ES8403899A1 - Process for the preparation of new benzamide derivatives - Google Patents
Process for the preparation of new benzamide derivativesInfo
- Publication number
- ES8403899A1 ES8403899A1 ES520622A ES520622A ES8403899A1 ES 8403899 A1 ES8403899 A1 ES 8403899A1 ES 520622 A ES520622 A ES 520622A ES 520622 A ES520622 A ES 520622A ES 8403899 A1 ES8403899 A1 ES 8403899A1
- Authority
- ES
- Spain
- Prior art keywords
- group
- alkyl
- alkylthio
- alkoxy
- hydrogen
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Abstract
Pharmaceutical compositions comprising compounds of formula (I) or pharmaceutically acceptable salts and/or the corresponding N-oxides and/or solvates: < IMAGE > where: R1 is a C1-6 alkoxy or C1-6 alkylthio group and one of R2, R3 and R4 is hydrogen, the second is C1-6 alkylthio and the third is selected from the group of constituents comprising hydrogen, halogen, CF3, C1-6 alkyl, C1-6 alkoxy, C1-6 alkylthio, C1-7 acyl, C1-7 acyl amino, C1-6 alkyl sulphonyl, C1-6 alkyl sulphinyl, hydroxy, nitro or amino, aminocarbonyl or aminosulphonyl optionally N-substituted by one or two C1-6 alkyl groups or R1 is joined to R2 to form C1-2 alkylenedioxy and one of R3 and R4 is C1-6 alkylthio and the other is selected from the group of substituents specified above R5 is hydrogen or C1-6 alkyl R6 is C1-7 alkyl or a -(CH2)sR7 group, where s is from 0 to 2 and R7 is a C3-8 cycloalkyl group or a -(CH2)tR8 group, where t is 1 or 2 and R8 is C2-5 alkinyl or a phenyl group optionally substituted by one or two substituents selected from C1-6 alkyl, C1-4 alkoxy, trifluoromethyl and halogen, or a thienyl group and p and q are, separately, from 0 to 2, and a pharmaceutically acceptable vehicle, new compounds of formula (I) which have useful pharmacological activity and a process for their preparation.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB8118603 | 1981-06-17 | ||
GB8118604 | 1981-06-17 | ||
GB8119997 | 1981-06-29 | ||
GB8119998 | 1981-06-29 |
Publications (2)
Publication Number | Publication Date |
---|---|
ES520622A0 ES520622A0 (en) | 1984-04-01 |
ES8403899A1 true ES8403899A1 (en) | 1984-04-01 |
Family
ID=27449253
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES513160A Granted ES513160A0 (en) | 1981-06-17 | 1982-06-16 | A PROCEDURE FOR THE PREPARATION OF NEW BENZAMINE DERIVATIVES. |
ES520622A Expired ES8403899A1 (en) | 1981-06-17 | 1983-03-15 | Process for the preparation of new benzamide derivatives |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES513160A Granted ES513160A0 (en) | 1981-06-17 | 1982-06-16 | A PROCEDURE FOR THE PREPARATION OF NEW BENZAMINE DERIVATIVES. |
Country Status (1)
Country | Link |
---|---|
ES (2) | ES513160A0 (en) |
-
1982
- 1982-06-16 ES ES513160A patent/ES513160A0/en active Granted
-
1983
- 1983-03-15 ES ES520622A patent/ES8403899A1/en not_active Expired
Also Published As
Publication number | Publication date |
---|---|
ES520622A0 (en) | 1984-04-01 |
ES8307805A1 (en) | 1983-08-01 |
ES513160A0 (en) | 1983-08-01 |
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