FI883667A0 - 2 - / (4-PIPERIDINYL) METHYL / -1,2,3,4-TETRAHYDROISOKINOLINE DERIVATIVES, DERAS FRAMSTAELLNING OCH TERAPEUTISKA ANVAENDNING. - Google Patents
2 - / (4-PIPERIDINYL) METHYL / -1,2,3,4-TETRAHYDROISOKINOLINE DERIVATIVES, DERAS FRAMSTAELLNING OCH TERAPEUTISKA ANVAENDNING.Info
- Publication number
- FI883667A0 FI883667A0 FI883667A FI883667A FI883667A0 FI 883667 A0 FI883667 A0 FI 883667A0 FI 883667 A FI883667 A FI 883667A FI 883667 A FI883667 A FI 883667A FI 883667 A0 FI883667 A0 FI 883667A0
- Authority
- FI
- Finland
- Prior art keywords
- tetrahydroisokinoline
- terapeutiska
- anvaendning
- piperidinyl
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR8711288A FR2619110B1 (en) | 1987-08-07 | 1987-08-07 | ((PIPERIDINYL-4) METHYL) -2 TETRAHYDRO-1,2,3,4 ISOQUINOLEINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
FR8718342A FR2625504B2 (en) | 1987-08-07 | 1987-12-30 | ((BENZOYL-1 PIPERIDINYL-4) METHYL) -2 TETRAHYDRO-1,2,3,4 ISOQUINOLEINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
FR8805130A FR2630114B2 (en) | 1987-08-07 | 1988-04-19 | (PIPERIDINYL-4) METHYL) -2 TETRAHYDRO-1,2,3,4 ISOQUINOLEINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
FR8805129A FR2630113B2 (en) | 1987-08-07 | 1988-04-19 | ((PIPERIDINYL-4) METHYL) -2 TETRAHYDRO-1,2,3,4 ISOQUINOLEINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
Publications (2)
Publication Number | Publication Date |
---|---|
FI883667A0 true FI883667A0 (en) | 1988-08-05 |
FI883667A FI883667A (en) | 1989-02-08 |
Family
ID=27446582
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI883667A FI883667A (en) | 1987-08-07 | 1988-08-05 | 2 - / (4-PIPERIDINYL) METHYL / -1,2,3,4-TETRAHYDROISOKINOLINE DERIVATIVES, DERAS FRAMSTAELLNING OCH TERAPEUTISKA ANVAENDNING. |
Country Status (10)
Country | Link |
---|---|
US (2) | US4885302A (en) |
EP (1) | EP0306375A1 (en) |
JP (1) | JPH01100167A (en) |
KR (1) | KR890003733A (en) |
AU (1) | AU598149B2 (en) |
DK (1) | DK437588A (en) |
FI (1) | FI883667A (en) |
IL (1) | IL87339A0 (en) |
NO (1) | NO883485L (en) |
NZ (1) | NZ225708A (en) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3717561A1 (en) * | 1987-05-25 | 1988-12-08 | Thomae Gmbh Dr K | INDOL, ISOCHINOLINE AND BENZAZEPINE DERIVATIVES, MEDICINAL PRODUCTS CONTAINING THESE COMPOUNDS AND METHOD FOR THE PRODUCTION THEREOF |
IL89156A (en) * | 1988-07-12 | 1993-05-13 | Synthelabo | Derivatives of 2-((4-piperidinyl) methyl)- 1,2,3,4- tetrahydroisoquinoline, their preparation and their application in therapeutics |
US4963563A (en) * | 1989-10-13 | 1990-10-16 | Abbott Laboratories | 6-substituted-1,2,3,4-tetrahydroisoquinolines |
FR2661178B1 (en) * | 1990-04-24 | 1993-03-12 | Synthelabo | DERIVATIVES OF [(TETRAHYDRO-1,2,3,4 ISOQUINOLEINYL-2) METHYL] -4 PIPERIDINECARBOXYLATES-1 OF ALKYL, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION. |
US5096908A (en) * | 1990-05-04 | 1992-03-17 | Eli Lilly And Company | Method of inhibiting gastric acid secretion |
US5258379A (en) * | 1990-05-04 | 1993-11-02 | Eli Lilly And Company | Method of inhibiting gastric acid secretion with n-arylpiperazines |
GB9319534D0 (en) * | 1993-09-22 | 1993-11-10 | Boots Co Plc | Therapeutic agents |
FR2747386B1 (en) * | 1996-04-12 | 1998-05-15 | Synthelabo | DERIVATIVES OF 3 - [(1,2,3,4-TETRAHYDROISOQUINOLEIN-2-YL) METHYL] -8-AZABICYCLO [3.2.1] OCTANE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
WO1997049695A1 (en) * | 1996-06-25 | 1997-12-31 | Smithkline Beecham P.L.C. | Sulfonamide derivatives as 5ht7 receptor antagonists |
US5912342A (en) * | 1997-08-12 | 1999-06-15 | Heinonen; Petri | Compounds a containing a solid support |
AUPP891299A0 (en) * | 1999-02-26 | 1999-03-25 | Fujisawa Pharmaceutical Co., Ltd. | New 6-membered cyclic compounds |
US6664293B2 (en) | 1999-02-26 | 2003-12-16 | Fujiwawa Pharmaceutical Co., Ltd. | Amide compounds for the potentiation of cholinergic activity |
CL2007002958A1 (en) * | 2006-10-12 | 2008-05-09 | Epix Delaware Inc | COMPOUNDS DERIVED FROM HETEROARIL-CARBOXAMIDA, ANTAGONISTS OF THE CHEMIOQUINE RECEPTOR; PHARMACEUTICAL COMPOSITION; AND USE FOR THE TREATMENT OR PREVENTION OF SUCH DISEASES AS REJECTION OF ORGAN TRANSPLANTS, Rheumatoid Arthritis, LUPUS, ENTR |
US20100331298A1 (en) * | 2007-12-10 | 2010-12-30 | Cytopathfinder, Inc. | Carboxamide Compounds and Their Use |
EP2280766A1 (en) * | 2007-12-11 | 2011-02-09 | CytoPathfinder, Inc. | Carboxamide compounds and their use as chemokine receptor agonists |
JP6053519B2 (en) | 2009-06-26 | 2016-12-27 | サノフイ | Novel fumarate salt of histamine H3 receptor antagonist |
WO2022174083A1 (en) * | 2021-02-12 | 2022-08-18 | Recovery Therapeutics, Inc. | Compounds, compositions, and methods for modulating fgf activity |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2922786A (en) * | 1956-12-12 | 1960-01-26 | Bristol Myers Co | Therapeutic compounds |
FR1580180A (en) * | 1967-03-14 | 1969-09-05 | ||
FR7607M (en) * | 1968-04-25 | 1970-01-19 | ||
GB1250719A (en) * | 1969-03-19 | 1971-10-20 | ||
FR2426046A1 (en) * | 1978-05-18 | 1979-12-14 | Synthelabo | TETRAHYDRO-ISOQUINOLEINE DERIVATIVE, ITS PREPARATION AND THERAPEUTIC APPLICATION |
US4495354A (en) * | 1982-03-29 | 1985-01-22 | Hoffmann-La Roche Inc. | Process for bicyclic diketones |
IL89156A (en) * | 1988-07-12 | 1993-05-13 | Synthelabo | Derivatives of 2-((4-piperidinyl) methyl)- 1,2,3,4- tetrahydroisoquinoline, their preparation and their application in therapeutics |
-
1988
- 1988-08-03 EP EP88402022A patent/EP0306375A1/en not_active Withdrawn
- 1988-08-04 IL IL87339A patent/IL87339A0/en unknown
- 1988-08-05 DK DK437588A patent/DK437588A/en not_active Application Discontinuation
- 1988-08-05 NO NO88883485A patent/NO883485L/en unknown
- 1988-08-05 JP JP63197010A patent/JPH01100167A/en active Pending
- 1988-08-05 KR KR1019880010015A patent/KR890003733A/en not_active Application Discontinuation
- 1988-08-05 AU AU20475/88A patent/AU598149B2/en not_active Ceased
- 1988-08-05 NZ NZ225708A patent/NZ225708A/en unknown
- 1988-08-05 US US07/228,748 patent/US4885302A/en not_active Expired - Fee Related
- 1988-08-05 FI FI883667A patent/FI883667A/en not_active Application Discontinuation
-
1989
- 1989-08-30 US US07/400,811 patent/US4945096A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
AU598149B2 (en) | 1990-06-14 |
IL87339A0 (en) | 1989-01-31 |
US4945096A (en) | 1990-07-31 |
NZ225708A (en) | 1990-04-26 |
DK437588A (en) | 1989-03-28 |
EP0306375A1 (en) | 1989-03-08 |
NO883485D0 (en) | 1988-08-05 |
DK437588D0 (en) | 1988-08-05 |
NO883485L (en) | 1989-02-08 |
AU2047588A (en) | 1989-02-09 |
KR890003733A (en) | 1989-04-17 |
US4885302A (en) | 1989-12-05 |
FI883667A (en) | 1989-02-08 |
JPH01100167A (en) | 1989-04-18 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA | Application withdrawn |
Owner name: SYNTHELABO |