ES490503A0 - Un procedimiento para preparar nuevos compuestos de cefem - Google Patents

Un procedimiento para preparar nuevos compuestos de cefem

Info

Publication number
ES490503A0
ES490503A0 ES490503A ES490503A ES490503A0 ES 490503 A0 ES490503 A0 ES 490503A0 ES 490503 A ES490503 A ES 490503A ES 490503 A ES490503 A ES 490503A ES 490503 A0 ES490503 A0 ES 490503A0
Authority
ES
Spain
Prior art keywords
procedure
preparing new
cefem compounds
new cefem
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES490503A
Other languages
English (en)
Other versions
ES8103102A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Fujisawa Pharmaceutical Co Ltd
Original Assignee
Fujisawa Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fujisawa Pharmaceutical Co Ltd filed Critical Fujisawa Pharmaceutical Co Ltd
Publication of ES490503A0 publication Critical patent/ES490503A0/es
Publication of ES8103102A1 publication Critical patent/ES8103102A1/es
Priority claimed from AU23283/84A external-priority patent/AU2328384A/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D257/00Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04Five-membered rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/101,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D249/12Oxygen or sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/081,2,4-Thiadiazoles; Hydrogenated 1,2,4-thiadiazoles
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
ES490503A 1978-07-10 1980-04-11 Un procedimiento para preparar nuevos compuestos de cefem Expired ES8103102A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB7829357 1978-07-10
GB7850334 1978-12-29
AU23283/84A AU2328384A (en) 1978-12-29 1984-01-13 1,2,4-thiadiazole derivatives

Publications (2)

Publication Number Publication Date
ES490503A0 true ES490503A0 (es) 1981-02-16
ES8103102A1 ES8103102A1 (es) 1981-02-16

Family

ID=32965858

Family Applications (3)

Application Number Title Priority Date Filing Date
ES482323A Expired ES482323A1 (es) 1978-07-10 1979-07-09 Un procedimiento para preparar nuevos compuestos de cefem.
ES490503A Expired ES8103102A1 (es) 1978-07-10 1980-04-11 Un procedimiento para preparar nuevos compuestos de cefem
ES490504A Expired ES8103072A1 (es) 1978-07-10 1980-04-11 Procedimiento para preparar nuevos compuestos de tiadiazoli-lo

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES482323A Expired ES482323A1 (es) 1978-07-10 1979-07-09 Un procedimiento para preparar nuevos compuestos de cefem.

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES490504A Expired ES8103072A1 (es) 1978-07-10 1980-04-11 Procedimiento para preparar nuevos compuestos de tiadiazoli-lo

Country Status (9)

Country Link
US (3) US4268509A (es)
EP (2) EP0007470B1 (es)
JP (1) JPS63264471A (es)
AR (1) AR226539A1 (es)
AU (1) AU533708B2 (es)
DE (1) DE2966293D1 (es)
DK (1) DK289079A (es)
ES (3) ES482323A1 (es)
HU (1) HU183010B (es)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1592149A (en) * 1976-10-08 1981-07-01 Fujisawa Pharmaceutical Co 3 7-disubstituted-3-cephem-4-carboxylic acid compounds and processes for preparation thereof
FR2387235A1 (fr) * 1978-01-23 1978-11-10 Fujisawa Pharmaceutical Co Procede de preparation de composes d'acide 3,7-disubstitue-3-cephem-4-carboxylique et nouveaux produits ainsi obtenus, ayant une forte activite antibacterienne
US4332798A (en) * 1978-12-29 1982-06-01 Fujisawa Pharmaceutical Co., Ltd. 7-Amino-thia-diazole oxyimino derivatives of cephem and cephem compounds
AU536842B2 (en) * 1978-12-29 1984-05-24 Fujisawa Pharmaceutical Co., Ltd. Cephalosporin antibiotics
US4390534A (en) * 1978-12-29 1983-06-28 Fujisawa Pharmaceutical Co., Ltd. Cephem and cepham compounds
US4567275A (en) * 1978-12-29 1986-01-28 Fujisawa Pharmaceutical Co., Ltd. Cephem and cepham compounds and processes for preparation thereof
US4331666A (en) * 1979-05-11 1982-05-25 Farmitalia Carlo Erba S.P.A. 3-[(8-Carboxy-6-tetrazolo[1,5-b]pyridazinyl)-thiomethyl]-7-[2-(2-amino-4-thiazolyl)-2-methoxyimino-acetamido]-3-cephem-4-carboxylic acid
MA18891A1 (fr) * 1979-07-05 1981-04-01 Ciba Geigy Ag Composes d'amino-thiadiazolyle,procede pour leur preparation
EP0025017A1 (de) * 1979-08-28 1981-03-11 Ciba-Geigy Ag Polyazathiaverbindungen, Verfahren zu ihrer Herstellung, pharmazeutische Präparate enthaltend solche Verbindungen und Verwendung von letzteren
US4381299A (en) * 1980-03-07 1983-04-26 Fujisawa Pharmaceutical Co., Ltd. 7-Amino-thiadiazole oxyimino derivatives of cephem and cepham compounds
US4405617A (en) * 1980-02-11 1983-09-20 Fujisawa Pharmaceutical Co., Ltd. 3-(Propynyltetrazol)thiomethyl-3-cephems
GR78245B (es) * 1980-09-12 1984-09-26 Ciba Geigy Ag
US4431642A (en) * 1980-12-01 1984-02-14 Fujisawa Pharmaceutical Co., Ltd. Cephem compounds
US4521413A (en) * 1981-09-14 1985-06-04 Fujisawa Pharmaceutical Co., Ltd. Cephem compounds
US4563449A (en) * 1982-07-19 1986-01-07 Fujisawa Pharmaceutical Co., Ltd. Cephem compounds
CA1293719C (en) * 1986-09-22 1991-12-31 Takao Takaya Cephem compounds and processes for preparation thereof
FR2729948A1 (fr) * 1995-01-31 1996-08-02 Oreal Nouveaux derives d'arginine, procede de preparation, utilisations et compositions les comprenant
TW473479B (en) * 1997-12-19 2002-01-21 Takeda Chemical Industries Ltd Phosphonocephem derivatives, their production and use
US8673894B2 (en) 2010-05-07 2014-03-18 Hoffmann-La Roche Inc. 2,5,6,7-tetrahydro-[1,4]oxazepin-3-ylamine or 2,3,6,7-tetrahydro-[1,4]oxazepin-5-ylamine compounds
US20130065874A1 (en) 2011-09-09 2013-03-14 Cubist Pharmaceuticals, Inc. Methods for treating intrapulmonary infections
US8809314B1 (en) 2012-09-07 2014-08-19 Cubist Pharmacueticals, Inc. Cephalosporin compound
US8476425B1 (en) 2012-09-27 2013-07-02 Cubist Pharmaceuticals, Inc. Tazobactam arginine compositions
UY35103A (es) 2012-10-29 2014-05-30 Glaxo Group Ltd Compuestos de cefem 2-sustituidos
US9872906B2 (en) 2013-03-15 2018-01-23 Merck Sharp & Dohme Corp. Ceftolozane antibiotic compositions
CA2906151A1 (en) 2013-03-15 2014-09-18 Merck Sharp & Dohme Corp. Ceftolozane antibiotic compositions
US20140274997A1 (en) 2013-03-15 2014-09-18 Cubist Pharmaceuticals, Inc. Cephalosporin pharmaceutical compositions
WO2015035376A2 (en) 2013-09-09 2015-03-12 Calixa Therapeutics, Inc. Treating infections with ceftolozane/tazobactam in subjects having impaired renal function
US8906898B1 (en) 2013-09-27 2014-12-09 Calixa Therapeutics, Inc. Solid forms of ceftolozane

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1399086A (en) * 1971-05-14 1975-06-25 Glaxo Lab Ltd Cephalosporin compounds
US4093803A (en) * 1971-05-14 1978-06-06 Glaxo Laboratories Limited 7β-[2-Etherified oximino-2-(thienyl-, furyl- or pyridylacetamido)] cephalosporins
BE791214A (fr) * 1972-05-08 1973-05-10 Glaxo Lab Ltd Procede de preparation d'isomeres de derives d'acide hydroxyiminoacetique etherifie purs
DK154939C (da) * 1974-12-19 1989-06-12 Takeda Chemical Industries Ltd Analogifremgangsmaade til fremstilling af thiazolylacetamido-cephemforbindelser eller farmaceutisk acceptable salte eller estere deraf
US4166115A (en) * 1976-04-12 1979-08-28 Fujisawa Pharmaceutical Co., Ltd. Syn 7-oxoimino substituted derivatives of cephalosporanic acid
GB1592149A (en) 1976-10-08 1981-07-01 Fujisawa Pharmaceutical Co 3 7-disubstituted-3-cephem-4-carboxylic acid compounds and processes for preparation thereof
PH17188A (en) * 1977-03-14 1984-06-14 Fujisawa Pharmaceutical Co New cephem and cepham compounds and their pharmaceutical compositions and method of use
US4468515A (en) * 1978-12-29 1984-08-28 Fujisawa Pharmaceutical Co., Ltd. 2-Substituted oxyimino-2-(5-amino-1,2,4-thiadiazol-3-yl)acetic acids

Also Published As

Publication number Publication date
AU4869579A (en) 1980-02-07
EP0007470A2 (en) 1980-02-06
DE2966293D1 (en) 1983-11-17
JPS63264471A (ja) 1988-11-01
US4447429A (en) 1984-05-08
ES482323A1 (es) 1980-08-16
US4585872A (en) 1986-04-29
ES490504A0 (es) 1981-02-16
ES8103102A1 (es) 1981-02-16
US4268509A (en) 1981-05-19
AU533708B2 (en) 1983-12-08
ES8103072A1 (es) 1981-02-16
EP0036673A1 (en) 1981-09-30
AR226539A1 (es) 1982-07-30
DK289079A (da) 1980-01-11
JPH0368028B2 (es) 1991-10-25
EP0007470B1 (en) 1983-10-12
EP0007470A3 (en) 1980-04-16
EP0036673B1 (en) 1984-07-11
HU183010B (en) 1984-04-28

Similar Documents

Publication Publication Date Title
ES490503A0 (es) Un procedimiento para preparar nuevos compuestos de cefem
ES496948A0 (es) Un procedimiento para preparar compuestos de cefem
AR226423A1 (es) Un procedimiento para preparar compuestos de acidos 3-cefem-4-carboxilicos-7-sustituidos
MX5973E (es) Procedimiento para preparar compuestos cefem
ES489222A0 (es) Un procedimiento para preparar un compuesto de guanidinotia-zol
ES493061A0 (es) Un procedimiento para preparar un lipopolisacarido
ES490166A0 (es) Un procedimiento para preparar mercaptoacildipeptidos
ES487847A0 (es) Un procedimiento para preparar nuevas fenetanolaminas
ES492032A0 (es) Procedimiento para preparar compuestos de cefem
ES492002A0 (es) Un procedimiento para preparar compuestos de cefem
AR222999A1 (es) Un procedimiento para preparar compuestos de imidazolilo
ES486425A0 (es) Un procedimiento para preparar nuevas 4-arilpiperinas.
ES503134A0 (es) Un procedimiento para preparar nuevos compuestos de cefem
ES497302A0 (es) Un procedimiento para preparar 9-aminoalquilfluorenos
ES491221A0 (es) Un procedimiento para preparar un compuesto de 1,8-naftiri- dina
AR223978A1 (es) Un procedimiento para preparar un mercaptano
ES505498A0 (es) Un procedimiento para preparar nuevos compuestos de cefem
ES494459A0 (es) Un procedimiento para preparar cetoximinoeteres
ES505496A0 (es) Un procedimiento para preparar nuevos compuestos de cefem
AR226420A1 (es) Un procedimiento para preparar compuestos de s o o-isotioureido o isoureido-alquilen(c3-c8)-amino-5-piridilmetil-4-pirimidona
ES493759A0 (es) Un procedimiento para preparar benzoxazepinas
ES489590A0 (es) Un procedimiento para preparar arilalquil- y ariloxi-alquil-fosfonatos
AR226418A1 (es) Un procedimiento para preparar compuestos de 2,4-dicloro-piridina
ES505714A0 (es) Un procedimiento para preparar compuestos de cefem
ES498168A0 (es) Un procedimiento para preparar alcohilfosfonoditioato de al-cohilo

Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19990301