FI51939B - - Google Patents

Info

Publication number
FI51939B
FI51939B FI2170/70A FI217070A FI51939B FI 51939 B FI51939 B FI 51939B FI 2170/70 A FI2170/70 A FI 2170/70A FI 217070 A FI217070 A FI 217070A FI 51939 B FI51939 B FI 51939B
Authority
FI
Finland
Application number
FI2170/70A
Other languages
Finnish (fi)
Other versions
FI51939C (fi
Inventor
Eberhard Woitun
Berthold Narr
Wolfgang Schroeter
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19691940572 external-priority patent/DE1940572A1/de
Priority claimed from DE19702032686 external-priority patent/DE2032686A1/de
Priority claimed from DE19702032687 external-priority patent/DE2032687A1/de
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of FI51939B publication Critical patent/FI51939B/fi
Application granted granted Critical
Publication of FI51939C publication Critical patent/FI51939C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
FI702170A 1969-08-08 1970-08-06 Menetelmä uusien verihiutaleiden kasautumista estävien 2-aminoalkyylia mino-tieno(3,2-d)pyrimidiinien valmistamiseksi FI51939C (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19691940572 DE1940572A1 (de) 1969-08-08 1969-08-08 Neue 2-Aminoalkylamino-thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung
DE19702032686 DE2032686A1 (de) 1970-07-02 1970-07-02 Verfahren zur Herstellung von neuen 2 Aminoalkylamino thieno eckige Klammer auf 3,2 d eckige Klammer zu Pynmidinen
DE19702032687 DE2032687A1 (en) 1970-07-02 1970-07-02 Cardiovascular 2-aminoalkylamino-thienopyrimidines - and 4-morpholino derivatives from 4-diethanolamino-compounds by intramolecular cyclisa

Publications (2)

Publication Number Publication Date
FI51939B true FI51939B (fr) 1977-01-31
FI51939C FI51939C (fi) 1977-05-10

Family

ID=27182086

Family Applications (1)

Application Number Title Priority Date Filing Date
FI702170A FI51939C (fi) 1969-08-08 1970-08-06 Menetelmä uusien verihiutaleiden kasautumista estävien 2-aminoalkyylia mino-tieno(3,2-d)pyrimidiinien valmistamiseksi

Country Status (14)

Country Link
US (1) US3838121A (fr)
JP (1) JPS519759B1 (fr)
BE (1) BE754606A (fr)
BG (1) BG17591A3 (fr)
CH (5) CH547301A (fr)
ES (5) ES382551A1 (fr)
FI (1) FI51939C (fr)
FR (1) FR2068478B1 (fr)
IE (1) IE34687B1 (fr)
IL (1) IL35078A (fr)
NL (1) NL7011592A (fr)
NO (1) NO130538C (fr)
PH (1) PH9574A (fr)
SE (1) SE386449B (fr)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6187777B1 (en) 1998-02-06 2001-02-13 Amgen Inc. Compounds and methods which modulate feeding behavior and related diseases
EP1608652A1 (fr) * 2003-03-31 2005-12-28 Vernalis (Cambridge) Limited Composes pyrazolopyrimidines et leur utilisation en medecine
GB0423653D0 (en) 2004-10-25 2004-11-24 Piramed Ltd Pharmaceutical compounds
EP1847543A1 (fr) 2006-04-19 2007-10-24 Boehringer Ingelheim Pharma GmbH & Co. KG Dihydrothienopyrimidines pour le traitement de maladies inflammatoires
PT1874781E (pt) * 2006-04-19 2009-07-27 Boehringer Ingelheim Int Di-hidro-tienopirimidinas para o tratamento de doenças inflamatórias
CL2007001167A1 (es) 2006-04-26 2008-01-25 Genentech Inc Compuestos derivados de pirimidina condensada, inhibidores de p13-quinasa; procesos para preparar los compuestos; composicion farmaceutica que los comprende; uso de los compuestos en la preparacion de medicamentos; proceso para preparar la composicion farmaceutica; y kit que incluye a la composicionfarmaceutica.
US7846929B2 (en) 2006-04-26 2010-12-07 Genentech, Inc. Phosphoinositide 3-kinase inhibitor compounds and methods of use
CL2007001165A1 (es) * 2006-04-26 2008-01-25 Hoffmann La Roche 2-(1h-indazol-4-il)-6-(4-metanosulfonil-piperazin-1-ilmetil)-4-morfolin-4-il-tieno[3,2-d]pirimidina; procedimiento de preparacion; composicion farmaceutica; proceso de preparacion de dicha composicion; kit farmaceutico; y uso para tratar enfermedades tales como cancer, desordenes inmunes y enfermedades cardiovasculares.
KR101460816B1 (ko) 2006-12-07 2014-11-12 에프. 호프만-라 로슈 아게 포스포이노시타이드 3-키나제 억제제 화합물 및 그의 사용 방법
KR101507182B1 (ko) * 2006-12-07 2015-03-30 제넨테크, 인크. 포스포이노시타이드 3-키나제 억제제 화합물 및 그의 사용 방법
WO2009050242A2 (fr) * 2007-10-19 2009-04-23 Boehringer Ingelheim International Gmbh Pipérazino-dihydrothiénopyrimidines substituées par un hétérocycle
BRPI0818006B8 (pt) * 2007-10-19 2021-05-25 Boehringer Ingelheim Int compostos de piperidino-di-hidrotienopirimidinas substituídas, uso dos mesmos e formulações farmacêuticas
ATE537175T1 (de) 2007-10-19 2011-12-15 Boehringer Ingelheim Int Neue piperazino-dihydrothienopyrimidin-derivate
GB0721095D0 (en) * 2007-10-26 2007-12-05 Piramed Ltd Pharmaceutical compounds
CA2761445A1 (fr) 2009-05-27 2010-12-02 Genentech, Inc. Composes pyrimidines bicycliques inhibiteurs de pi3k selectifs pour p110 delta, et procedes d'utilisation
US8158625B2 (en) * 2009-05-27 2012-04-17 Genentech, Inc. Bicyclic indole-pyrimidine PI3K inhibitor compounds selective for P110 delta, and methods of use
NZ599939A (en) * 2009-10-12 2014-02-28 Hoffmann La Roche Combinations of a pi3k inhibitor and a mek inhibitor
US9802954B2 (en) 2011-08-24 2017-10-31 Boehringer Ingelheim International Gmbh Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthma
US20130059866A1 (en) 2011-08-24 2013-03-07 Boehringer Ingelheim International Gmbh Novel piperidino-dihydrothienopyrimidine sulfoxides and their use for treating copd and asthma

Also Published As

Publication number Publication date
ES382548A1 (es) 1973-04-01
BG17591A3 (fr) 1973-11-10
NL7011592A (fr) 1971-02-10
CH547299A (de) 1974-03-29
CH547304A (de) 1974-03-29
CH546251A (de) 1974-02-28
NO130538B (fr) 1974-09-23
ES382549A1 (es) 1973-04-01
FI51939C (fi) 1977-05-10
IL35078A (en) 1974-09-10
FR2068478B1 (fr) 1974-08-30
IL35078A0 (en) 1970-10-30
SE386449B (sv) 1976-08-09
NO130538C (fr) 1975-01-08
PH9574A (en) 1976-01-16
ES382550A1 (es) 1973-04-16
ES382552A1 (es) 1973-04-16
IE34687B1 (en) 1975-07-23
BE754606A (fr) 1971-02-08
FR2068478A1 (fr) 1971-08-27
US3838121A (en) 1974-09-24
ES382551A1 (es) 1973-04-01
CH547300A (de) 1974-03-29
IE34687L (en) 1971-02-08
JPS519759B1 (fr) 1976-03-30
CH547301A (de) 1974-03-29

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