ES8307805A1 - Process for the preparation of new benzamide derivatives - Google Patents
Process for the preparation of new benzamide derivativesInfo
- Publication number
- ES8307805A1 ES8307805A1 ES513160A ES513160A ES8307805A1 ES 8307805 A1 ES8307805 A1 ES 8307805A1 ES 513160 A ES513160 A ES 513160A ES 513160 A ES513160 A ES 513160A ES 8307805 A1 ES8307805 A1 ES 8307805A1
- Authority
- ES
- Spain
- Prior art keywords
- group
- alkyl
- alkylthio
- alkoxy
- hydrogen
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Abstract
Pharmaceutical compositions comprising compounds of formula (I) or pharmaceutically acceptable salts and/or the corresponding N-oxides and/or solvates: <IMAGE> where: R1 is a C1-6 alkoxy or C1-6 alkylthio group; and one of R2, R3 and R4 is hydrogen, the second is C1-6 alkylthio and the third is selected from the group of constituents comprising hydrogen, halogen, CF3, C1-6 alkyl, C1-6 alkoxy, C1-6 alkylthio, C1-7 acyl, C1-7 acyl amino, C1-6 alkyl sulphonyl, C1-6 alkyl sulphinyl, hydroxy, nitro or amino, aminocarbonyl or aminosulphonyl optionally N-substituted by one or two C1-6 alkyl groups; or R1 is joined to R2 to form C1-2 alkylenedioxy; and one of R3 and R4 is C1-6 alkylthio and the other is selected from the group of substituents specified above; R5 is hydrogen or C1-6 alkyl; R6 is C1-7 alkyl or a -(CH2)sR7 group, where s is from 0 to 2 and R7 is a C3-8 cycloalkyl group or a -(CH2)tR8 group, where t is 1 or 2 and R8 is C2-5 alkinyl or a phenyl group optionally substituted by one or two substituents selected from C1-6 alkyl, C1-4 alkoxy, trifluoromethyl and halogen, or a thienyl group; and p and q are, separately, from 0 to 2, and a pharmaceutically acceptable vehicle, new compounds of formula (I) which have useful pharmacological activity and a process for their preparation.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB8118604 | 1981-06-17 | ||
GB8118603 | 1981-06-17 | ||
GB8119997 | 1981-06-29 | ||
GB8119998 | 1981-06-29 |
Publications (2)
Publication Number | Publication Date |
---|---|
ES8307805A1 true ES8307805A1 (en) | 1983-08-01 |
ES513160A0 ES513160A0 (en) | 1983-08-01 |
Family
ID=27449253
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES513160A Granted ES513160A0 (en) | 1981-06-17 | 1982-06-16 | A PROCEDURE FOR THE PREPARATION OF NEW BENZAMINE DERIVATIVES. |
ES520622A Expired ES8403899A1 (en) | 1981-06-17 | 1983-03-15 | Process for the preparation of new benzamide derivatives |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES520622A Expired ES8403899A1 (en) | 1981-06-17 | 1983-03-15 | Process for the preparation of new benzamide derivatives |
Country Status (1)
Country | Link |
---|---|
ES (2) | ES513160A0 (en) |
-
1982
- 1982-06-16 ES ES513160A patent/ES513160A0/en active Granted
-
1983
- 1983-03-15 ES ES520622A patent/ES8403899A1/en not_active Expired
Also Published As
Publication number | Publication date |
---|---|
ES520622A0 (en) | 1984-04-01 |
ES513160A0 (en) | 1983-08-01 |
ES8403899A1 (en) | 1984-04-01 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ES8101072A1 (en) | Azabicycloalkyl derivatives, a process for their preparation and pharmaceutical compositions containing them. | |
LV11035A (en) | New Benzimidazoline-2-Oxo-1-Carboxylic Derivatives Used As Serotonin (5-HT) Receptor Antagonists | |
DE3069408D1 (en) | 5-oxo- and 5-thioxoproline derivatives, process for their production and pharmaceutical compositions containing them | |
ES8404349A1 (en) | Nortropyl benzopyrrolinone compounds, process for their preparation and pharmaceutical compositions containing them. | |
DE3372965D1 (en) | Amide derivatives | |
DE3850742D1 (en) | New 4-oxobenzotriazines and 4-oxoquinazolines. | |
ES8203364A1 (en) | Aniline derivatives. | |
ES8307244A1 (en) | Azobicycloalkylbenzamides, process for their preparation and pharmaceutical compositions containing them. | |
ES8300762A1 (en) | Azabicycloalkane derivatives, their preparation and use. | |
ES8506634A1 (en) | Amide derivatives of azabicycloalkanes. | |
ES8305359A1 (en) | Bicyclo (3,2,1) octylbenzamides, a process for their preparation and pharmaceutical compositions containing them. | |
ES8203901A1 (en) | Pharmaceutically active compounds. | |
ES8307805A1 (en) | Process for the preparation of new benzamide derivatives | |
FI802384A (en) | NYA 3-AMINO-1-BENZOXEPINE DERIVATIVES AND DERAS SALTER; FOERFARANDE FOER DERAS FRAMSTAELLNING SAMT CEILING MODEL INNEHAOLLANDE DESSA FOERENINGAR | |
ES8402299A1 (en) | N-azabicycloalkane benzamides, process for their preparation and pharmaceutical compositions containing them. | |
ES8105713A1 (en) | Levorotatory and dextrorotatory enantiomers of 3-methoxycyproheptadine and analogs thereof, process for their preparation and antipsychotic pharmaceutical compositions. |