ES8206492A1 - Process for the preparation of 2-methylene-quinoxaline-1,4-dioxide derivatives - Google Patents

Process for the preparation of 2-methylene-quinoxaline-1,4-dioxide derivatives

Info

Publication number
ES8206492A1
ES8206492A1 ES505442A ES505442A ES8206492A1 ES 8206492 A1 ES8206492 A1 ES 8206492A1 ES 505442 A ES505442 A ES 505442A ES 505442 A ES505442 A ES 505442A ES 8206492 A1 ES8206492 A1 ES 8206492A1
Authority
ES
Spain
Prior art keywords
group
general formula
alpha
hydroxyl
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES505442A
Other languages
Spanish (es)
Other versions
ES505442A0 (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Egyt Gyogyszervegyeszeti Gyar
Original Assignee
Egyt Gyogyszervegyeszeti Gyar
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Egyt Gyogyszervegyeszeti Gyar filed Critical Egyt Gyogyszervegyeszeti Gyar
Publication of ES8206492A1 publication Critical patent/ES8206492A1/en
Publication of ES505442A0 publication Critical patent/ES505442A0/en
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/36—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
    • C07D241/50—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to ring nitrogen atoms
    • C07D241/52—Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

2-Methylene-1,4-dioxide derivatives of the general formula (I> < IMAGE > wherein A represents a hydroxyl or an amino group, or a group of the general formula -NH-COOR1, wherein R1 denotes a C1-4 alkyl group or a group of the general formula -NH-CX-NH2, wherein X stands for oxygen or sulfur or a group of the formula -NH-C(=NH)-NH2 or a group of the general formula -NH-R2, wherein R2 represents C1-6 alkyl, phenyl, benzyl, hydroxyl or hydroxy-(C2-4alkyl) or a group of the general formula -NH-CO-R3, wherein R3 stands for a C1-20alkyl group, a phenyl group optionally substituted by one, two or three identical or different substituent(s) selected from the group consisting of hydroxyl, amino, nitro, C1-4alkyl, C1-4 alkoxy or halogen a piperidyl, a pyridyl, a furyl, a nitrofuryl, a pyrazinyl, a pyrimidyl, a naphthyl, a hydroxynaphthyl, a phenylalkyl, an 1,2,4-triazinyl, an alpha , alpha -diphenyl- alpha - hydroxymethyl, a cyanomethyl, a halomethyl or a hydroxymethyl group, are prepared by dehydrating new compounds of the general formula (II> < IMAGE > wherein A has the same meanings as above. The compounds of the general formula (I) possessing bactericidal and weight-gain increasing properties can be obtained in a high purity with an excellent yield by the process according to the invention. A process for the preparation of the new compounds of formula (II) is also disclosed.
ES505442A 1980-09-12 1981-09-12 PROCEDURE FOR THE PREPARATION OF 2-METHYLENE-QUINO-XALINO-1,4-DIOXIDES DERIVATIVES Granted ES505442A0 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU224080 1980-09-12

Publications (2)

Publication Number Publication Date
ES8206492A1 true ES8206492A1 (en) 1982-08-16
ES505442A0 ES505442A0 (en) 1982-08-16

Family

ID=10958457

Family Applications (1)

Application Number Title Priority Date Filing Date
ES505442A Granted ES505442A0 (en) 1980-09-12 1981-09-12 PROCEDURE FOR THE PREPARATION OF 2-METHYLENE-QUINO-XALINO-1,4-DIOXIDES DERIVATIVES

Country Status (14)

Country Link
AR (1) AR226749A1 (en)
BE (1) BE890300A (en)
CA (1) CA1154770A (en)
DE (1) DE3136092A1 (en)
DK (1) DK405181A (en)
ES (1) ES505442A0 (en)
FI (1) FI812835L (en)
FR (1) FR2490226A1 (en)
GB (1) GB2083817A (en)
IL (1) IL63803A0 (en)
IT (1) IT1139962B (en)
PT (1) PT73655B (en)
SE (1) SE8105427L (en)
YU (1) YU218781A (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102617493B (en) * 2012-02-22 2014-06-04 中国农业大学 Mequindox artificial antigens and antibodies prepared by same

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1469485A (en) * 1964-09-16 1967-02-17 Pfizer & Co C Process for the preparation of a new series of schiff bases
US3493572A (en) * 1968-07-05 1970-02-03 Pfizer & Co C Process for producing quinoxaline-di-n-oxides
US3926992A (en) * 1972-11-03 1975-12-16 Pfizer Aldol products of 2-quinoxalinecarboxaldehy-1,4-dioxides
US4221791A (en) * 1979-05-21 1980-09-09 International Minerals & Chemical Corp. Substituted quinoxaline dioxides

Also Published As

Publication number Publication date
IT8123898A0 (en) 1981-09-11
PT73655B (en) 1982-11-22
PT73655A (en) 1981-10-01
YU218781A (en) 1983-04-30
FR2490226A1 (en) 1982-03-19
IT1139962B (en) 1986-09-24
GB2083817A (en) 1982-03-31
DE3136092A1 (en) 1982-05-27
IL63803A0 (en) 1981-12-31
AR226749A1 (en) 1982-08-13
BE890300A (en) 1982-03-10
SE8105427L (en) 1982-03-13
CA1154770A (en) 1983-10-04
ES505442A0 (en) 1982-08-16
DK405181A (en) 1982-03-13
FI812835L (en) 1982-03-13

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