ES518137A0 - Procedimiento para la preparacion de n-piridil-amidas de acido 1-fenil-ciclopentancarboxilico. - Google Patents

Procedimiento para la preparacion de n-piridil-amidas de acido 1-fenil-ciclopentancarboxilico.

Info

Publication number
ES518137A0
ES518137A0 ES518137A ES518137A ES518137A0 ES 518137 A0 ES518137 A0 ES 518137A0 ES 518137 A ES518137 A ES 518137A ES 518137 A ES518137 A ES 518137A ES 518137 A0 ES518137 A0 ES 518137A0
Authority
ES
Spain
Prior art keywords
piridil
amides
phenyl
procedure
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES518137A
Other languages
English (en)
Other versions
ES8401942A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Medea Research SRL
Original Assignee
Medea Research SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from IT8125570A external-priority patent/IT1226048B/it
Priority claimed from IT24116/82A external-priority patent/IT1154522B/it
Application filed by Medea Research SRL filed Critical Medea Research SRL
Publication of ES518137A0 publication Critical patent/ES518137A0/es
Publication of ES8401942A1 publication Critical patent/ES8401942A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72Nitrogen atoms
    • C07D213/75Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ES518137A 1981-12-14 1982-12-13 Procedimiento para la preparacion de n-piridil-amidas de acido 1-fenil-ciclopentancarboxilico. Expired ES8401942A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT8125570A IT1226048B (it) 1981-12-14 1981-12-14 Composti ad attivita'antiinfiammatoria, processo per la loro preparazione e composizioni farmaceutiche relative
IT24116/82A IT1154522B (it) 1982-11-08 1982-11-08 Composti ad attivita' antiinfirmmatoria, processo per la loro preparazione e composizioni farmaceutiche relative

Publications (2)

Publication Number Publication Date
ES518137A0 true ES518137A0 (es) 1984-01-16
ES8401942A1 ES8401942A1 (es) 1984-01-16

Family

ID=26328463

Family Applications (1)

Application Number Title Priority Date Filing Date
ES518137A Expired ES8401942A1 (es) 1981-12-14 1982-12-13 Procedimiento para la preparacion de n-piridil-amidas de acido 1-fenil-ciclopentancarboxilico.

Country Status (3)

Country Link
EP (1) EP0081756B1 (es)
DE (1) DE3263567D1 (es)
ES (1) ES8401942A1 (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI1945632T1 (sl) 2005-11-08 2014-03-31 Vertex Pharmaceuticals Incorporated Heterocikliäśni modulatorji za prenaĺ alce z atp-vezavno kaseto
US7671221B2 (en) 2005-12-28 2010-03-02 Vertex Pharmaceuticals Incorporated Modulators of ATP-Binding Cassette transporters
US7754739B2 (en) 2007-05-09 2010-07-13 Vertex Pharmaceuticals Incorporated Modulators of CFTR
JP5497633B2 (ja) 2007-05-09 2014-05-21 バーテックス ファーマシューティカルズ インコーポレイテッド Cftrのモジュレーター
WO2009073757A1 (en) 2007-12-07 2009-06-11 Vertex Pharmaceuticals Incorporated Solid forms of 3-(6-(1-(2,2-difluorobenzo[d][1,3] dioxol-5-yl) cyclopropanecarboxamido)-3-methylpyridin-2-yl) benzoic acid
WO2009076142A2 (en) 2007-12-07 2009-06-18 Vertex Pharmaceuticals Incorporated Processes for producing cycloalkylcarboxiamido-pyridine benzoic acids
CA3039943C (en) 2008-02-28 2021-07-13 Vertex Pharmaceuticals Incorporated Heteroaryl derivatives as cftr modulators
SI2615085T1 (sl) * 2008-03-31 2015-11-30 Vertex Pharmaceuticals Incorporated Piridilni derivati kot cftr-modulatorji
AU2013270464B2 (en) * 2008-03-31 2016-05-26 Vertex Pharmaceuticals Incorporated Pyridyl derivatives as CFTR modulators
CA2795804C (en) 2010-04-07 2021-10-26 Vertex Pharmaceuticals Incorporated Pharmaceutical compositions of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl) cyclopropanecarboxamido)-3-methylpyriodin-2-yl)benzoic acid and administration thereof
CA2930199C (en) 2013-11-12 2022-10-25 Vertex Pharmaceuticals Incorporated Process of preparing pharmaceutical compositions for the treatment of cftr mediated diseases
EP2878339A1 (en) 2013-12-02 2015-06-03 Siena Biotech S.p.A. SIP3 antagonists
PT3221692T (pt) 2014-11-18 2021-09-10 Vertex Pharma Processo de realização de testagem de alta produtividade por cromatografia líquida de alta eficiência

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1584802A (es) * 1968-09-09 1970-01-02

Also Published As

Publication number Publication date
DE3263567D1 (en) 1985-06-20
EP0081756B1 (en) 1985-05-15
EP0081756A1 (en) 1983-06-22
ES8401942A1 (es) 1984-01-16

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 20001009