FI882945A0 - Process for the preparation of antihypertensive and antiarrhythmic trans-2,2-dimethylchroman-3-ol derivatives - Google Patents
Process for the preparation of antihypertensive and antiarrhythmic trans-2,2-dimethylchroman-3-ol derivativesInfo
- Publication number
- FI882945A0 FI882945A0 FI882945A FI882945A FI882945A0 FI 882945 A0 FI882945 A0 FI 882945A0 FI 882945 A FI882945 A FI 882945A FI 882945 A FI882945 A FI 882945A FI 882945 A0 FI882945 A0 FI 882945A0
- Authority
- FI
- Finland
- Prior art keywords
- dimethylchroman
- antiarrhythmic
- antihypertensive
- trans
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
- C07F9/65586—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system at least one of the hetero rings does not contain nitrogen as ring hetero atom
-
- C—CHEMISTRY; METALLURGY
- C10—PETROLEUM, GAS OR COKE INDUSTRIES; TECHNICAL GASES CONTAINING CARBON MONOXIDE; FUELS; LUBRICANTS; PEAT
- C10L—FUELS NOT OTHERWISE PROVIDED FOR; NATURAL GAS; SYNTHETIC NATURAL GAS OBTAINED BY PROCESSES NOT COVERED BY SUBCLASSES C10G, C10K; LIQUEFIED PETROLEUM GAS; ADDING MATERIALS TO FUELS OR FIRES TO REDUCE SMOKE OR UNDESIRABLE DEPOSITS OR TO FACILITATE SOOT REMOVAL; FIRELIGHTERS
- C10L1/00—Liquid carbonaceous fuels
- C10L1/32—Liquid carbonaceous fuels consisting of coal-oil suspensions or aqueous emulsions or oil emulsions
Applications Claiming Priority (6)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR8708830 | 1987-06-23 | ||
FR8708830A FR2617165B1 (en) | 1987-06-23 | 1987-06-23 | DIMETHYL-2, 2 CHROMANNOL-3 DERIVATIVES |
FR8800278 | 1988-01-12 | ||
FR8800278A FR2625744B1 (en) | 1988-01-12 | 1988-01-12 | 2,2-DIMETHYL DERIVATIVES CHROMANNOL-3 PROCESS FOR OBTAINING AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME |
FR8803064A FR2628424B1 (en) | 1988-03-09 | 1988-03-09 | 2,2-DIMETHYL DERIVATIVES CHROMANNOL-3 PROCESS FOR OBTAINING AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME |
FR8803064 | 1988-03-09 |
Publications (4)
Publication Number | Publication Date |
---|---|
FI882945A0 true FI882945A0 (en) | 1988-06-20 |
FI882945A FI882945A (en) | 1988-12-24 |
FI90343B FI90343B (en) | 1993-10-15 |
FI90343C FI90343C (en) | 1994-01-25 |
Family
ID=27251476
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI882945A FI90343C (en) | 1987-06-23 | 1988-06-20 | Process for the preparation of antihypertensive and antiarrhythmic trans-2,2-dimethylchroman-3-parent derivatives |
Country Status (9)
Country | Link |
---|---|
EP (1) | EP0296975A1 (en) |
JP (1) | JPS6426578A (en) |
KR (1) | KR890000470A (en) |
DK (1) | DK343388A (en) |
FI (1) | FI90343C (en) |
IL (1) | IL86798A (en) |
NO (1) | NO170216C (en) |
NZ (1) | NZ225117A (en) |
PT (1) | PT87788B (en) |
Families Citing this family (27)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3726261A1 (en) * | 1986-12-23 | 1988-07-07 | Merck Patent Gmbh | CHROME DERIVATIVES |
US5387587A (en) * | 1986-12-23 | 1995-02-07 | Merck Patent Gesellschaft Mit Beschrankter Haftung | Chroman derivatives |
US5284838A (en) * | 1987-06-23 | 1994-02-08 | Elf Sanofi | Use of 2,2-dimethylchroman-3-ol derivatives in the treatment of asthma |
US4971982A (en) * | 1987-07-06 | 1990-11-20 | Hoffmann-La Roche Inc. | Benzopyran derivatives |
US5021432A (en) * | 1988-04-26 | 1991-06-04 | Yoshitomi Pharmaceutical Industries, Ltd. | Benzopyran compound and its pharmaceutical use |
JPH03500542A (en) * | 1988-05-09 | 1991-02-07 | ビーチャム グループ ピーエルシー | Novel compounds and treatments |
US5254557A (en) * | 1988-05-09 | 1993-10-19 | Beecham Group P.L.C. | Compound and treatment |
DE3837809A1 (en) * | 1988-11-08 | 1990-05-10 | Merck Patent Gmbh | tetralin |
DE68921972T2 (en) * | 1988-12-13 | 1995-11-16 | Beecham Group Plc | Benzopyran and related compounds. |
US5239090A (en) * | 1989-02-01 | 1993-08-24 | Beecham Group P.L.C. | Certain optically active 3,4-dihydrobenzopyran-4-ols which are intermediates |
GB8902118D0 (en) * | 1989-02-01 | 1989-03-22 | Beecham Group Plc | Chemical process |
US5066816A (en) * | 1989-03-03 | 1991-11-19 | Yoshitomi Pharmaceutical Industries, Ltd. | Processes for preparing optically active 3,4-dihydro-3,4-epoxy-2h-1-benzopyran compounds and intermediates therefor |
US5162553A (en) * | 1989-03-03 | 1992-11-10 | Yoshitomi Pharmaceutical Industries, Ltd. | Processes for preparing optically active 3,4-dihydro-3,4-epoxy-2H-1-benzopyran compounds and intermediates therefor |
FR2645021A1 (en) * | 1989-03-30 | 1990-10-05 | Sanofi Sa | USE OF A POTASSIC AGONIST IN THE TREATMENT OF GLAUCOMA |
DE3923839A1 (en) * | 1989-07-19 | 1991-01-31 | Beiersdorf Ag | New benzopyran derivs. (I) as vasodilators and spasmolytic agents - for treatment of hypertension, angina, migrating, asthma etc. |
GB8916683D0 (en) * | 1989-07-21 | 1989-09-06 | Beecham Group Plc | Novel compounds |
DE3924417A1 (en) * | 1989-07-24 | 1991-01-31 | Merck Patent Gmbh | chroman |
DE3926001A1 (en) * | 1989-08-05 | 1991-02-07 | Merck Patent Gmbh | chroman |
FR2657872B2 (en) * | 1989-11-06 | 1992-06-12 | Sanofi Sa | AMIDINO-4 CHROMAN DERIVATIVE, PROCESS FOR OBTAINING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME. |
FR2654103B1 (en) * | 1989-11-06 | 1992-02-21 | Sanofi Sa | AMIDINO-4 CHROMANNE DERIVATIVES, PROCESS FOR OBTAINING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME. |
US5185345A (en) * | 1989-11-06 | 1993-02-09 | Sanofi | 4-amidino pyrano (3,2-c) pyridine derivatives, and pharmaceutical compositions containing them |
DE4115465A1 (en) * | 1991-05-11 | 1992-11-12 | Beiersdorf Ag | NEW 2H-BENZO (B) PYRANE DERIVATIVES SUBSTITUTED IN 4-POSITION BY ARYL OR N-HETEROARYL, METHODS FOR THEIR PRODUCTION AND THEIR USE AND THE PREPARATIONS CONTAINING THE COMPOUNDS |
HUT70745A (en) * | 1991-12-05 | 1995-10-30 | Smithkline Beecham Plc | Pharmaceutical composition for treatment of disorders of respiratory tract and hypertension containing (3s,4r)-3,4-dihydro-2,2-dimethyl-4-(2-oxo-piperidinyl)-6-pentafluorethyl-2h-1-benzopyranol |
GB9203596D0 (en) * | 1992-02-20 | 1992-04-08 | Smithkline Beecham Plc | Novel process |
GB9207400D0 (en) * | 1992-04-02 | 1992-05-13 | Smithkline Beecham Plc | Novel use |
KR100231634B1 (en) * | 1992-08-17 | 1999-11-15 | 나가야마 오사무 | Benzopyran derivatives |
US6031115A (en) * | 1993-05-14 | 2000-02-29 | Smithkline Beecham Plc | Process for preparing epoxides |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0076075B1 (en) * | 1981-09-25 | 1986-11-20 | Beecham Group Plc | Pharmaceutically active benzopyran compounds |
EP0107423B1 (en) * | 1982-10-19 | 1986-07-23 | Beecham Group Plc | Novel chromans and chromenes |
EP0172352B1 (en) * | 1984-06-22 | 1990-08-29 | Beecham Group Plc | Active benzopyran compounds |
DE3726261A1 (en) * | 1986-12-23 | 1988-07-07 | Merck Patent Gmbh | CHROME DERIVATIVES |
-
1988
- 1988-06-20 FI FI882945A patent/FI90343C/en not_active IP Right Cessation
- 1988-06-20 IL IL86798A patent/IL86798A/en not_active IP Right Cessation
- 1988-06-21 NZ NZ225117A patent/NZ225117A/en unknown
- 1988-06-22 NO NO882762A patent/NO170216C/en unknown
- 1988-06-22 PT PT87788A patent/PT87788B/en not_active IP Right Cessation
- 1988-06-22 DK DK343388A patent/DK343388A/en unknown
- 1988-06-23 EP EP88401580A patent/EP0296975A1/en not_active Withdrawn
- 1988-06-23 KR KR1019880007608A patent/KR890000470A/en not_active Application Discontinuation
- 1988-06-23 JP JP63155989A patent/JPS6426578A/en active Pending
Also Published As
Publication number | Publication date |
---|---|
NO170216B (en) | 1992-06-15 |
DK343388D0 (en) | 1988-06-22 |
NO882762D0 (en) | 1988-06-22 |
FI90343C (en) | 1994-01-25 |
EP0296975A1 (en) | 1988-12-28 |
JPS6426578A (en) | 1989-01-27 |
PT87788B (en) | 1992-10-30 |
NO882762L (en) | 1988-12-27 |
IL86798A0 (en) | 1988-11-30 |
NZ225117A (en) | 1990-02-26 |
DK343388A (en) | 1988-12-24 |
FI882945A (en) | 1988-12-24 |
PT87788A (en) | 1988-07-01 |
IL86798A (en) | 1992-12-01 |
NO170216C (en) | 1992-09-23 |
KR890000470A (en) | 1989-03-14 |
FI90343B (en) | 1993-10-15 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
BB | Publication of examined application | ||
PC | Transfer of assignment of patent |
Owner name: MERCK PATENT GMBH |
|
MM | Patent lapsed | ||
MM | Patent lapsed |
Owner name: MERCK PATENT GMBH |