ES538518A0 - Un procedimiento para preparar derivados de 3-aminopirazolo-(3,4-d)-pirimidina - Google Patents

Un procedimiento para preparar derivados de 3-aminopirazolo-(3,4-d)-pirimidina

Info

Publication number
ES538518A0
ES538518A0 ES538518A ES538518A ES538518A0 ES 538518 A0 ES538518 A0 ES 538518A0 ES 538518 A ES538518 A ES 538518A ES 538518 A ES538518 A ES 538518A ES 538518 A0 ES538518 A0 ES 538518A0
Authority
ES
Spain
Prior art keywords
aminopyrazole
preparing
procedure
pirimidine derivatives
pirimidine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES538518A
Other languages
English (en)
Other versions
ES8608520A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Takeda Pharmaceutical Co Ltd
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP23700083A external-priority patent/JPS60126285A/ja
Priority claimed from JP12568984A external-priority patent/JPS615082A/ja
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of ES538518A0 publication Critical patent/ES538518A0/es
Publication of ES8608520A1 publication Critical patent/ES8608520A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ES538518A 1983-12-14 1984-12-12 Un procedimiento para preparar derivados de 3-aminopirazolo-(3,4-d)-pirimidina Expired ES8608520A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP23700083A JPS60126285A (ja) 1983-12-14 1983-12-14 3−アミノピラゾロ〔3,4−d〕ピリミジン誘導体
JP12568984A JPS615082A (ja) 1984-06-18 1984-06-18 3−アミノピラゾロ〔3,4−d〕ピリミジン誘導体

Publications (2)

Publication Number Publication Date
ES538518A0 true ES538518A0 (es) 1986-06-16
ES8608520A1 ES8608520A1 (es) 1986-06-16

Family

ID=26462044

Family Applications (1)

Application Number Title Priority Date Filing Date
ES538518A Expired ES8608520A1 (es) 1983-12-14 1984-12-12 Un procedimiento para preparar derivados de 3-aminopirazolo-(3,4-d)-pirimidina

Country Status (10)

Country Link
US (1) US4603203A (es)
EP (1) EP0166054B1 (es)
KR (1) KR910006866B1 (es)
CA (1) CA1263386A (es)
DE (1) DE3477783D1 (es)
DK (1) DK165409C (es)
ES (1) ES8608520A1 (es)
GR (1) GR81241B (es)
IE (1) IE58160B1 (es)
PT (1) PT79667B (es)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0237289A3 (en) * 1986-03-14 1988-07-27 Takeda Chemical Industries, Ltd. Pyrazolo [3,4-d] pyrimidine derivatives, their production and use
US4912104A (en) * 1987-08-31 1990-03-27 Takeda Chemical Industries, Ltd. Tricyclic fused pryimidine derivatives, and their use as pharmaceuticals
US4885300A (en) * 1988-03-03 1989-12-05 Ortho Pharmaceutical Corporation 4-Substituted pyrazolo[3,4-D]pyrimidine derivatives
EP0353941A3 (en) * 1988-08-02 1991-05-02 Takeda Chemical Industries, Ltd. Medicament for psoriasis containing derivatives of 3-aminopyrazolo [3,4-d]pyrimidine
JP3116230B2 (ja) * 1989-02-15 2000-12-11 武田薬品工業株式会社 三環式縮合ピリミジン誘導体
US5290782A (en) * 1989-09-01 1994-03-01 Kyowa Hakko Kogyo Co., Ltd. Xanthine derivatives
SE9701398D0 (sv) * 1997-04-15 1997-04-15 Astra Pharma Prod Novel compounds
EP1713815A4 (en) * 2004-02-11 2009-03-11 Smithkline Beecham Corp PTH AGONISTS
WO2007143705A2 (en) 2006-06-06 2007-12-13 Intra-Cellular Therapies, Inc. Organic compounds
JP5701608B2 (ja) 2007-12-06 2015-04-15 イントラ−セルラー・セラピーズ・インコーポレイテッドIntra−Cellular Therapies, Inc. 有機化合物
BRPI0922809A2 (pt) 2008-12-06 2018-05-29 Intracellular Therapies Inc compostos orgânicos
EA201170773A1 (ru) 2008-12-06 2012-01-30 Интра-Селлулар Терапиз, Инк. Органические соединения
EP2367430B1 (en) 2008-12-06 2014-08-13 Intra-Cellular Therapies, Inc. Organic compounds
JP2012526810A (ja) 2009-05-13 2012-11-01 イントラ−セルラー・セラピーズ・インコーポレイテッド 有機化合物
US9434730B2 (en) 2010-05-31 2016-09-06 Intra-Cellular Therapies, Inc. PDE1 inhibitor compounds
EP2590657A4 (en) 2010-05-31 2014-02-12 Intra Cellular Therapies Inc ORGANIC CONNECTIONS
EP2968338B1 (en) 2013-03-15 2019-01-09 Intra-Cellular Therapies, Inc. Pde1 inhibitors for use in the treatment and/or prevention of cns injuries, and pns diseases, disorders or injuries
US9546175B2 (en) 2014-08-07 2017-01-17 Intra-Cellular Therapies, Inc. Organic compounds
US10131671B2 (en) 2014-08-07 2018-11-20 Intra-Cellular Therapies, Inc. Organic compounds
US10285992B2 (en) 2014-08-07 2019-05-14 Intra-Cellular Therapies, Inc. Combinations of PDE1 inhibitors and NEP inhibitors and associated methods
RU2711442C2 (ru) 2014-09-17 2020-01-17 Интра-Селлулар Терапиз, Инк. Соединения и способы
US10105349B2 (en) 2014-12-06 2018-10-23 Intra-Cellular Therapies, Inc. Organic compounds
MX371158B (es) 2014-12-06 2020-01-20 Intra Cellular Therapies Inc Compuestos inhibidores de pde2.
US12364695B2 (en) 2020-06-02 2025-07-22 Intra-Cellular Therapies, Inc. Methods of treating inflammatory disease

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1567781A (en) * 1976-05-15 1980-05-21 Fisons Ltd Pyrazolopyrimidines
JPS58500966A (ja) * 1981-04-22 1983-06-09 ビイク グルデン ロンベルク ヒエ−ミツシエ フアブリ−ク ゲゼルシヤフト ミツト ベシユレンクテル ハフツング 新規ピラゾロ〔3,4−d〕ピリミジン、その製法及びこれを含有する医薬品

Also Published As

Publication number Publication date
IE843207L (en) 1985-06-14
KR910006866B1 (ko) 1991-09-09
DK165409B (da) 1992-11-23
IE58160B1 (en) 1993-07-28
DE3477783D1 (en) 1989-05-24
EP0166054A1 (en) 1986-01-02
ES8608520A1 (es) 1986-06-16
DK165409C (da) 1993-04-05
GR81241B (en) 1985-04-16
KR850004752A (ko) 1985-07-27
PT79667A (en) 1985-01-01
PT79667B (en) 1986-12-10
EP0166054B1 (en) 1989-04-19
DK584284A (da) 1985-06-15
DK584284D0 (da) 1984-12-07
CA1263386A (en) 1989-11-28
US4603203A (en) 1986-07-29

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19970401