ES550039A0 - Procedimiento para preparar n-(-(1'-alil-2'-pirrolidinil)- metil)-2-metoxi-4,5-azimido-benzamida a escala industrial - Google Patents
Procedimiento para preparar n-(-(1'-alil-2'-pirrolidinil)- metil)-2-metoxi-4,5-azimido-benzamida a escala industrialInfo
- Publication number
- ES550039A0 ES550039A0 ES550039A ES550039A ES550039A0 ES 550039 A0 ES550039 A0 ES 550039A0 ES 550039 A ES550039 A ES 550039A ES 550039 A ES550039 A ES 550039A ES 550039 A0 ES550039 A0 ES 550039A0
- Authority
- ES
- Spain
- Prior art keywords
- methyl
- methoxy
- azimido
- benzamide
- pirrolidinil
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 238000000034 method Methods 0.000 title abstract 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 3
- KXDAEFPNCMNJSK-UHFFFAOYSA-N Benzamide Chemical compound NC(=O)C1=CC=CC=C1 KXDAEFPNCMNJSK-UHFFFAOYSA-N 0.000 abstract 2
- IJMHZPFHUPXVMQ-UHFFFAOYSA-N 4,5-diacetamido-2-methoxybenzoic acid Chemical compound COC1=CC(NC(C)=O)=C(NC(C)=O)C=C1C(O)=O IJMHZPFHUPXVMQ-UHFFFAOYSA-N 0.000 abstract 1
- LYFZXIXVTGAHSZ-UHFFFAOYSA-N 4,5-diamino-2-methoxybenzoic acid Chemical compound COC1=CC(N)=C(N)C=C1C(O)=O LYFZXIXVTGAHSZ-UHFFFAOYSA-N 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 238000002360 preparation method Methods 0.000 abstract 1
- 238000003786 synthesis reaction Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
- C07D207/09—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pyrrole Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR8419322A FR2574795B1 (fr) | 1984-12-18 | 1984-12-18 | Nouveau procede industriel de synthese du n-((1'-allyl 2'-pyrrolidinyl) methyl) 2-methoxy 4,5-azimido benzamide |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES8703455A1 ES8703455A1 (es) | 1987-02-16 |
| ES550039A0 true ES550039A0 (es) | 1987-02-16 |
Family
ID=9310704
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES550039A Expired ES8703455A1 (es) | 1984-12-18 | 1985-12-17 | Procedimiento para preparar n-(-(1'-alil-2'-pirrolidinil)- metil)-2-metoxi-4,5-azimido-benzamida a escala industrial |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US4804765A (es) |
| EP (1) | EP0190524B1 (es) |
| AT (1) | ATE61366T1 (es) |
| BE (1) | BE903850A (es) |
| CH (1) | CH669380A5 (es) |
| DE (1) | DE3582058D1 (es) |
| ES (1) | ES8703455A1 (es) |
| FR (1) | FR2574795B1 (es) |
| IT (1) | IT1182091B (es) |
| YU (1) | YU44164B (es) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4943574A (en) * | 1987-06-01 | 1990-07-24 | Janssen Pharmaceutica N.V. | (1H-azol-1-ylmethyl) substituted benzotriazole derivatives and pharmaceutical compositions containing them |
| CN113024432A (zh) * | 2019-12-24 | 2021-06-25 | 上海科胜药物研发有限公司 | 一种氨磺必利药典杂质的制备方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA517588A (en) * | 1955-10-18 | General Mills | Process of preparing n-fatty pyrrolidines | |
| FR6787M (es) * | 1967-08-17 | 1969-03-17 | ||
| FR2097041B3 (es) * | 1970-07-29 | 1973-04-27 | Videment Jean | |
| US4039672A (en) * | 1975-01-11 | 1977-08-02 | Societe D'etudes Scientifiques Et Industrielles De L'ile-De-France | N-(1'-allypyrrolidinyl 2'-methyl) 2-methoxy 4,5-azimido benzamide and its pharmaceutically acceptable salts |
| US4146630A (en) * | 1976-11-12 | 1979-03-27 | Boehringer Mannheim Gmbh | Blood pressure lowering and adrenergic β-receptor inhibiting 3-(4-phenoxymethylpiperidino)-propyl-phenyl ethers |
| FR2415099A1 (fr) * | 1978-01-20 | 1979-08-17 | Ile De France | Nouveaux derives de 4-amino-5-alkylsulfonyl ortho-anisamides, leurs procedes de preparation et leur application comme psychotropes |
| FR2440946A2 (fr) * | 1978-01-20 | 1980-06-06 | Ile De France | Nouveaux benzamides heterocycliques substitues, leurs procedes de preparation et leur application comme modificateurs du comportement |
-
1984
- 1984-12-18 FR FR8419322A patent/FR2574795B1/fr not_active Expired
-
1985
- 1985-12-13 YU YU1947/85A patent/YU44164B/xx unknown
- 1985-12-13 BE BE1/011398A patent/BE903850A/fr not_active IP Right Cessation
- 1985-12-16 IT IT48935/85A patent/IT1182091B/it active
- 1985-12-17 AT AT85402512T patent/ATE61366T1/de not_active IP Right Cessation
- 1985-12-17 DE DE8585402512T patent/DE3582058D1/de not_active Expired - Fee Related
- 1985-12-17 EP EP85402512A patent/EP0190524B1/fr not_active Expired - Lifetime
- 1985-12-17 CH CH5367/85A patent/CH669380A5/fr not_active IP Right Cessation
- 1985-12-17 ES ES550039A patent/ES8703455A1/es not_active Expired
- 1985-12-18 US US06/810,669 patent/US4804765A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| YU194785A (en) | 1987-10-31 |
| BE903850A (fr) | 1986-06-13 |
| EP0190524B1 (fr) | 1991-03-06 |
| IT1182091B (it) | 1987-09-30 |
| YU44164B (en) | 1990-02-28 |
| IT8548935A0 (it) | 1985-12-16 |
| FR2574795B1 (fr) | 1987-11-20 |
| US4804765A (en) | 1989-02-14 |
| ATE61366T1 (de) | 1991-03-15 |
| FR2574795A1 (fr) | 1986-06-20 |
| CH669380A5 (es) | 1989-03-15 |
| EP0190524A1 (fr) | 1986-08-13 |
| DE3582058D1 (de) | 1991-04-11 |
| ES8703455A1 (es) | 1987-02-16 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 19960603 |