3 (en) |
FI (1) | FI940775A (en) |
FR (1) | FR2680506B1 (en) |
HU (1) | HUT68255A (en) |
MX (1) | MX9204635A (en) |
NO (1) | NO940027L (en) |
NZ (1) | NZ243972A (en) |
SK (1) | SK19094A3 (en) |
TW (1) | TW222620B (en) |
WO (1) | WO1993004038A1 (en) |
YU (1) | YU78092A (en) |
ZA (1) | ZA926189B (en) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5646176A (en) * | 1992-12-24 | 1997-07-08 | Bristol-Myers Squibb Company | Phosphonooxymethyl ethers of taxane derivatives |
US5684175A (en) * | 1993-02-05 | 1997-11-04 | Napro Biotherapeutics, Inc. | C-2' hydroxyl-benzyl protected, N-carbamate protected (2R, 3S)- 3-phenylisoserine and production process therefor |
ATE253563T1 (en) * | 1993-02-05 | 2003-11-15 | Bryn Mawr College | SYNTHESIS OF TAXOL, ITS ANALOGUES AND INTERMEDIATS WITH VARIABLE A-RING SIDE CHAINS |
US5580899A (en) * | 1995-01-09 | 1996-12-03 | The Liposome Company, Inc. | Hydrophobic taxane derivatives |
US5675025A (en) * | 1995-06-07 | 1997-10-07 | Napro Biotherapeutics, Inc. | Paclitaxel synthesis from precursor compounds and methods of producing the same |
US6051600A (en) * | 1995-09-12 | 2000-04-18 | Mayhew; Eric | Liposomal hydrolysis-promoting hydrophobic taxane derivatives |
US6107332A (en) | 1995-09-12 | 2000-08-22 | The Liposome Company, Inc. | Hydrolysis-promoting hydrophobic taxane derivatives |
US5688977A (en) * | 1996-02-29 | 1997-11-18 | Napro Biotherapeutics, Inc. | Method for docetaxel synthesis |
US6107497A (en) * | 1996-02-29 | 2000-08-22 | Napro Biotherapeutics, Inc. | Intermediate for use in docetaxel synthesis and production method therefor |
US5750737A (en) * | 1996-09-25 | 1998-05-12 | Sisti; Nicholas J. | Method for paclitaxel synthesis |
US6025516A (en) * | 1998-10-14 | 2000-02-15 | Chiragene, Inc. | Resolution of 2-hydroxy-3-amino-3-phenylpropionamide and its conversion to C-13 sidechain of taxanes |
US6452025B1 (en) | 2001-04-25 | 2002-09-17 | Napro Biotherapeutics, Inc. | Three-step conversion of protected taxane ester to paclitaxel |
DE60309847T2 (en) * | 2002-02-27 | 2007-10-18 | Ferring B.V. | INTERMEDIATE PRODUCTS AND METHOD FOR THE PRODUCTION OF HEPTAPEPTIDE OXYTOCINANALOGA |
CN104582732A (en) | 2012-06-15 | 2015-04-29 | 布里格姆及妇女医院股份有限公司 | Compositions for treating cancer and methods for making the same |
MX2016012893A (en) | 2014-04-03 | 2017-05-12 | Invictus Oncology Pvt Ltd | Supramolecular combinatorial therapeutics. |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2629818B1 (en) * | 1988-04-06 | 1990-11-16 | Centre Nat Rech Scient | PROCESS FOR THE PREPARATION OF TAXOL |
FR2629819B1 (en) * | 1988-04-06 | 1990-11-16 | Rhone Poulenc Sante | PROCESS FOR THE PREPARATION OF BACCATIN III AND DESACETYL-10 BACCATIN III DERIVATIVES |
FR2662440B1 (en) * | 1990-05-22 | 1992-07-31 | Rhone Poulenc Sante | PROCESS FOR THE STEREOSELECTIVE PREPARATION OF PHENYLISOSERIN DERIVATIVES. |
FR2662441B1 (en) * | 1990-05-22 | 1992-10-23 | Rhone Poulenc Sante | PROCESS FOR THE ENANTIOSELECTIVE PREPARATION OF PHENYLISOSERIN DERIVATIVES. |
-
1991
- 1991-08-19 FR FR919110398A patent/FR2680506B1/en not_active Expired - Fee Related
-
1992
- 1992-08-11 MX MX9204635A patent/MX9204635A/en unknown
- 1992-08-17 NZ NZ243972A patent/NZ243972A/en unknown
- 1992-08-17 CZ CS94354A patent/CZ35494A3/en unknown
- 1992-08-17 EP EP92918283A patent/EP0599973A1/en not_active Ceased
- 1992-08-17 AU AU24904/92A patent/AU2490492A/en not_active Abandoned
- 1992-08-17 WO PCT/FR1992/000795 patent/WO1993004038A1/en not_active Application Discontinuation
- 1992-08-17 HU HU9400478A patent/HUT68255A/en unknown
- 1992-08-17 ZA ZA926189A patent/ZA926189B/en unknown
- 1992-08-17 JP JP5504146A patent/JPH06510033A/en active Pending
- 1992-08-17 EP EP92402293A patent/EP0528729A1/en active Pending
- 1992-08-17 TW TW081106473A patent/TW222620B/zh active
- 1992-08-17 CA CA002113827A patent/CA2113827A1/en not_active Abandoned
- 1992-08-17 SK SK190-94A patent/SK19094A3/en unknown
- 1992-08-19 YU YU78092A patent/YU78092A/en unknown
-
1994
- 1994-01-04 NO NO940027A patent/NO940027L/en unknown
- 1994-02-18 FI FI940775A patent/FI940775A/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
AU2490492A (en) | 1993-03-16 |
YU78092A (en) | 1995-10-03 |
JPH06510033A (en) | 1994-11-10 |
NO940027D0 (en) | 1994-01-04 |
SK19094A3 (en) | 1994-09-07 |
HU9400478D0 (en) | 1994-06-28 |
CA2113827A1 (en) | 1993-03-04 |
EP0599973A1 (en) | 1994-06-08 |
HUT68255A (en) | 1995-06-28 |
MX9204635A (en) | 1993-02-01 |
ZA926189B (en) | 1993-03-01 |
FR2680506A1 (en) | 1993-02-26 |
WO1993004038A1 (en) | 1993-03-04 |
TW222620B (en) | 1994-04-21 |
CZ35494A3 (en) | 1994-07-13 |
NO940027L (en) | 1994-01-04 |
EP0528729A1 (en) | 1993-02-24 |
FI940775A (en) | 1994-02-18 |
FR2680506B1 (en) | 1994-09-02 |
NZ243972A (en) | 1994-11-25 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD | Application lapsed |