ES544522A0 - Un procedimiento para la preparacion de analogos de benzodiazepina. - Google Patents
Un procedimiento para la preparacion de analogos de benzodiazepina.Info
- Publication number
- ES544522A0 ES544522A0 ES544522A ES544522A ES544522A0 ES 544522 A0 ES544522 A0 ES 544522A0 ES 544522 A ES544522 A ES 544522A ES 544522 A ES544522 A ES 544522A ES 544522 A0 ES544522 A0 ES 544522A0
- Authority
- ES
- Spain
- Prior art keywords
- procedure
- preparation
- benzodiazepine analogs
- benzodiazepine
- analogs
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
- C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US62485284A | 1984-06-26 | 1984-06-26 | |
US74197385A | 1985-06-10 | 1985-06-10 |
Publications (2)
Publication Number | Publication Date |
---|---|
ES8609278A1 ES8609278A1 (es) | 1986-09-01 |
ES544522A0 true ES544522A0 (es) | 1986-09-01 |
Family
ID=27089772
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES544522A Expired ES8609278A1 (es) | 1984-06-26 | 1985-06-25 | Un procedimiento para la preparacion de analogos de benzodiazepina. |
ES551565A Expired ES8706147A1 (es) | 1984-06-26 | 1986-02-01 | Un procedimiento para la preparacion de analogos de benzodiazepina |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES551565A Expired ES8706147A1 (es) | 1984-06-26 | 1986-02-01 | Un procedimiento para la preparacion de analogos de benzodiazepina |
Country Status (3)
Country | Link |
---|---|
EP (1) | EP0167920A3 (es) |
DK (1) | DK287185A (es) |
ES (2) | ES8609278A1 (es) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4755508A (en) * | 1984-06-26 | 1988-07-05 | Merck & Co., Inc. | Benzodiazepine analogs and use as antogonists of gastrin and cholecystokinin |
US4820834A (en) * | 1984-06-26 | 1989-04-11 | Merck & Co., Inc. | Benzodiazepine analogs |
CA2056809A1 (en) * | 1990-12-07 | 1992-06-08 | Mark G. Bock | Benzodiazepine analogs |
US5206237A (en) * | 1991-05-14 | 1993-04-27 | Merck & Co., Inc. | Benzodiazepine analogs |
US6458784B1 (en) | 1994-06-29 | 2002-10-01 | Smithkline Beecham Corporation | Vitronectin receptor antagonists |
US5977101A (en) * | 1995-06-29 | 1999-11-02 | Smithkline Beecham Corporation | Benzimidazoles/Imidazoles Linked to a Fibrinogen Receptor Antagonist Template Having Vitronectin Receptor Antagonist Activity |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3419545A (en) * | 1961-05-29 | 1968-12-31 | Warner Lambert Pharmaceutical | Process of preparing 7-halo-2-dimethylamino - 5-phenyl-3h-1,4-benzodiazepine 4-oxides |
NL289735A (es) * | 1962-03-09 | |||
US3320239A (en) * | 1965-03-22 | 1967-05-16 | Hoffmann La Roche | Certain 2, 3-bis(substituted amino)-5-aryl-3h-1, 4-benzodiazepine-4-oxide compounds and their preparation |
-
1985
- 1985-06-25 DK DK287185A patent/DK287185A/da not_active Application Discontinuation
- 1985-06-25 EP EP85107844A patent/EP0167920A3/en not_active Withdrawn
- 1985-06-25 ES ES544522A patent/ES8609278A1/es not_active Expired
-
1986
- 1986-02-01 ES ES551565A patent/ES8706147A1/es not_active Expired
Also Published As
Publication number | Publication date |
---|---|
EP0167920A3 (en) | 1986-11-05 |
EP0167920A2 (en) | 1986-01-15 |
ES551565A0 (es) | 1987-06-01 |
DK287185D0 (da) | 1985-06-25 |
ES8706147A1 (es) | 1987-06-01 |
ES8609278A1 (es) | 1986-09-01 |
DK287185A (da) | 1986-02-24 |
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