FI935117A - Nya antiinflammatoriska isoxazoliner - Google Patents

Nya antiinflammatoriska isoxazoliner Download PDF

Info

Publication number
FI935117A
FI935117A FI935117A FI935117A FI935117A FI 935117 A FI935117 A FI 935117A FI 935117 A FI935117 A FI 935117A FI 935117 A FI935117 A FI 935117A FI 935117 A FI935117 A FI 935117A
Authority
FI
Finland
Prior art keywords
isoxazoline
inflammatory
inflammatory isoxazoline
Prior art date
Application number
FI935117A
Other languages
English (en)
Other versions
FI935117A0 (fi
Inventor
Akemi Ando
Rodney William Stevens
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI935117A0 publication Critical patent/FI935117A0/fi
Publication of FI935117A publication Critical patent/FI935117A/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/04Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI935117A 1992-11-20 1993-11-18 Nya antiinflammatoriska isoxazoliner FI935117A (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP4312259A JP2738486B2 (ja) 1992-11-20 1992-11-20 抗炎症剤としての新規なイソオキサゾリン類

Publications (2)

Publication Number Publication Date
FI935117A0 FI935117A0 (fi) 1993-11-18
FI935117A true FI935117A (fi) 1994-05-21

Family

ID=18027089

Family Applications (1)

Application Number Title Priority Date Filing Date
FI935117A FI935117A (fi) 1992-11-20 1993-11-18 Nya antiinflammatoriska isoxazoliner

Country Status (9)

Country Link
US (1) US5552424A (fi)
EP (1) EP0669914A1 (fi)
JP (1) JP2738486B2 (fi)
KR (1) KR0163648B1 (fi)
CN (1) CN1035054C (fi)
AU (1) AU675256B2 (fi)
CA (1) CA2149245C (fi)
FI (1) FI935117A (fi)
WO (1) WO1994012481A1 (fi)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20030129186A1 (en) 2001-07-25 2003-07-10 Biomarin Pharmaceutical Inc. Compositions and methods for modulating blood-brain barrier transport
KR100594544B1 (ko) * 2003-08-27 2006-06-30 주식회사 엘지생명과학 이소옥사졸린 구조를 갖는 캐스파제 저해제
EP1727542A4 (en) * 2004-03-26 2009-08-05 Cytokine Pharmasciences Inc COMPOUNDS, COMPOSITIONS, METHODS OF MANUFACTURE, AND METHODS OF USE FOR INHIBITING MACROPHAGE MIGRATION INHIBITION FACTOR
SI1889198T1 (sl) 2005-04-28 2015-02-27 Proteus Digital Health, Inc. Farma-informacijski sistem
EP2063905B1 (en) 2006-09-18 2014-07-30 Raptor Pharmaceutical Inc Treatment of liver disorders by administration of receptor-associated protein (rap)-conjugates
US20080262057A1 (en) * 2007-04-20 2008-10-23 Dow Agrosciences Llc Diarylisoxazolines
DK2398500T3 (da) 2009-02-20 2019-05-13 2 Bbb Medicines B V Glutathion-baseret lægemiddelafgivelsessystem
ES2942923T3 (es) 2009-05-06 2023-06-07 Laboratory Skin Care Inc Composiciones de administración dérmica que comprenden complejos de agente activo-partículas de fosfato de calcio y métodos de uso de las mismas
US20120077778A1 (en) 2010-09-29 2012-03-29 Andrea Bourdelais Ladder-Frame Polyether Conjugates

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL81887A0 (en) * 1986-03-14 1987-10-20 Syntex Inc Dihydroisoxazole derivatives,their preparation and pharmaceutical compositions containing them
IE59813B1 (en) * 1986-05-09 1994-04-06 Warner Lambert Co Styryl pyrazoles, isoxazoles and analogs thereof having activity as 5-lipoxy-genase inhibitors and pharmaceutical compositions containing them
CA1334975C (en) * 1987-11-13 1995-03-28 James H. Holms Furan and pyrrole containing lipoxygenase inhibiting compounds
GB9012252D0 (en) * 1990-06-01 1990-07-18 Lilly Industries Ltd Pharmaceutical compounds

Also Published As

Publication number Publication date
AU5359994A (en) 1994-06-22
WO1994012481A1 (en) 1994-06-09
JPH06157485A (ja) 1994-06-03
US5552424A (en) 1996-09-03
CA2149245C (en) 1997-08-26
FI935117A0 (fi) 1993-11-18
CN1091132A (zh) 1994-08-24
KR0163648B1 (ko) 1998-12-01
AU675256B2 (en) 1997-01-30
JP2738486B2 (ja) 1998-04-08
CA2149245A1 (en) 1994-06-09
CN1035054C (zh) 1997-06-04
EP0669914A1 (en) 1995-09-06
KR950704273A (ko) 1995-11-17

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