ES458709A1 - Procedimiento para la preparacion de benzamidas de 3-amino- pirrolidinas. - Google Patents

Procedimiento para la preparacion de benzamidas de 3-amino- pirrolidinas.

Info

Publication number
ES458709A1
ES458709A1 ES458709A ES458709A ES458709A1 ES 458709 A1 ES458709 A1 ES 458709A1 ES 458709 A ES458709 A ES 458709A ES 458709 A ES458709 A ES 458709A ES 458709 A1 ES458709 A1 ES 458709A1
Authority
ES
Spain
Prior art keywords
treating allergy
aminopyrrolidines
ameliorating
asthma
disclosed
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES458709A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
AH Robins Co Inc
Original Assignee
AH Robins Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by AH Robins Co Inc filed Critical AH Robins Co Inc
Publication of ES458709A1 publication Critical patent/ES458709A1/es
Expired legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)

Abstract

Un procedimiento para la preparación de benzamidas de 3-aminopirrolidinas que tienen la fórmula: *** ver imagen 01 donde: R es hidrógeno, cicloalcohilo inferior, fenil-alcohilo inferior o alcohilo inferior, R1 es hidrógeno o alcohilo inferior, X es hidrógeno, nitro, amino, acetamida, dialcohilamino inferior, hidroxilo, alcohilo o alcoxi inferior o alcohilo inferior-sulfonilamino, e Y es hidrógeno, nitro o sulfamoílo, caracterizado por el hecho de que una 3-aminopirrolidina que tiene la fórmula *** ver imagen 02 o alcohilo inferior-sulfonilamino , e Y es hidrógeno, nitro o sulfamoílo, caracterizado por el hecho de que una 3-aminopirrolidina que tiene la fórmula *** ver imagen 03
ES458709A 1976-05-12 1977-05-11 Procedimiento para la preparacion de benzamidas de 3-amino- pirrolidinas. Expired ES458709A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/685,576 US4049821A (en) 1976-05-12 1976-05-12 Method of treating allergy

Publications (1)

Publication Number Publication Date
ES458709A1 true ES458709A1 (es) 1978-03-01

Family

ID=24752795

Family Applications (1)

Application Number Title Priority Date Filing Date
ES458709A Expired ES458709A1 (es) 1976-05-12 1977-05-11 Procedimiento para la preparacion de benzamidas de 3-amino- pirrolidinas.

Country Status (17)

Country Link
US (1) US4049821A (es)
JP (1) JPS52142061A (es)
AU (1) AU516329B2 (es)
BE (1) BE854507A (es)
DE (1) DE2721259A1 (es)
DK (1) DK207677A (es)
ES (1) ES458709A1 (es)
FI (1) FI771499A (es)
FR (1) FR2421613A1 (es)
GB (1) GB1582163A (es)
IE (1) IE45384B1 (es)
NL (1) NL7705215A (es)
NZ (1) NZ184073A (es)
PH (1) PH13688A (es)
PT (1) PT66532B (es)
SE (1) SE7705445L (es)
ZA (1) ZA772527B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4544654A (en) * 1984-03-20 1985-10-01 Schering A.G. Substituted sulfonamidobenzamides, antiarrhythmic agents and compositions thereof
JP2002505684A (ja) * 1997-06-18 2002-02-19 メルク エンド カンパニー インコーポレーテッド α１ａアドレナリン受容体拮抗薬
US6037354A (en) * 1997-06-18 2000-03-14 Merck & Co., Inc. Alpha 1a adrenergic receptor antagonists
FR2812635B1 (fr) * 2000-08-01 2002-10-11 Aventis Pharma Sa Nouveaux composes heterocycliques, preparation et utilisation comme medicaments notamment comme anti- bacteriens
US6673829B2 (en) * 2001-09-14 2004-01-06 Novo Nordisk A/S Aminoazetidine,-pyrrolidine and -piperidine derivatives
JP4619655B2 (ja) 2001-09-14 2011-01-26 ハイ・ポイント・ファーマスーティカルズ、エルエルシー 新規アミノアゼチジン、−ピロリジンおよび−ピペリジン誘導体
US7141529B2 (en) * 2003-03-21 2006-11-28 Chevron U.S.A. Inc. Metal loaded microporous material for hydrocarbon isomerization processes
JP2008502684A (ja) * 2004-06-15 2008-01-31 メルク　エンド　カムパニー　インコーポレーテッド アルツハイマー病を治療するためのベータ−セクレターゼ阻害剤として有用なピロリジン−３−イル化合物

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3342826A (en) * 1964-01-13 1967-09-19 Ile De France Heterocyclic aminoalkyl benzamides
GB1364231A (en) * 1968-12-23 1974-08-21 Robins Co Inc A H N-/1-substituted-3-pyrrolidinyl/benzamides and thiobenzamides
US3577440A (en) * 1968-12-23 1971-05-04 Robins Co Inc A H 1-substituted-3-amido-pyrrolidines
GB1392194A (en) * 1971-09-23 1975-04-30 Wyeth John & Brother Ltd Pyrrolidine derivatives
US3966957A (en) * 1972-04-03 1976-06-29 A. H. Robins Company, Incorporated Method for controlling emesis with N-(1-substituted-3-pyrrolidinyl)benzamides and thiobenzamides

Also Published As

Publication number Publication date
NL7705215A (nl) 1977-11-15
FR2421613A1 (fr) 1979-11-02
ZA772527B (en) 1978-04-26
PT66532B (en) 1978-10-17
GB1582163A (en) 1980-12-31
JPS52142061A (en) 1977-11-26
SE7705445L (sv) 1977-11-13
BE854507A (fr) 1977-09-01
FI771499A (es) 1977-11-13
IE45384L (en) 1977-11-12
IE45384B1 (en) 1982-08-11
AU516329B2 (en) 1981-05-28
NZ184073A (en) 1985-03-20
DE2721259A1 (de) 1977-11-24
PH13688A (en) 1980-09-01
DK207677A (da) 1977-11-13
PT66532A (en) 1977-06-01
DE2721259C2 (es) 1988-04-28
US4049821A (en) 1977-09-20
AU2510777A (en) 1978-11-16

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