FI811855A7 - Menetelmä N-aryyli-N'-/(1,4,5,6- tetrahydropyrimidin-2-yyli)- tai (4,5,6,7-tetrahydro-1-H-1,3-diatsepinyyli)/ureoiden valmistamiseksi suolistohäiriöiden hoitoon tai antihypeantihypertensiiviksi aineiksi. - Google Patents

Menetelmä N-aryyli-N'-/(1,4,5,6- tetrahydropyrimidin-2-yyli)- tai (4,5,6,7-tetrahydro-1-H-1,3-diatsepinyyli)/ureoiden valmistamiseksi suolistohäiriöiden hoitoon tai antihypeantihypertensiiviksi aineiksi. Download PDF

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Publication number
FI811855A7
FI811855A7 FI811855A FI811855A FI811855A7 FI 811855 A7 FI811855 A7 FI 811855A7 FI 811855 A FI811855 A FI 811855A FI 811855 A FI811855 A FI 811855A FI 811855 A7 FI811855 A7 FI 811855A7
Authority
FI
Finland
Prior art keywords
antihypeantihypertensive
tetrahydropyrimidin
diazepinyl
ureas
tetrahydro
Prior art date
Application number
FI811855A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI811855L (fi
Inventor
C Royce Rasmussen
Original Assignee
Mcneilab Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/159,986 external-priority patent/US4466966A/en
Priority claimed from US06/159,988 external-priority patent/US4285948A/en
Application filed by Mcneilab Inc filed Critical Mcneilab Inc
Publication of FI811855L publication Critical patent/FI811855L/fi
Publication of FI811855A7 publication Critical patent/FI811855A7/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/04Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/06Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D239/08Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms directly attached in position 2
    • C07D239/12Nitrogen atoms not forming part of a nitro radical
    • C07D239/16Nitrogen atoms not forming part of a nitro radical acylated on said nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI811855A 1980-06-16 1981-06-15 Menetelmä N-aryyli-N'-/(1,4,5,6- tetrahydropyrimidin-2-yyli)- tai (4,5,6,7-tetrahydro-1-H-1,3-diatsepinyyli)/ureoiden valmistamiseksi suolistohäiriöiden hoitoon tai antihypeantihypertensiiviksi aineiksi. FI811855A7 (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US15998780A 1980-06-16 1980-06-16
US15998580A 1980-06-16 1980-06-16
US06/159,986 US4466966A (en) 1980-06-16 1980-06-16 N-aryl-N'-(1,4,5,6-tetrahydropyrimidin-2-yl)ureas for intestinal disorders
US06/159,988 US4285948A (en) 1980-06-16 1980-06-16 N-Aryl-N'-(1,4,5,6-tetrahydropyrimidine-2-yl)ureas as antihypertensives

Publications (2)

Publication Number Publication Date
FI811855L FI811855L (fi) 1981-12-17
FI811855A7 true FI811855A7 (fi) 1981-12-17

Family

ID=27496405

Family Applications (1)

Application Number Title Priority Date Filing Date
FI811855A FI811855A7 (fi) 1980-06-16 1981-06-15 Menetelmä N-aryyli-N'-/(1,4,5,6- tetrahydropyrimidin-2-yyli)- tai (4,5,6,7-tetrahydro-1-H-1,3-diatsepinyyli)/ureoiden valmistamiseksi suolistohäiriöiden hoitoon tai antihypeantihypertensiiviksi aineiksi.

Country Status (15)

Country Link
EP (1) EP0042279B1 (cg-RX-API-DMAC10.html)
CA (1) CA1151167A (cg-RX-API-DMAC10.html)
DE (1) DE3172886D1 (cg-RX-API-DMAC10.html)
DK (1) DK260281A (cg-RX-API-DMAC10.html)
ES (1) ES503013A0 (cg-RX-API-DMAC10.html)
FI (1) FI811855A7 (cg-RX-API-DMAC10.html)
GR (1) GR74547B (cg-RX-API-DMAC10.html)
HK (1) HK24686A (cg-RX-API-DMAC10.html)
IL (1) IL63099A (cg-RX-API-DMAC10.html)
MY (1) MY8600520A (cg-RX-API-DMAC10.html)
NO (1) NO812023L (cg-RX-API-DMAC10.html)
NZ (1) NZ197385A (cg-RX-API-DMAC10.html)
PH (1) PH16725A (cg-RX-API-DMAC10.html)
PT (1) PT73196B (cg-RX-API-DMAC10.html)
YU (1) YU151781A (cg-RX-API-DMAC10.html)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE177078T1 (de) * 1993-10-21 1999-03-15 Searle & Co Amidino-derivate als no-synthetase inhibitoren

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL267923A (cg-RX-API-DMAC10.html) * 1960-08-05
US4204000A (en) * 1975-03-31 1980-05-20 William H. Rorer, Inc. Anti-ulcer amidinoureas

Also Published As

Publication number Publication date
YU151781A (en) 1984-02-29
NO812023L (no) 1981-12-17
ES8304093A1 (es) 1983-02-16
PH16725A (en) 1984-01-25
IL63099A (en) 1985-03-31
MY8600520A (en) 1986-12-31
EP0042279A2 (en) 1981-12-23
EP0042279A3 (en) 1982-08-25
PT73196A (en) 1981-07-01
IL63099A0 (en) 1981-09-13
FI811855L (fi) 1981-12-17
DK260281A (da) 1981-12-17
HK24686A (en) 1986-04-11
PT73196B (en) 1983-04-26
EP0042279B1 (en) 1985-11-13
GR74547B (cg-RX-API-DMAC10.html) 1984-06-29
ES503013A0 (es) 1983-02-16
CA1151167A (en) 1983-08-02
NZ197385A (en) 1984-08-24
DE3172886D1 (en) 1985-12-19

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Owner name: MCNEILAB, INC.