ES426003A1 - Un procedimiento para preparar nuevos compuestos de cefa- losporina. - Google Patents
Un procedimiento para preparar nuevos compuestos de cefa- losporina.Info
- Publication number
- ES426003A1 ES426003A1 ES426003A ES426003A ES426003A1 ES 426003 A1 ES426003 A1 ES 426003A1 ES 426003 A ES426003 A ES 426003A ES 426003 A ES426003 A ES 426003A ES 426003 A1 ES426003 A1 ES 426003A1
- Authority
- ES
- Spain
- Prior art keywords
- amino
- ureidophenyl
- acetamidocephalosporins
- alpha
- aminocephalosporin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 229930186147 Cephalosporin Natural products 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 230000010933 acylation Effects 0.000 abstract 1
- 238000005917 acylation reaction Methods 0.000 abstract 1
- -1 alpha -amino-(ureidophenyl)acetamido substituent Chemical group 0.000 abstract 1
- 239000003242 anti bacterial agent Substances 0.000 abstract 1
- 229940124587 cephalosporin Drugs 0.000 abstract 1
- 150000001780 cephalosporins Chemical class 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/02—Preparation
- C07D501/04—Preparation from compounds already containing the ring or condensed ring systems, e.g. by dehydrogenation of the ring, by introduction, elimination or modification of substituents
- C07D501/06—Acylation of 7-aminocephalosporanic acid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C275/28—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C275/42—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by carboxyl groups
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Cephalosporin Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/357,763 US4007173A (en) | 1973-05-07 | 1973-05-07 | α-amino-α-(ureidophenyl)acetamidocephalosporins |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES426003A1 true ES426003A1 (es) | 1976-07-01 |
Family
ID=23406931
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES426003A Expired ES426003A1 (es) | 1973-05-07 | 1974-05-06 | Un procedimiento para preparar nuevos compuestos de cefa- losporina. |
Country Status (22)
| Country | Link |
|---|---|
| US (5) | US4007173A (es) |
| JP (1) | JPS5013391A (es) |
| AR (1) | AR206315A1 (es) |
| AT (1) | AT329753B (es) |
| AU (1) | AU475779B2 (es) |
| BE (1) | BE814546A (es) |
| CA (1) | CA1041085A (es) |
| CH (1) | CH595389A5 (es) |
| CS (1) | CS181264B2 (es) |
| DD (1) | DD114267A5 (es) |
| DE (1) | DE2422068A1 (es) |
| ES (1) | ES426003A1 (es) |
| FR (2) | FR2228475B1 (es) |
| GB (2) | GB1456144A (es) |
| HU (1) | HU168312B (es) |
| IE (1) | IE39549B1 (es) |
| IL (1) | IL44680A (es) |
| IN (1) | IN141295B (es) |
| LU (1) | LU69997A1 (es) |
| NL (1) | NL7405990A (es) |
| SE (1) | SE430506B (es) |
| ZA (1) | ZA742353B (es) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5716116B2 (es) * | 1974-02-08 | 1982-04-02 | ||
| US4060610A (en) | 1974-12-27 | 1977-11-29 | Smithkline Corporation | Pharmaceutical compositions comprising 7-acyl-3-(substituted triazolyl thiomethyl)-cephalosporins and methods of treating bacterial infections |
| US3989694A (en) | 1974-12-27 | 1976-11-02 | Smithkline Corporation | 7-Acyl-3-(substituted triazolyl thiomethyl)cephalosporins |
| US4286089A (en) | 1974-12-27 | 1981-08-25 | Smithkline Corporation | 7-Acyl-3-(substituted tetrazolyl thiomethyl)cephalosporins |
| US4080451A (en) * | 1975-03-27 | 1978-03-21 | Pfizer Inc. | Cephalosporin derivatives |
| US4183925A (en) * | 1975-03-27 | 1980-01-15 | Pfizer Inc. | 7-Aminophenylacetamido-Δ3 -cephem antibacterial agents and method of use |
| US4254273A (en) * | 1975-06-11 | 1981-03-03 | Merck & Co., Inc. | Process for preparing esters of α-methyl-3,4-dihydroxyphenylalanine |
| US4220644A (en) | 1976-05-03 | 1980-09-02 | Smithkline Corporation | 7-Acylamino-3-(substituted tetrazolyl thiomethyl) cephalosporins |
| GB1579532A (en) * | 1976-05-21 | 1980-11-19 | Farmaceutici Italia | Cephalosporins |
| US4236001A (en) * | 1976-12-01 | 1980-11-25 | Smithkline Corporation | 7β-Acyloxy-3-heterocyclicthiomethyl cephalosporins |
| LU77786A1 (de) * | 1977-07-15 | 1979-03-26 | Ciba Geigy Ag | Verfahren zur herstellung neuer benzopyranderivate |
| EP0016900B1 (de) * | 1977-07-18 | 1983-11-16 | Ciba-Geigy Ag | Zwischenprodukte für die Herstellung von Cephalosporinderivaten, Verfahren zu ihrer Herstellung und Verwendung |
| US4313945A (en) * | 1978-11-23 | 1982-02-02 | Ciba-Geigy Corporation | 7-Thiazolyl-acetamido-cephem derivatives with terminal aminocarboxylic acid grouping |
| US4409215A (en) * | 1979-11-19 | 1983-10-11 | Fujisawa Pharmaceutical Co., Ltd. | 7-Acylamino-3-substituted cephalosporanic acid derivatives and processes for the preparation thereof |
| US5256405A (en) * | 1991-12-30 | 1993-10-26 | Tom's Of Maine | Herbal deodorant |
| AU2629795A (en) * | 1994-12-12 | 1996-07-03 | Chugai Seiyaku Kabushiki Kaisha | Aniline derivative having the effect of inhibiting nitrogen monoxide synthase |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3341531A (en) * | 1967-02-15 | 1967-09-12 | American Cyanamid Co | Substituted 7-acetylamino cephalosporanic acids |
| US3464985A (en) * | 1967-08-18 | 1969-09-02 | Bristol Myers Co | 7 - (d - alpha - amino - (acetamidophenylacetamido))-cephalosporanic acids and derivatives thereof |
| US3573295A (en) * | 1968-07-01 | 1971-03-30 | Bristol Myers Co | Process for the preparation of 7-aminocephalosporanic acid |
| US3641021A (en) * | 1969-04-18 | 1972-02-08 | Lilly Co Eli | 3 7-(ring-substituted) cephalosporin compounds |
| US3634418A (en) * | 1969-08-20 | 1972-01-11 | Bristol Myers Co | 3 - azidomethyl - 7-(alpha-aminophenyl(or thienyl)acetamido)ceph - 3 -em-4-oic acids |
| US3692779A (en) * | 1970-08-12 | 1972-09-19 | Bristol Myers Co | 7-{8 n-(substituted-imidoyl)aminoacetamide{9 cephalosporanic acids and derivatives thereof |
| US3855213A (en) * | 1971-02-18 | 1974-12-17 | Smith Kline French Lab | 3-heterocyclic thiomethyl-cephalosporins |
| US3867380A (en) * | 1971-02-18 | 1975-02-18 | Smithkline Corp | 3-Heterocyclic thiomethylcephalosporins |
| US3704297A (en) * | 1971-03-05 | 1972-11-28 | American Home Prod | 7 - (1,4 - cyclohexadienylacylamido)cephalosporanic acids and related compounds |
| US3813376A (en) * | 1972-08-31 | 1974-05-28 | Bristol Myers Co | 7-(o-aminomethylphenyl-acetamido)-3-(3-hydroxypyridazin-6-ylthiomethyl)-3-cephem-4-carboxylic acid |
| AR205537A1 (es) * | 1973-05-10 | 1976-05-14 | Fujisawa Pharmaceutical Co | Procedimiento para la preparacion de derivados de acido 7-substituido fenilglicinamido - 3 - substituido - 3 - cefem - 4 - carboxilicos |
-
1973
- 1973-05-07 US US05/357,763 patent/US4007173A/en not_active Expired - Lifetime
-
1974
- 1974-01-01 AR AR253626A patent/AR206315A1/es active
- 1974-04-11 ZA ZA00742353A patent/ZA742353B/xx unknown
- 1974-04-22 IL IL44680A patent/IL44680A/en unknown
- 1974-04-24 CA CA198,020A patent/CA1041085A/en not_active Expired
- 1974-04-29 SE SE7405695A patent/SE430506B/xx unknown
- 1974-04-30 GB GB1883474A patent/GB1456144A/en not_active Expired
- 1974-04-30 GB GB22076A patent/GB1456145A/en not_active Expired
- 1974-05-01 JP JP49049628A patent/JPS5013391A/ja active Pending
- 1974-05-02 CH CH600274A patent/CH595389A5/xx not_active IP Right Cessation
- 1974-05-03 NL NL7405990A patent/NL7405990A/xx not_active Application Discontinuation
- 1974-05-03 BE BE143918A patent/BE814546A/xx not_active IP Right Cessation
- 1974-05-06 LU LU69997A patent/LU69997A1/xx unknown
- 1974-05-06 ES ES426003A patent/ES426003A1/es not_active Expired
- 1974-05-06 DD DD178295A patent/DD114267A5/xx unknown
- 1974-05-06 AU AU68656/74A patent/AU475779B2/en not_active Expired
- 1974-05-06 AT AT369374A patent/AT329753B/de not_active IP Right Cessation
- 1974-05-07 FR FR7415681A patent/FR2228475B1/fr not_active Expired
- 1974-05-07 DE DE2422068A patent/DE2422068A1/de not_active Withdrawn
- 1974-05-07 CS CS7400003283A patent/CS181264B2/cs unknown
- 1974-05-07 HU HUSI1401A patent/HU168312B/hu unknown
- 1974-05-07 IE IE965/74A patent/IE39549B1/xx unknown
-
1975
- 1975-04-18 IN IN774/CAL/1975A patent/IN141295B/en unknown
- 1975-11-21 FR FR7535593A patent/FR2299318A1/fr active Granted
-
1976
- 1976-10-01 US US05/728,583 patent/US4067977A/en not_active Expired - Lifetime
- 1976-10-01 US US05/728,582 patent/US4067978A/en not_active Expired - Lifetime
- 1976-10-01 US US05/728,580 patent/US4067976A/en not_active Expired - Lifetime
- 1976-10-10 US US05/728,581 patent/US4091227A/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| JPS5013391A (es) | 1975-02-12 |
| NL7405990A (es) | 1974-11-11 |
| ATA369374A (de) | 1975-08-15 |
| IE39549L (en) | 1974-11-07 |
| CH595389A5 (es) | 1978-02-15 |
| AT329753B (de) | 1976-05-25 |
| BE814546A (fr) | 1974-11-04 |
| GB1456144A (en) | 1976-11-17 |
| FR2299318A1 (fr) | 1976-08-27 |
| LU69997A1 (es) | 1974-09-25 |
| IL44680A0 (en) | 1974-06-30 |
| DE2422068A1 (de) | 1974-11-28 |
| HU168312B (es) | 1976-03-28 |
| IE39549B1 (en) | 1978-11-08 |
| US4067978A (en) | 1978-01-10 |
| IN141295B (es) | 1977-02-12 |
| IL44680A (en) | 1977-03-31 |
| DD114267A5 (es) | 1975-07-20 |
| CS181264B2 (en) | 1978-03-31 |
| US4067976A (en) | 1978-01-10 |
| AU475779B2 (en) | 1976-09-02 |
| US4067977A (en) | 1978-01-10 |
| FR2299318B1 (es) | 1978-05-12 |
| FR2228475B1 (es) | 1978-07-28 |
| US4091227A (en) | 1978-05-23 |
| CA1041085A (en) | 1978-10-24 |
| US4007173A (en) | 1977-02-08 |
| AU6865674A (en) | 1975-11-06 |
| AR206315A1 (es) | 1976-07-15 |
| ZA742353B (en) | 1975-04-30 |
| GB1456145A (en) | 1976-11-17 |
| SE430506B (sv) | 1983-11-21 |
| FR2228475A1 (es) | 1974-12-06 |
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