ES8302647A1 - Un procedimiento para la preparacion de guanidinas - Google Patents
Un procedimiento para la preparacion de guanidinasInfo
- Publication number
- ES8302647A1 ES8302647A1 ES502487A ES502487A ES8302647A1 ES 8302647 A1 ES8302647 A1 ES 8302647A1 ES 502487 A ES502487 A ES 502487A ES 502487 A ES502487 A ES 502487A ES 8302647 A1 ES8302647 A1 ES 8302647A1
- Authority
- ES
- Spain
- Prior art keywords
- guanidines
- antidiarrhoeal
- medicaments
- manufacturing
- compositions containing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/20—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
Abstract
PROCEDIMIENTO PARA LA OBTENCION DE GUANIDINAS Y DE SUS SALES DE ADICION DE ACIDO FISIOLOGICAMENTE COMPATIBLES, DE FORMULA (I), EN LA QUE R Y R SON ALQUILO INFERIOR O TRIFLUOROMETILO; Y R Y R SON HIDROGENO, ALQUILO INFERIOR, O JUNTOS REPRESENTAN DIMETILENO O TRIMETILENO; COMPUESTOS QUE TIENEN APLICACIONES FARMACOLOGICAS POR SU ACTIVIDAD ANTIDIARREICA. CONSISTE EN LA REACCION DE CONDENSACION DE UN DERIVADO REACTIVO DE UN ACIDO DE FORMULA (II), O UNA SAL DE ADICION DE ACIDO RESPECTIVA, CON UN COMPUESTO DE FORMULA (III), EN LAS QUE R -R TIENEN EL MISMO SIGNIFICADO QUE EN LA FORMULA (I). LA REACCION SE LLEVA A CABO SIGUIENDO METODOS CONVENCIONALES.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB8017377 | 1980-05-27 | ||
| GB8104410 | 1981-02-12 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES502487A0 ES502487A0 (es) | 1983-02-01 |
| ES8302647A1 true ES8302647A1 (es) | 1983-02-01 |
Family
ID=26275656
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES502487A Expired ES8302647A1 (es) | 1980-05-27 | 1981-05-26 | Un procedimiento para la preparacion de guanidinas |
| ES514336A Expired ES8305317A1 (es) | 1980-05-27 | 1982-06-16 | Un procedimiento para la preparacion de guanidinas. |
| ES514335A Granted ES514335A0 (es) | 1980-05-27 | 1982-06-16 | Un procedimiento para la preparacion de guanidinas. |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES514336A Expired ES8305317A1 (es) | 1980-05-27 | 1982-06-16 | Un procedimiento para la preparacion de guanidinas. |
| ES514335A Granted ES514335A0 (es) | 1980-05-27 | 1982-06-16 | Un procedimiento para la preparacion de guanidinas. |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US4443467A (es) |
| EP (1) | EP0040947B1 (es) |
| AU (1) | AU539121B2 (es) |
| CA (1) | CA1158558A (es) |
| DE (1) | DE3175672D1 (es) |
| DK (1) | DK228381A (es) |
| ES (3) | ES8302647A1 (es) |
| FI (1) | FI811601L (es) |
| GB (1) | GB2080107B (es) |
| GR (1) | GR74922B (es) |
| IL (1) | IL62809A (es) |
| IT (1) | IT1136619B (es) |
| MX (1) | MX6962E (es) |
| MY (1) | MY8700598A (es) |
| NZ (1) | NZ197026A (es) |
| PH (2) | PH16855A (es) |
| PT (1) | PT73087B (es) |
| ZW (1) | ZW11381A1 (es) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4714707A (en) * | 1984-01-13 | 1987-12-22 | Rorer Pharmaceutical Corporation | Aryl substituted heterocycles for treating gastrointestinal motility dysfunction |
| GB8525013D0 (en) * | 1985-10-10 | 1985-11-13 | Wyeth John & Brother Ltd | Antidiarrhoel agents |
| DK153442C (da) * | 1985-10-14 | 1988-12-19 | Poul Bachmann | Middel, baseret paa pektinholdigt materiale, til behandling og forebyggelse af diarre hos mennesker og dyr |
| GB8806224D0 (en) * | 1988-03-16 | 1988-04-13 | Johnson Matthey Plc | Platinum chemotherapeutic product |
| US20050191403A1 (en) * | 2002-05-23 | 2005-09-01 | Glutagen Pty Ltd | Palliative treatment for gluten intolerance |
| US7976872B2 (en) * | 2006-07-24 | 2011-07-12 | L. Perrigo Company | Method for distributing a pharmaceutically active compound in an excipient |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1530675A (en) * | 1976-06-05 | 1978-11-01 | Wyeth John & Brother Ltd | Guanidine derivatives |
-
1981
- 1981-05-01 CA CA000376666A patent/CA1158558A/en not_active Expired
- 1981-05-06 AU AU70203/81A patent/AU539121B2/en not_active Ceased
- 1981-05-06 IL IL62809A patent/IL62809A/xx unknown
- 1981-05-07 NZ NZ197026A patent/NZ197026A/en unknown
- 1981-05-08 GR GR64893A patent/GR74922B/el unknown
- 1981-05-11 ZW ZW113/81A patent/ZW11381A1/xx unknown
- 1981-05-11 US US06/262,148 patent/US4443467A/en not_active Expired - Fee Related
- 1981-05-15 PH PH25641A patent/PH16855A/en unknown
- 1981-05-19 DE DE8181302211T patent/DE3175672D1/de not_active Expired
- 1981-05-19 GB GB8115356A patent/GB2080107B/en not_active Expired
- 1981-05-19 EP EP81302211A patent/EP0040947B1/en not_active Expired
- 1981-05-20 IT IT21847/81A patent/IT1136619B/it active
- 1981-05-22 MX MX819461U patent/MX6962E/es unknown
- 1981-05-25 DK DK228381A patent/DK228381A/da unknown
- 1981-05-25 FI FI811601A patent/FI811601L/fi not_active Application Discontinuation
- 1981-05-26 ES ES502487A patent/ES8302647A1/es not_active Expired
- 1981-05-26 PT PT73087A patent/PT73087B/pt unknown
-
1982
- 1982-06-16 ES ES514336A patent/ES8305317A1/es not_active Expired
- 1982-06-16 ES ES514335A patent/ES514335A0/es active Granted
- 1982-07-30 PH PH27647A patent/PH17361A/en unknown
-
1987
- 1987-12-30 MY MY598/87A patent/MY8700598A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL62809A0 (en) | 1981-07-31 |
| FI811601L (fi) | 1981-11-28 |
| DK228381A (da) | 1981-11-28 |
| AU539121B2 (en) | 1984-09-13 |
| US4443467A (en) | 1984-04-17 |
| ZW11381A1 (en) | 1982-11-17 |
| GB2080107B (en) | 1986-02-26 |
| GB2080107A (en) | 1982-02-03 |
| ES8305316A1 (es) | 1983-04-16 |
| GR74922B (es) | 1984-07-12 |
| EP0040947A1 (en) | 1981-12-02 |
| MX6962E (es) | 1987-01-08 |
| ES514336A0 (es) | 1983-04-16 |
| NZ197026A (en) | 1984-05-31 |
| DE3175672D1 (en) | 1987-01-15 |
| MY8700598A (en) | 1987-12-31 |
| PT73087B (en) | 1985-01-08 |
| ES514335A0 (es) | 1983-04-16 |
| IL62809A (en) | 1984-03-30 |
| AU7020381A (en) | 1981-12-03 |
| ES502487A0 (es) | 1983-02-01 |
| EP0040947B1 (en) | 1986-12-03 |
| IT1136619B (it) | 1986-09-03 |
| PH16855A (en) | 1984-03-19 |
| PH17361A (en) | 1984-08-01 |
| ES8305317A1 (es) | 1983-04-16 |
| PT73087A (en) | 1981-06-01 |
| CA1158558A (en) | 1983-12-13 |
| IT8121847A0 (it) | 1981-05-20 |
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