FI912409A0 - BICYCLISKA 1-AZA CYCLOALKANER. - Google Patents

BICYCLISKA 1-AZA CYCLOALKANER.

Info

Publication number
FI912409A0
FI912409A0 FI912409A FI912409A FI912409A0 FI 912409 A0 FI912409 A0 FI 912409A0 FI 912409 A FI912409 A FI 912409A FI 912409 A FI912409 A FI 912409A FI 912409 A0 FI912409 A0 FI 912409A0
Authority
FI
Finland
Prior art keywords
cycloalkaner
bicycliska
aza
aza cycloalkaner
Prior art date
Application number
FI912409A
Other languages
Finnish (fi)
Other versions
FI912409A (en
Inventor
Gerhard Kuollut-Avlide Walther
Ulrike Kuefner-Muehl
Werner Stransky
Karl-Heinz Weber
Helmut Ensinger
Franz Josef Kuhn
Enzio Mueller
Original Assignee
Boehringer Ingelheim Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Kg filed Critical Boehringer Ingelheim Kg
Publication of FI912409A0 publication Critical patent/FI912409A0/en
Publication of FI912409A publication Critical patent/FI912409A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Hospice & Palliative Care (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Psychiatry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI912409A 1990-05-19 1991-05-17 BICYCLISKA 1-AZA CYCLOALKANER. FI912409A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4016212 1990-05-19
DE4018886 1990-06-13

Publications (2)

Publication Number Publication Date
FI912409A0 true FI912409A0 (en) 1991-05-17
FI912409A FI912409A (en) 1991-11-20

Family

ID=25893382

Family Applications (1)

Application Number Title Priority Date Filing Date
FI912409A FI912409A (en) 1990-05-19 1991-05-17 BICYCLISKA 1-AZA CYCLOALKANER.

Country Status (14)

Country Link
EP (1) EP0458214A1 (en)
JP (1) JP2853837B2 (en)
KR (1) KR910020009A (en)
AU (1) AU648789B2 (en)
CA (1) CA2042860A1 (en)
CZ (1) CZ281837B6 (en)
FI (1) FI912409A (en)
HU (1) HUT58091A (en)
IE (1) IE911688A1 (en)
IL (1) IL98176A0 (en)
NO (1) NO911934L (en)
PT (1) PT97703A (en)
SK (1) SK279168B6 (en)
YU (1) YU84791A (en)

Families Citing this family (34)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK0456519T3 (en) * 1990-05-11 1994-11-07 Sankyo Co Piperidyloxy and quinuclidinyloxyisoxazole derivatives, their preparation and their therapeutic use
GB9122988D0 (en) * 1991-10-30 1991-12-18 Ici Plc Heterocyclic compounds
GB9127279D0 (en) * 1991-12-23 1992-02-19 Ici Plc Heterocyclic derivatives
AU3901393A (en) * 1992-04-10 1993-11-18 Zeneca Limited Biphenylylquinuclidine derivatives as squalene synthase inhibitors
GB9211796D0 (en) * 1992-06-04 1992-07-15 Ici Plc Heterocyclic derivatives
IT1255179B (en) * 1992-06-26 1995-10-20 Enzo Cereda AZACICLO AND AZABICICLO ALCHILIDEN IDROSSILAMINE
GB9216721D0 (en) * 1992-08-06 1992-09-23 Ici Plc Therapeutic heterocyclic derivatives
GB9218334D0 (en) * 1992-08-28 1992-10-14 Ici Plc Heterocyclic compounds
IL107184A (en) * 1992-10-09 1997-08-14 Abbott Lab Heterocyclic ether compounds that enhance cognitive function
DE4236331A1 (en) * 1992-10-28 1994-05-05 Boehringer Ingelheim Kg Synergistic combination
GB9226573D0 (en) * 1992-12-21 1993-02-17 Ici Plc Heterocyclic compounds
IL109451A0 (en) * 1993-04-29 1994-07-31 Zeneca Ltd Heterocyclic derivatives
US5998404A (en) 1994-10-24 1999-12-07 Eli Lilly And Company Heterocyclic compounds and their use
US5512574A (en) * 1994-12-21 1996-04-30 American Home Products Corporation Quinuclidine and azabicyclo 2.2.1! heptane pyrazinyl ethers as muscarinic agonists
JPH11500113A (en) * 1995-02-17 1999-01-06 ノボ ノルディスク アクティーゼルスカブ Use of heterocyclic compounds
US6040442A (en) * 1995-06-01 2000-03-21 Eli Lilly And Company Process for preparing 1,2,5-thiadiazole containing ethers
WO1997020819A1 (en) * 1995-12-06 1997-06-12 Eli Lilly And Company Composition for treating pain
EP0912183A4 (en) * 1996-04-23 1999-08-04 Lilly Co Eli Heterocyclic compounds
AU2003250322B2 (en) * 2002-08-14 2010-01-21 Neurosearch A/S Novel quinuclidine derivatives and their use
GB0220581D0 (en) 2002-09-04 2002-10-09 Novartis Ag Organic Compound
US7750022B2 (en) 2003-08-13 2010-07-06 Neurosearch A/S Quinuclidine derivatives and their pharmaceutical use
US7655657B2 (en) 2003-12-22 2010-02-02 Abbott Laboratories Fused bicycloheterocycle substituted quinuclidine derivatives
US20050137203A1 (en) * 2003-12-22 2005-06-23 Jianguo Ji 3-quinuclidinyl amino-substituted biaryl derivatives
WO2006065233A1 (en) * 2004-12-10 2006-06-22 Abbott Laboratories Fused bicycloheterocycle substituted quinuclidine derivatives
US7160876B2 (en) 2003-12-22 2007-01-09 Abbott Laboratories Fused bicycloheterocycle substituted quinuclidine derivatives
PE20060437A1 (en) 2004-06-18 2006-06-08 Novartis Ag AZA-BICYCLONONE COMPOUNDS AS CHOLINERGIC LINKS OF nAChR
GB0415746D0 (en) 2004-07-14 2004-08-18 Novartis Ag Organic compounds
GB0521508D0 (en) 2005-10-21 2005-11-30 Novartis Ag Organic compounds
GB0525672D0 (en) 2005-12-16 2006-01-25 Novartis Ag Organic compounds
GB0525673D0 (en) 2005-12-16 2006-01-25 Novartis Ag Organic compounds
CN115135383B (en) 2020-02-18 2024-06-11 吉利德科学公司 Antiviral compounds
TW202322824A (en) 2020-02-18 2023-06-16 美商基利科學股份有限公司 Antiviral compounds
TW202245800A (en) 2020-02-18 2022-12-01 美商基利科學股份有限公司 Antiviral compounds
AU2022256476A1 (en) 2021-04-16 2023-10-12 Gilead Sciences, Inc. Methods of preparing carbanucleosides using amides

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE321933B (en) * 1967-10-05 1970-03-23 Astra Ab
FR2014831A1 (en) * 1968-08-01 1970-04-24 Sogeras Quinuclidinyl and quinuclidinylalkyl ethers with cholino - lytic, antihistaminic and neurosedative activity
GB8615785D0 (en) * 1986-06-27 1986-08-06 Beecham Group Plc Compounds
DE3854932T2 (en) * 1987-04-15 1996-06-13 Beecham Group Plc Azabicyclene derivatives substituted on the bridgehead
GB8718445D0 (en) * 1987-08-04 1987-09-09 Wyeth John & Brother Ltd Pyridyl-ethers
CA1307790C (en) * 1987-08-04 1992-09-22 Ian Anthony Cliffe Ethers
DE8817121U1 (en) * 1988-11-22 1993-02-04 Boehringer Ingelheim Kg, 55218 Ingelheim New quinuclidines

Also Published As

Publication number Publication date
KR910020009A (en) 1991-12-19
CZ281837B6 (en) 1997-02-12
FI912409A (en) 1991-11-20
AU7713091A (en) 1991-11-21
SK279168B6 (en) 1998-07-08
NO911934D0 (en) 1991-05-16
NO911934L (en) 1991-11-20
IL98176A0 (en) 1992-06-21
YU84791A (en) 1994-06-10
IE911688A1 (en) 1991-11-20
EP0458214A1 (en) 1991-11-27
PT97703A (en) 1992-02-28
HUT58091A (en) 1992-01-28
CS144891A3 (en) 1992-05-13
JPH04226981A (en) 1992-08-17
AU648789B2 (en) 1994-05-05
CA2042860A1 (en) 1991-11-20
HU911663D0 (en) 1991-11-28
JP2853837B2 (en) 1999-02-03

Similar Documents

Publication Publication Date Title
FI912409A0 (en) BICYCLISKA 1-AZA CYCLOALKANER.
FI912924A (en) LADDADE ORGANISKA POLYMERMIKROPAERLOR I PAPPERSFRAMSTAELLNINGSPROCESS.
FI913886A0 (en) PRESSPARTI I EN PAPPERSMASKIN.
FI902263A0 (en) TEMPERATURKOMPENSATION I EN HELIX-RESONATOR.
FI900937A (en) ANORDNING FOER AXIALLAGRET I EN BORRMASKIN.
FI902908A0 (en) MATRISFILMSTRUKTUR I SYNNERHET FOER ELEKTROLUMINECENS DISPLAYENHET.
FI914255A (en) I UV-LJUS HAERDBAR ORGANOPOLYSIL-OXANKOMPOSITION.
FI900987A (en) ANORDNING I TRAEBEARBETNINGSMASKINER.
FI915029A (en) ANORDNING I EN ENVIRA-TORKNINGSGRUPP.
FI915058A (en) KOMBINERAT AXIAL- OCH RADIALLAGER FOER ANVAENDNING I SAENKBORRVERKTYG.
FI903165A (en) LAGRINGSSYSTEM I AUTOMATLAGER.
FI903033A (en) TAKET I EN JAERNVAEGSVAGN.
FI901282A (en) MANTELKONSTRUKTUR FOER PRESSPARTIET I EN PAPPERSMASKIN.
FI901608A0 (en) FRAMMATNINGSANORDNING FOER TRAED I SKOGSARBETSMASKINENS FLERFUNKTIONSDEL.
FI901348A0 (en) MAETNINGSFOENSTER I MAETCELL.
FI906158A (en) SAEKERHETSLAOS AVSETT FOER LUCKORNA I TVAETTMASKINSTRUMMAN.
FI905093A (en) HOERNKONSTRUKTION I TIMMERHUS.
FI912479A (en) SJAELVBORRANDE SKRUV FOER TRAEDELAR I FAESTORGAN.
FI903694A0 (en) I BACKHOPPNING ANVAENT STAOLFARTSPAOR.
FI905272A (en) I ANDNINGSSKYDD INSTAELLBAR GAS- ELLER TRYCKSKILLNADSDETEKTOR.
FI904030A0 (en) ANORDNING FOER HYDRAULISK KRETS I TRAEVARUBIL.
FI904626A (en) KYLAVDELNING FOER GLASSKIVOR I EN HAERDNINGSANLAEGGNING.
FI905877A0 (en) TELEFONNUMMERANTECKNINGSBLOCK I SKIVFORM.
FI902382A0 (en) VAENDMEKANIS FOER HJUL I MOTORCYKELS SIDOVAGN.
FI910336A0 (en) I VAEGGELEMENTPRODUKTION ANVAENDBART OEPPNINGSFORMSYSTEM.

Legal Events

Date Code Title Description
FD Application lapsed