FI912409A0 - BICYCLISKA 1-AZA CYCLOALKANER. - Google Patents
BICYCLISKA 1-AZA CYCLOALKANER.Info
- Publication number
- FI912409A0 FI912409A0 FI912409A FI912409A FI912409A0 FI 912409 A0 FI912409 A0 FI 912409A0 FI 912409 A FI912409 A FI 912409A FI 912409 A FI912409 A FI 912409A FI 912409 A0 FI912409 A0 FI 912409A0
- Authority
- FI
- Finland
- Prior art keywords
- cycloalkaner
- bicycliska
- aza
- aza cycloalkaner
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- Hospice & Palliative Care (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Psychiatry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE4016212 | 1990-05-19 | ||
DE4018886 | 1990-06-13 |
Publications (2)
Publication Number | Publication Date |
---|---|
FI912409A0 true FI912409A0 (en) | 1991-05-17 |
FI912409A FI912409A (en) | 1991-11-20 |
Family
ID=25893382
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI912409A FI912409A (en) | 1990-05-19 | 1991-05-17 | BICYCLISKA 1-AZA CYCLOALKANER. |
Country Status (14)
Country | Link |
---|---|
EP (1) | EP0458214A1 (en) |
JP (1) | JP2853837B2 (en) |
KR (1) | KR910020009A (en) |
AU (1) | AU648789B2 (en) |
CA (1) | CA2042860A1 (en) |
CZ (1) | CZ281837B6 (en) |
FI (1) | FI912409A (en) |
HU (1) | HUT58091A (en) |
IE (1) | IE911688A1 (en) |
IL (1) | IL98176A0 (en) |
NO (1) | NO911934L (en) |
PT (1) | PT97703A (en) |
SK (1) | SK279168B6 (en) |
YU (1) | YU84791A (en) |
Families Citing this family (34)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK0456519T3 (en) * | 1990-05-11 | 1994-11-07 | Sankyo Co | Piperidyloxy and quinuclidinyloxyisoxazole derivatives, their preparation and their therapeutic use |
GB9122988D0 (en) * | 1991-10-30 | 1991-12-18 | Ici Plc | Heterocyclic compounds |
GB9127279D0 (en) * | 1991-12-23 | 1992-02-19 | Ici Plc | Heterocyclic derivatives |
AU3901393A (en) * | 1992-04-10 | 1993-11-18 | Zeneca Limited | Biphenylylquinuclidine derivatives as squalene synthase inhibitors |
GB9211796D0 (en) * | 1992-06-04 | 1992-07-15 | Ici Plc | Heterocyclic derivatives |
IT1255179B (en) * | 1992-06-26 | 1995-10-20 | Enzo Cereda | AZACICLO AND AZABICICLO ALCHILIDEN IDROSSILAMINE |
GB9216721D0 (en) * | 1992-08-06 | 1992-09-23 | Ici Plc | Therapeutic heterocyclic derivatives |
GB9218334D0 (en) * | 1992-08-28 | 1992-10-14 | Ici Plc | Heterocyclic compounds |
IL107184A (en) * | 1992-10-09 | 1997-08-14 | Abbott Lab | Heterocyclic ether compounds that enhance cognitive function |
DE4236331A1 (en) * | 1992-10-28 | 1994-05-05 | Boehringer Ingelheim Kg | Synergistic combination |
GB9226573D0 (en) * | 1992-12-21 | 1993-02-17 | Ici Plc | Heterocyclic compounds |
IL109451A0 (en) * | 1993-04-29 | 1994-07-31 | Zeneca Ltd | Heterocyclic derivatives |
US5998404A (en) | 1994-10-24 | 1999-12-07 | Eli Lilly And Company | Heterocyclic compounds and their use |
US5512574A (en) * | 1994-12-21 | 1996-04-30 | American Home Products Corporation | Quinuclidine and azabicyclo 2.2.1! heptane pyrazinyl ethers as muscarinic agonists |
JPH11500113A (en) * | 1995-02-17 | 1999-01-06 | ノボ ノルディスク アクティーゼルスカブ | Use of heterocyclic compounds |
US6040442A (en) * | 1995-06-01 | 2000-03-21 | Eli Lilly And Company | Process for preparing 1,2,5-thiadiazole containing ethers |
WO1997020819A1 (en) * | 1995-12-06 | 1997-06-12 | Eli Lilly And Company | Composition for treating pain |
EP0912183A4 (en) * | 1996-04-23 | 1999-08-04 | Lilly Co Eli | Heterocyclic compounds |
AU2003250322B2 (en) * | 2002-08-14 | 2010-01-21 | Neurosearch A/S | Novel quinuclidine derivatives and their use |
GB0220581D0 (en) | 2002-09-04 | 2002-10-09 | Novartis Ag | Organic Compound |
US7750022B2 (en) | 2003-08-13 | 2010-07-06 | Neurosearch A/S | Quinuclidine derivatives and their pharmaceutical use |
US7655657B2 (en) | 2003-12-22 | 2010-02-02 | Abbott Laboratories | Fused bicycloheterocycle substituted quinuclidine derivatives |
US20050137203A1 (en) * | 2003-12-22 | 2005-06-23 | Jianguo Ji | 3-quinuclidinyl amino-substituted biaryl derivatives |
WO2006065233A1 (en) * | 2004-12-10 | 2006-06-22 | Abbott Laboratories | Fused bicycloheterocycle substituted quinuclidine derivatives |
US7160876B2 (en) | 2003-12-22 | 2007-01-09 | Abbott Laboratories | Fused bicycloheterocycle substituted quinuclidine derivatives |
PE20060437A1 (en) | 2004-06-18 | 2006-06-08 | Novartis Ag | AZA-BICYCLONONE COMPOUNDS AS CHOLINERGIC LINKS OF nAChR |
GB0415746D0 (en) | 2004-07-14 | 2004-08-18 | Novartis Ag | Organic compounds |
GB0521508D0 (en) | 2005-10-21 | 2005-11-30 | Novartis Ag | Organic compounds |
GB0525672D0 (en) | 2005-12-16 | 2006-01-25 | Novartis Ag | Organic compounds |
GB0525673D0 (en) | 2005-12-16 | 2006-01-25 | Novartis Ag | Organic compounds |
CN115135383B (en) | 2020-02-18 | 2024-06-11 | 吉利德科学公司 | Antiviral compounds |
TW202322824A (en) | 2020-02-18 | 2023-06-16 | 美商基利科學股份有限公司 | Antiviral compounds |
TW202245800A (en) | 2020-02-18 | 2022-12-01 | 美商基利科學股份有限公司 | Antiviral compounds |
AU2022256476A1 (en) | 2021-04-16 | 2023-10-12 | Gilead Sciences, Inc. | Methods of preparing carbanucleosides using amides |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE321933B (en) * | 1967-10-05 | 1970-03-23 | Astra Ab | |
FR2014831A1 (en) * | 1968-08-01 | 1970-04-24 | Sogeras | Quinuclidinyl and quinuclidinylalkyl ethers with cholino - lytic, antihistaminic and neurosedative activity |
GB8615785D0 (en) * | 1986-06-27 | 1986-08-06 | Beecham Group Plc | Compounds |
DE3854932T2 (en) * | 1987-04-15 | 1996-06-13 | Beecham Group Plc | Azabicyclene derivatives substituted on the bridgehead |
GB8718445D0 (en) * | 1987-08-04 | 1987-09-09 | Wyeth John & Brother Ltd | Pyridyl-ethers |
CA1307790C (en) * | 1987-08-04 | 1992-09-22 | Ian Anthony Cliffe | Ethers |
DE8817121U1 (en) * | 1988-11-22 | 1993-02-04 | Boehringer Ingelheim Kg, 55218 Ingelheim | New quinuclidines |
-
1991
- 1991-05-15 YU YU84791A patent/YU84791A/en unknown
- 1991-05-16 SK SK1448-91A patent/SK279168B6/en unknown
- 1991-05-16 NO NO91911934A patent/NO911934L/en unknown
- 1991-05-16 CZ CS911448A patent/CZ281837B6/en not_active IP Right Cessation
- 1991-05-17 IL IL98176A patent/IL98176A0/en unknown
- 1991-05-17 EP EP91108054A patent/EP0458214A1/en not_active Ceased
- 1991-05-17 PT PT97703A patent/PT97703A/en not_active Application Discontinuation
- 1991-05-17 HU HU911663A patent/HUT58091A/en unknown
- 1991-05-17 FI FI912409A patent/FI912409A/en not_active Application Discontinuation
- 1991-05-17 CA CA002042860A patent/CA2042860A1/en not_active Abandoned
- 1991-05-17 IE IE168891A patent/IE911688A1/en unknown
- 1991-05-17 JP JP3113418A patent/JP2853837B2/en not_active Expired - Lifetime
- 1991-05-18 KR KR1019910008106A patent/KR910020009A/en not_active Application Discontinuation
- 1991-05-20 AU AU77130/91A patent/AU648789B2/en not_active Ceased
Also Published As
Publication number | Publication date |
---|---|
KR910020009A (en) | 1991-12-19 |
CZ281837B6 (en) | 1997-02-12 |
FI912409A (en) | 1991-11-20 |
AU7713091A (en) | 1991-11-21 |
SK279168B6 (en) | 1998-07-08 |
NO911934D0 (en) | 1991-05-16 |
NO911934L (en) | 1991-11-20 |
IL98176A0 (en) | 1992-06-21 |
YU84791A (en) | 1994-06-10 |
IE911688A1 (en) | 1991-11-20 |
EP0458214A1 (en) | 1991-11-27 |
PT97703A (en) | 1992-02-28 |
HUT58091A (en) | 1992-01-28 |
CS144891A3 (en) | 1992-05-13 |
JPH04226981A (en) | 1992-08-17 |
AU648789B2 (en) | 1994-05-05 |
CA2042860A1 (en) | 1991-11-20 |
HU911663D0 (en) | 1991-11-28 |
JP2853837B2 (en) | 1999-02-03 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD | Application lapsed |