ES458709A1 - Procedimiento para la preparacion de benzamidas de 3-amino- pirrolidinas. - Google Patents
Procedimiento para la preparacion de benzamidas de 3-amino- pirrolidinas.Info
- Publication number
- ES458709A1 ES458709A1 ES458709A ES458709A ES458709A1 ES 458709 A1 ES458709 A1 ES 458709A1 ES 458709 A ES458709 A ES 458709A ES 458709 A ES458709 A ES 458709A ES 458709 A1 ES458709 A1 ES 458709A1
- Authority
- ES
- Spain
- Prior art keywords
- treating allergy
- aminopyrrolidines
- ameliorating
- asthma
- disclosed
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyrrole Compounds (AREA)
Abstract
Un procedimiento para la preparación de benzamidas de 3-aminopirrolidinas que tienen la fórmula: *** ver imagen 01 donde: R es hidrógeno, cicloalcohilo inferior, fenil-alcohilo inferior o alcohilo inferior, R1 es hidrógeno o alcohilo inferior, X es hidrógeno, nitro, amino, acetamida, dialcohilamino inferior, hidroxilo, alcohilo o alcoxi inferior o alcohilo inferior-sulfonilamino, e Y es hidrógeno, nitro o sulfamoílo, caracterizado por el hecho de que una 3-aminopirrolidina que tiene la fórmula *** ver imagen 02 o alcohilo inferior-sulfonilamino , e Y es hidrógeno, nitro o sulfamoílo, caracterizado por el hecho de que una 3-aminopirrolidina que tiene la fórmula *** ver imagen 03
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US05/685,576 US4049821A (en) | 1976-05-12 | 1976-05-12 | Method of treating allergy |
Publications (1)
Publication Number | Publication Date |
---|---|
ES458709A1 true ES458709A1 (es) | 1978-03-01 |
Family
ID=24752795
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES458709A Expired ES458709A1 (es) | 1976-05-12 | 1977-05-11 | Procedimiento para la preparacion de benzamidas de 3-amino- pirrolidinas. |
Country Status (17)
Country | Link |
---|---|
US (1) | US4049821A (es) |
JP (1) | JPS52142061A (es) |
AU (1) | AU516329B2 (es) |
BE (1) | BE854507A (es) |
DE (1) | DE2721259A1 (es) |
DK (1) | DK207677A (es) |
ES (1) | ES458709A1 (es) |
FI (1) | FI771499A (es) |
FR (1) | FR2421613A1 (es) |
GB (1) | GB1582163A (es) |
IE (1) | IE45384B1 (es) |
NL (1) | NL7705215A (es) |
NZ (1) | NZ184073A (es) |
PH (1) | PH13688A (es) |
PT (1) | PT66532B (es) |
SE (1) | SE7705445L (es) |
ZA (1) | ZA772527B (es) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4544654A (en) * | 1984-03-20 | 1985-10-01 | Schering A.G. | Substituted sulfonamidobenzamides, antiarrhythmic agents and compositions thereof |
JP2002505684A (ja) * | 1997-06-18 | 2002-02-19 | メルク エンド カンパニー インコーポレーテッド | α1aアドレナリン受容体拮抗薬 |
US6037354A (en) * | 1997-06-18 | 2000-03-14 | Merck & Co., Inc. | Alpha 1a adrenergic receptor antagonists |
FR2812635B1 (fr) * | 2000-08-01 | 2002-10-11 | Aventis Pharma Sa | Nouveaux composes heterocycliques, preparation et utilisation comme medicaments notamment comme anti- bacteriens |
US6673829B2 (en) * | 2001-09-14 | 2004-01-06 | Novo Nordisk A/S | Aminoazetidine,-pyrrolidine and -piperidine derivatives |
JP4619655B2 (ja) | 2001-09-14 | 2011-01-26 | ハイ・ポイント・ファーマスーティカルズ、エルエルシー | 新規アミノアゼチジン、−ピロリジンおよび−ピペリジン誘導体 |
US7141529B2 (en) * | 2003-03-21 | 2006-11-28 | Chevron U.S.A. Inc. | Metal loaded microporous material for hydrocarbon isomerization processes |
JP2008502684A (ja) * | 2004-06-15 | 2008-01-31 | メルク エンド カムパニー インコーポレーテッド | アルツハイマー病を治療するためのベータ−セクレターゼ阻害剤として有用なピロリジン−3−イル化合物 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3342826A (en) * | 1964-01-13 | 1967-09-19 | Ile De France | Heterocyclic aminoalkyl benzamides |
GB1364231A (en) * | 1968-12-23 | 1974-08-21 | Robins Co Inc A H | N-/1-substituted-3-pyrrolidinyl/benzamides and thiobenzamides |
US3577440A (en) * | 1968-12-23 | 1971-05-04 | Robins Co Inc A H | 1-substituted-3-amido-pyrrolidines |
GB1392194A (en) * | 1971-09-23 | 1975-04-30 | Wyeth John & Brother Ltd | Pyrrolidine derivatives |
US3966957A (en) * | 1972-04-03 | 1976-06-29 | A. H. Robins Company, Incorporated | Method for controlling emesis with N-(1-substituted-3-pyrrolidinyl)benzamides and thiobenzamides |
-
1976
- 1976-05-12 US US05/685,576 patent/US4049821A/en not_active Expired - Lifetime
-
1977
- 1977-04-27 ZA ZA00772527A patent/ZA772527B/xx unknown
- 1977-05-10 SE SE7705445A patent/SE7705445L/xx unknown
- 1977-05-10 FR FR7714283A patent/FR2421613A1/fr not_active Withdrawn
- 1977-05-11 BE BE177478A patent/BE854507A/xx not_active IP Right Cessation
- 1977-05-11 PT PT66532A patent/PT66532B/pt unknown
- 1977-05-11 NZ NZ184073A patent/NZ184073A/en unknown
- 1977-05-11 ES ES458709A patent/ES458709A1/es not_active Expired
- 1977-05-11 NL NL7705215A patent/NL7705215A/xx unknown
- 1977-05-11 FI FI771499A patent/FI771499A/fi not_active Application Discontinuation
- 1977-05-11 DK DK207677A patent/DK207677A/da unknown
- 1977-05-11 PH PH19762A patent/PH13688A/en unknown
- 1977-05-11 GB GB19797/77A patent/GB1582163A/en not_active Expired
- 1977-05-11 DE DE19772721259 patent/DE2721259A1/de active Granted
- 1977-05-12 JP JP5482077A patent/JPS52142061A/ja active Pending
- 1977-05-12 IE IE976/77A patent/IE45384B1/en unknown
- 1977-05-12 AU AU25107/77A patent/AU516329B2/en not_active Expired
Also Published As
Publication number | Publication date |
---|---|
NL7705215A (nl) | 1977-11-15 |
FR2421613A1 (fr) | 1979-11-02 |
ZA772527B (en) | 1978-04-26 |
PT66532B (en) | 1978-10-17 |
GB1582163A (en) | 1980-12-31 |
JPS52142061A (en) | 1977-11-26 |
SE7705445L (sv) | 1977-11-13 |
BE854507A (fr) | 1977-09-01 |
FI771499A (es) | 1977-11-13 |
IE45384L (en) | 1977-11-12 |
IE45384B1 (en) | 1982-08-11 |
AU516329B2 (en) | 1981-05-28 |
NZ184073A (en) | 1985-03-20 |
DE2721259A1 (de) | 1977-11-24 |
PH13688A (en) | 1980-09-01 |
DK207677A (da) | 1977-11-13 |
PT66532A (en) | 1977-06-01 |
DE2721259C2 (es) | 1988-04-28 |
US4049821A (en) | 1977-09-20 |
AU2510777A (en) | 1978-11-16 |
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