ES426124A1 - Procedure for the preparation of new derivatives of cefalosporanic acid. (Machine-translation by Google Translate, not legally binding) - Google Patents
Procedure for the preparation of new derivatives of cefalosporanic acid. (Machine-translation by Google Translate, not legally binding)Info
- Publication number
- ES426124A1 ES426124A1 ES426124A ES426124A ES426124A1 ES 426124 A1 ES426124 A1 ES 426124A1 ES 426124 A ES426124 A ES 426124A ES 426124 A ES426124 A ES 426124A ES 426124 A1 ES426124 A1 ES 426124A1
- Authority
- ES
- Spain
- Prior art keywords
- group
- formula
- hydrogen atom
- amino
- translation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Cephalosporin Compounds (AREA)
Abstract
Preparation procedure, of new cephalosporanic acid derivatives of the formula: **(See formula)** wherein R1 is a nitro group, an alkoxy group, an alkanesulfonamido group or an alkolaminosulfonamido group, R2 is a hydrogen atom or a hydroxyl group, provided that R2 is a hydroxyl group when R1 is a nitro group or an alkoxy group ; R3 is a hydrogen atom or a heterocyclicothio group, in which the heterocyclic group may be substituted with an alcohol group, provided that R3 is a hydrogen atom when R1 is an alkoxy group and R2 is a hydroxyl group; X is an amino group or a protected amino group; M is a pharmaceutically acceptable, non-toxic hydrogen atom or cation; comprising reacting 7-amino-3-cephem-4-carboxylic acids substituted in position 3 of the formula: **(See formula)** wherein R3 and M are as defined above, or their derivatives at the carboxyl and/or amino groups, with substituted phenylglycine of the formula: **(See formula)** wherein R1, R2 and X are as defined above, or their reactive derivatives on the carboxyl group, and, if desired, remove the protecting group from the amino group from the reaction product. (Machine-translation by Google Translate, not legally binding)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP5231273A JPS49135989A (en) | 1973-05-10 | 1973-05-10 | |
JP48076785A JPS5934715B2 (en) | 1973-07-06 | 1973-07-06 | Method for producing 7-substituted acylamino-3-substituted-3-cephem-4-carboxylic acids |
JP49016552A JPS5857438B2 (en) | 1974-02-07 | 1974-02-07 | 7- dithicanphenylglycinamide -luka methyl -3- cefem -4- carbonsanyudotai no seizouhou |
Publications (1)
Publication Number | Publication Date |
---|---|
ES426124A1 true ES426124A1 (en) | 1976-11-01 |
Family
ID=27281453
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES426124A Expired ES426124A1 (en) | 1973-05-10 | 1974-05-09 | Procedure for the preparation of new derivatives of cefalosporanic acid. (Machine-translation by Google Translate, not legally binding) |
Country Status (1)
Country | Link |
---|---|
ES (1) | ES426124A1 (en) |
-
1974
- 1974-05-09 ES ES426124A patent/ES426124A1/en not_active Expired
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