ES8307805A1 - Process for the preparation of new benzamide derivatives - Google Patents

Process for the preparation of new benzamide derivatives

Info

Publication number
ES8307805A1
ES8307805A1 ES513160A ES513160A ES8307805A1 ES 8307805 A1 ES8307805 A1 ES 8307805A1 ES 513160 A ES513160 A ES 513160A ES 513160 A ES513160 A ES 513160A ES 8307805 A1 ES8307805 A1 ES 8307805A1
Authority
ES
Spain
Prior art keywords
group
alkyl
alkylthio
alkoxy
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES513160A
Other languages
Spanish (es)
Other versions
ES513160A0 (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Beecham Group PLC
Original Assignee
Beecham Group PLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beecham Group PLC filed Critical Beecham Group PLC
Publication of ES8307805A1 publication Critical patent/ES8307805A1/en
Publication of ES513160A0 publication Critical patent/ES513160A0/en
Granted legal-status Critical Current

Links

Abstract

Pharmaceutical compositions comprising compounds of formula (I) or pharmaceutically acceptable salts and/or the corresponding N-oxides and/or solvates: <IMAGE> where: R1 is a C1-6 alkoxy or C1-6 alkylthio group; and one of R2, R3 and R4 is hydrogen, the second is C1-6 alkylthio and the third is selected from the group of constituents comprising hydrogen, halogen, CF3, C1-6 alkyl, C1-6 alkoxy, C1-6 alkylthio, C1-7 acyl, C1-7 acyl amino, C1-6 alkyl sulphonyl, C1-6 alkyl sulphinyl, hydroxy, nitro or amino, aminocarbonyl or aminosulphonyl optionally N-substituted by one or two C1-6 alkyl groups; or R1 is joined to R2 to form C1-2 alkylenedioxy; and one of R3 and R4 is C1-6 alkylthio and the other is selected from the group of substituents specified above; R5 is hydrogen or C1-6 alkyl; R6 is C1-7 alkyl or a -(CH2)sR7 group, where s is from 0 to 2 and R7 is a C3-8 cycloalkyl group or a -(CH2)tR8 group, where t is 1 or 2 and R8 is C2-5 alkinyl or a phenyl group optionally substituted by one or two substituents selected from C1-6 alkyl, C1-4 alkoxy, trifluoromethyl and halogen, or a thienyl group; and p and q are, separately, from 0 to 2, and a pharmaceutically acceptable vehicle, new compounds of formula (I) which have useful pharmacological activity and a process for their preparation.
ES513160A 1981-06-17 1982-06-16 A PROCEDURE FOR THE PREPARATION OF NEW BENZAMINE DERIVATIVES. Granted ES513160A0 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB8118604 1981-06-17
GB8118603 1981-06-17
GB8119997 1981-06-29
GB8119998 1981-06-29

Publications (2)

Publication Number Publication Date
ES8307805A1 true ES8307805A1 (en) 1983-08-01
ES513160A0 ES513160A0 (en) 1983-08-01

Family

ID=27449253

Family Applications (2)

Application Number Title Priority Date Filing Date
ES513160A Granted ES513160A0 (en) 1981-06-17 1982-06-16 A PROCEDURE FOR THE PREPARATION OF NEW BENZAMINE DERIVATIVES.
ES520622A Expired ES8403899A1 (en) 1981-06-17 1983-03-15 Process for the preparation of new benzamide derivatives

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES520622A Expired ES8403899A1 (en) 1981-06-17 1983-03-15 Process for the preparation of new benzamide derivatives

Country Status (1)

Country Link
ES (2) ES513160A0 (en)

Also Published As

Publication number Publication date
ES520622A0 (en) 1984-04-01
ES513160A0 (en) 1983-08-01
ES8403899A1 (en) 1984-04-01

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